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Repositioning of 3-(isoxazol-3-yl)thiazolidin-4-one-based compounds via Inverse Virtual Screening: discovery of new ERα inhibitors with in vitro activity in breast cancer models 基于3-(异恶唑-3-基)噻唑烷-4-酮类化合物的重定位:通过反向虚拟筛选发现具有体外活性的新型ERα抑制剂,在乳腺癌模型中表现出效果 Colarusso, Ester; De Vita, Simona; Boccia, Eleonora; Scala, Maria Carmina; Ferraro, Maria Grazia; Iazzetti, Federica; Piccolo, Marialuisa; Pellecchia, Sofia; Sala, Marina; Pepe, Giacomo; Campiglia, Pietro; Bifulco, Giuseppe; Irace, Carlo; Giordano, Assunta; Lauro, Gianluigi 分享 收藏
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Railway Ground Truth and Digital Map Based on GNSS and Multi-sensor Big-Data Acquisition 基于GNSS和多传感器大数据采集的铁路地面实况与数字地图 Neri, Alessandro; Vennarini, Alessia; Ruggeri, Agostino; Marais, Juliette; Tmazirte, Nourdine Ait; Crespillo, Omar Garcia; Grosch, Anja; Ramirez, Maria-Eva; Arroyo, Juan-Gabriel; Ciaffi, Massimiliano; Emmanuele, Giusy; Cataffo, Vittorio; Campo Cascallana, Ricardo; Molina Marinas, Daniel; Valentini, Alessandro; Neri, Stefano; Memmi, Fabrizio; Alvarez-Palencia, Ramiro Valdes; Lauro, Gianluigi; Natale, Pasquale 分享 收藏
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Unveiling New Triazoloquinoxaline-Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9 揭示靶向选择性降解ncBAF染色质重塑亚基BRD9的新型三氮唑喹啉类PROTACs的设计 Pierri, Martina; Bove, Guglielmo; Gazzillo, Erica; Colarusso, Ester; Scala, Francesca; Pepe, Giacomo; Terracciano, Stefania; Chini, Maria Giovanna; Simonelli, Nicla; Bruno, Ines; Nebbioso, Angela; Campiglia, Pietro; Bifulco, Giuseppe; Altucci, Lucia; Del Gaudio, Nunzio; Lauro, Gianluigi 分享 收藏
Chemical Profiling of Polyphenolic Fraction of Cannabis sativa L. vr. Kompolti Industrial Inflorescences: Insights into Cannabidiol Neuroprotective Effects in a Cellular Model of Parkinson's Disease 大麻(Cannabis sativa L. vr. Kompolti)工业花簇多酚组分的化学分析:对帕金森病细胞模型中大麻二酚神经保护作用的见解 Fantasma, Francesca; D'Urso, Gilda; Martella, Noemi; Capuano, Alessandra; Boccia, Eleonora; Samukha, Vadym; De Felice, Vincenzo; Saviano, Gabriella; Trombetta, Federico; Lauro, Gianluigi; Segatto, Marco; Chini, Maria Giovanna; Bifulco, Giuseppe; Casapullo, Agostino; Iorizzi, Maria 分享 收藏
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition Lauro, Gianluigi; Aliberti, Michela; De Nisco, Mauro; Pedatella, Silvana; Pepe, Giacomo; Basilicata, Manuela Giovanna; Chini, Maria Giovanna; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Saviano, Anella; Campiglia, Pietro; Bertamino, Alessia; Ostacolo, Carmine; Ciaglia, Tania; Manfra, Michele; Bifulco, Giuseppe 分享 收藏
Optimization of Steroid Photochemistry and Its Application in the Synthesis of 5,6-Dihydro-Ophiopogonol A 类固醇光化学的优化及其在5,6-二氢-芒柄花酚A合成中的应用 Maioli, Chiara; Lauro, Gianluigi; Sategna, Anna; Caprioglio, Diego; Amin, Hawraz Ibrahim M.; D'Auria, Maurizio; Imperio, Daniela; Bifulco, Giuseppe; Minassi, Alberto 分享 收藏