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Francesco Ortuso

università magna graecia di catanzaro

46H指数
189论文数
5.7K被引数
收录论文 108
发表时间
Identification of New Putative Autotaxin Inhibitors via Structure-Based Virtual Screening and Evaluation of Their Antiproliferative Properties Against Ovarian and Breast Cancer Cells通过基于结构的虚拟筛选鉴定新型假定的自泌素抑制剂,并评估其对卵巢癌和乳腺癌细胞的抗增殖特性
err2026-09-08
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PREAI
errAngelina Boccarelli; Adriana Coricello; Francesca Alessandra Ambrosio; Valentina Leo; Salvatore Mirabile; Rosaria Gitto; Modesto de Candia; Marco Catto; Francesco Ortuso; Cosimo D. Altomare; Stefano Alcaro
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Leveraging Natural Compounds for Pancreatic Lipase Inhibition via Virtual Screening通过虚拟筛选利用天然化合物抑制胰脂肪酶
err2026-03-03
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errEmanuele Liborio Citriniti; Roberta Rocca; Claudia Sciacca; Nunzio Cardullo; Vera Muccilli; Francesco Ortuso; Stefano Alcaro
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Design, synthesis, and biological activity of 2-aroylbenzofuran-3-ols and 2-aroylbenzofuran derivatives: A new route towards hMAO-B inhibition2-芳酰基苯并呋喃-3-醇和2-芳酰基苯并呋喃衍生物的设计、合成及生物活性:一种新型hMAO-B抑制剂的合成路线
err2025-07-18
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PREAI
errPaolo Guglielmi; Michele Coluccia; Guya Diletta Marconi; Francesco Ortuso; Francesca Procopio; Simone Carradori; Jacopo Pizzicannella; Francesca Arrighi; Anna Troiani; Chiara Salvitti; Fernanda Borges; Daniel Chavarria; Paola Chimenti; Daniela Secci; Francesca Diomede
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Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies通过体内外研究探索 lithospermic acid 作为人碳酸酐酶 VA 和胰腺脂肪酶抑制剂的潜力
err2025-04-21
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errCitriniti, Emanuele Liborio; Rocca, Roberta; Costa, Giosue; Sciacca, Claudia; Cardullo, Nunzio; Muccilli, Vera; Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T.; Alcaro, Stefano; Ortuso, Francesco
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A Dynamic and Effective Peptide-Based Strategy for Promptly Addressing Emerging SARS-CoV-2 Variants of Concern一种动态有效的基于肽的策略,可迅速解决令人关注的新兴SARS-CoV-2变体
err2024-07-04
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errMurdocca, Michela; Romeo, Isabella; Citro, Gennaro; Latini, Andrea; Centofanti, Federica; Bugatti, Antonella; Caccuri, Francesca; Caruso, Arnaldo; Ortuso, Francesco; Alcaro, Stefano; Sangiuolo, Federica; Novelli, Giuseppe
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MAATrica: a measure for assessing consistency and methods in medicinal and nutraceutical chemistry papers
err2024-07-01
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errPanzarella, Giulia; Gallo, Alessandro; Coecke, Sandra; Querci, Maddalena; Ortuso, Francesco; Hofmann-Apitius, Martin; Veltri, Pierangelo; Bajorath, Juergen; Alcaro, Stefano
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Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches
err2024-06-28
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PREAI
errLombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura
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8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin?s antidepressant profile: Synthesis, biological evaluation and docking studies
err2023-02-01
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errMatos, Maria J.; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez-Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda; Vina, Dolores
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Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties基于色酮的类药物性能改善的单胺氧化酶B抑制剂的设计与合成
err2022-09-01
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PREAI
errReis, Joana; Fernandes, Carlos; Salem, Hoda; Maia, Marta; Tome, Claudia; Benfeito, Sofia; Teixeira, Jose; Oliveira, Paulo J.; Uriarte, Eugenio; Ortuso, Francesco; Alcaro, Stefano; Bagetta, Donatella; Cagide, Fernando; Borges, Fernanda
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Chromene Derivatives as Selective TERRA G-Quadruplex RNA Binders with Antiproliferative Properties
err2022-04-28
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errRocca, Roberta; Scionti, Francesca; Nadai, Matteo; Moraca, Federica; Maruca, Annalisa; Costa, Giosue; Catalano, Raffaella; Juli, Giada; Di Martino, Maria Teresa; Ortuso, Francesco; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco; Richter, Sara N.; Artese, Anna
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Molecular Modeling and Experimental Evaluation of Non-Chiral Components of Bergamot Essential Oil with Inhibitory Activity against Human Monoamine Oxidases
err2022-04-11
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errCatalano, Raffaella; Procopio, Francesca; Chavarria, Daniel; Benfeito, Sofia; Alcaro, Stefano; Borges, Fernanda; Ortuso, Francesco
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Identification of SET/EED dual binders as innovative PRC2 inhibitors
err2022-03-29
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PREAI
errCatalano, Raffaella; Maruca, Annalisa; Rocca, Roberta; Tassone, Pierfrancesco; Panzarella, Giulia; Costa, Giosue; Ortuso, Francesco; Alcaro, Stefano
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Exploring New Scaffolds for the Dual Inhibition of HIV-1 RT Polymerase and Ribonuclease Associated Functions
err2021-06-23
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errMeleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Matyus, Peter; Maccioni, Elias
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Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives
err2021-02-18
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errMeleddu, Rita; Deplano, Serenella; Maccioni, Elias; Ortuso, Francesco; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Angeli, Andrea; Angius, Rossella; Alcaro, Stefano; Supuran, Claudiu T.; Distinto, Simona
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Natural Products Extracted from Fungal Species as New Potential Anti-Cancer Drugs: A Structure-Based Drug Repurposing Approach Targeting HDAC7
err2020-11-25
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errMaruca, Annalisa; Rocca, Roberta; Catalano, Raffaella; Mesiti, Francesco; Costa, Giosue; Lanzillotta, Delia; Salatino, Alessandro; Ortuso, Francesco; Trapasso, Francesco; Alcaro, Stefano; Artese, Anna
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Multi-Targeting Bioactive Compounds Extracted from Essential Oils as Kinase Inhibitors
err2020-05-06
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errMaruca, Annalisa; Lanzillotta, Delia; Rocca, Roberta; Lupia, Antonio; Costa, Giosue; Catalano, Raffaella; Moraca, Federica; Gaudio, Eugenio; Ortuso, Francesco; Artese, Anna; Trapasso, Francesco; Alcaro, Stefano
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Folding intermediate states of the parallel human telomeric G-quadruplex DNA explored using Well-Tempered Metadynamics
err2020-02-21
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errRocca, Roberta; Palazzesi, Ferruccio; Amato, Jussara; Costa, Giosue; Ortuso, Francesco; Pagano, Bruno; Randazzo, Antonio; Novellino, Ettore; Alcaro, Stefano; Moraca, Federica; Artese, Anna
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New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII
err2020-02-13
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errMeleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Caboni, Pierluigi; Angeli, Andrea; Melis, Claudia; Deplano, Serenella; Alcaro, Stefano; Ortuso, Francesco; Supuran, Claudiu T.; Maccioni, Elias
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