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收藏Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies通过体内外研究探索 lithospermic acid 作为人碳酸酐酶 VA 和胰腺脂肪酶抑制剂的潜力
Citriniti, Emanuele Liborio; Rocca, Roberta; Costa, Giosue; Sciacca, Claudia; Cardullo, Nunzio; Muccilli, Vera; Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T.; Alcaro, Stefano; Ortuso, Francesco
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收藏A Dynamic and Effective Peptide-Based Strategy for Promptly Addressing Emerging SARS-CoV-2 Variants of Concern一种动态有效的基于肽的策略,可迅速解决令人关注的新兴SARS-CoV-2变体
Murdocca, Michela; Romeo, Isabella; Citro, Gennaro; Latini, Andrea; Centofanti, Federica; Bugatti, Antonella; Caccuri, Francesca; Caruso, Arnaldo; Ortuso, Francesco; Alcaro, Stefano; Sangiuolo, Federica; Novelli, Giuseppe
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收藏Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches
Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura
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收藏8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin?s antidepressant profile: Synthesis, biological evaluation and docking studies
Matos, Maria J.; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez-Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda; Vina, Dolores
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收藏Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties基于色酮的类药物性能改善的单胺氧化酶B抑制剂的设计与合成
Reis, Joana; Fernandes, Carlos; Salem, Hoda; Maia, Marta; Tome, Claudia; Benfeito, Sofia; Teixeira, Jose; Oliveira, Paulo J.; Uriarte, Eugenio; Ortuso, Francesco; Alcaro, Stefano; Bagetta, Donatella; Cagide, Fernando; Borges, Fernanda
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收藏Chromene Derivatives as Selective TERRA G-Quadruplex RNA Binders with Antiproliferative Properties
Rocca, Roberta; Scionti, Francesca; Nadai, Matteo; Moraca, Federica; Maruca, Annalisa; Costa, Giosue; Catalano, Raffaella; Juli, Giada; Di Martino, Maria Teresa; Ortuso, Francesco; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco; Richter, Sara N.; Artese, Anna
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收藏Exploring New Scaffolds for the Dual Inhibition of HIV-1 RT Polymerase and Ribonuclease Associated Functions
Meleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Matyus, Peter; Maccioni, Elias
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收藏Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives
Meleddu, Rita; Deplano, Serenella; Maccioni, Elias; Ortuso, Francesco; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Angeli, Andrea; Angius, Rossella; Alcaro, Stefano; Supuran, Claudiu T.; Distinto, Simona
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收藏Natural Products Extracted from Fungal Species as New Potential Anti-Cancer Drugs: A Structure-Based Drug Repurposing Approach Targeting HDAC7
Maruca, Annalisa; Rocca, Roberta; Catalano, Raffaella; Mesiti, Francesco; Costa, Giosue; Lanzillotta, Delia; Salatino, Alessandro; Ortuso, Francesco; Trapasso, Francesco; Alcaro, Stefano; Artese, Anna
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收藏Multi-Targeting Bioactive Compounds Extracted from Essential Oils as Kinase Inhibitors
Maruca, Annalisa; Lanzillotta, Delia; Rocca, Roberta; Lupia, Antonio; Costa, Giosue; Catalano, Raffaella; Moraca, Federica; Gaudio, Eugenio; Ortuso, Francesco; Artese, Anna; Trapasso, Francesco; Alcaro, Stefano
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收藏Folding intermediate states of the parallel human telomeric G-quadruplex DNA explored using Well-Tempered Metadynamics
Rocca, Roberta; Palazzesi, Ferruccio; Amato, Jussara; Costa, Giosue; Ortuso, Francesco; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Alcaro, Stefano; Moraca, Federica; Artese, Anna
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收藏New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII
Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Caboni, Pierluigi; Angeli, Andrea; Melis, Claudia; Deplano, Serenella; Alcaro, Stefano; Ortuso, Francesco; Supuran, Claudiu T.; Maccioni, Elias
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