David Calabrese - Publications, H-index & Citations

David Calabrese

national institutes of health

23H指数

43论文数

3.5K被引数

收录论文 24

发表时间

Structure–Activity Relationship Studies toward the Optimization of First-In-Class Selective Small Molecule Agonists of the GPCR Relaxin/Insulin-like Family Peptide Receptor 2 结构-活性关系研究以优化首创新药选择性小分子激动剂，针对GPCR松弛素/胰岛素样家族肽受体2

Journal of Medicinal Chemistry

IF6.8

2026-02-19

PREAI

Kenneth J. Wilson; Maria Esteban-Lopez; Courtney Myhr; Wenjuan Ye; Curtis E. Moore; Noel Southall; Xin Hu; Abhijeet Kapoor; Konstantinos Afratis; Christopher A. LeClair; Samuel A. Kotler; Pranav Shah; Elias Carvalho Padilha; Yuhong Fang; David Calabrese; Emmett R. George; Amy Wang; Xin Xu; Elena Barnaeva; Marc Ferrer; Mark Henderson; Irina Agoulnik; Alexander I. Agoulnik; Juan J. Marugan

Investigating the NRAS 5′ UTR as a target for small molecules

CELL CHEMICAL BIOLOGY

IF7.2

2023-06-01

OAAI

Balaratnam, Sumirtha; Torrey, Zachary R.; Calabrese, David R.; Banco, Michael T.; Yazdani, Kamyar; Liang, Xiao; Fullenkamp, Christopher R.; Seshadri, Srinath; Holewinski, Ronald J.; Andresson, Thorkell; Ferre-D'Amare, Adrian R.; Incarnato, Danny; Schneekloth, John S., Jr.

Machine Learning Informs RNA-Binding Chemical Space

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2023-02-06

OAAI

Yazdani, Kamyar; Jordan, Deondre; Yang, Mo; Fullenkamp, Christopher R.; Calabrese, David R.; Boer, Robert; Hilimire, Thomas; Allen, Timothy E. H.; Khan, Rabia T.; Schneekloth Jr, John S.

Targeting a noncanonical, hairpin-containing G-quadruplex structure from the MYCN gene

NUCLEIC ACIDS RESEARCH

IF13.1

2021-07-21

OAAI

Yang, Mo; Carter, Sakereh; Parmar, Shaifaly; Bume, Desta D.; Calabrese, David R.; Liang, Xiao; Yazdani, Kamyar; Xu, Man; Liu, Zhihui; Thiele, Carol J.; Schneekloth, John S., Jr.

Evidence for ligandable sites in structured RNA throughout the Protein Data Bank

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2019-06-01

OAAI

Hewitt, William M.; Calabrese, David R.; Schneekloth, John S., Jr.

Chemical and structural studies provide a mechanistic basis for recognition of the MYC G-quadruplex

NATURE COMMUNICATIONS

IF15.7

2018-10-12

136

OAAI

Calabrese, David R.; Chen, Xiang; Leon, Elena C.; Gaikwad, Snehal M.; Phyo, Zaw; Hewitt, William M.; Alden, Stephanie; Hilimire, Thomas A.; He, Fahu; Michalowski, Aleksandra M.; Simmons, John K.; Saunders, Lindsey B.; Zhang, Shuling; Connors, Daniel; Walters, Kylie J.; Mock, Beverly A.; Schneekloth, John S., Jr.

Characterization of clinically used oral antiseptics as quadruplex-binding ligands

NUCLEIC ACIDS RESEARCH

IF13.1

2018-02-22

OAAI

Calabrese, David R.; Zlotkowski, Katherine; Alden, Stephanie; Hewitt, William M.; Connelly, Colleen M.; Wilson, Robert M.; Gaikwad, Snehal; Chen, Lu; Guha, Rajarshi; Thomas, Craig J.; Mock, Beverly A.; Schneekloth, John S., Jr.

Effective targeting of MYC expression with a novel nucleic acid binding (G4-quadruplex) small molecule coupled with HDAC inhibition synergizes to limit myeloma growth

CANCER RESEARCH

IF16.6

2017-07-01

PREAI

Gaikwad, Snehal M.; Calabrese, David R.; Leon, Elena C.; Simmons, John K.; Zhang, Shuling; Michalowski, Aleksandra; Gorjifard, Sayeh; Phyo, Zaw; Connors, Daniel; Schneekloth, John S.; Mock, Beverly A.

Automated microfluidic sorting of mammalian cells labeled with magnetic microparticles for those that efficiently express and secrete a protein of interest

BIOTECHNOLOGY AND BIOENGINEERING

IF3.6

2017-06-06

PREAI

Droz, Xuan; Harraghy, Niamh; Lancon, Etienne; Le Fourn, Valerie; Calabrese, David; Colombet, Thierry; Liechti, Pascal; Rida, Amar; Girod, Pierre-Alain; Mermod, Nicolas

Role of Backbone Chemistry and Monomer Sequence in Amphiphilic Oligopeptide- and Oligopeptoid-Functionalized PDMS- and PEO-Based Block Copolymers for Marine Antifouling and Fouling Release Coatings

MACROMOLECULES

IF5.2

2017-03-23

PREAI

Patterson, Anastasia L.; Wenning, Brandon; Rizis, Georgios; Calabrese, David R.; Finlay, John A.; Franco, Sofia C.; Zuckermann, Ronald N.; Clare, Anthony S.; Kramer, Edward J.; Ober, Christopher K.; Segalman, Rachel A.

Selective inhibition of MYC expression by a small molecule G-quadruplex stabilizer

CANCER RESEARCH

IF16.6

2016-07-15

PREAI

Leon, Elena C.; Simmons, John K.; Calabrese, David; DuBois, Wendy; Felsenstein, Kenneth; Saunders, Lindsey B.; Zhang, Shuling; Michalowski, Aleksandra; Gonzalez, Frank; Mock, Beverly A.; Schneekloth, John S.

Small Molecule Microarrays Enable the Identification of a Selective, Quadruplex-Binding Inhibitor of MYC Expression

ACS CHEMICAL BIOLOGY

IF3.8

2015-11-06

127

OAAI

Felsenstein, Kenneth M.; Saunders, Lindsey B.; Simmons, John K.; Leon, Elena; Calabrese, David R.; Zhang, Shuling; Michalowski, Aleksandra; Gareiss, Peter; Mock, Beverly A.; Schneekloth, John S., Jr.

High-Quality Streamable Free-Viewpoint Video

ACM TRANSACTIONS ON GRAPHICS

IF9.5

2015-07-27

435

PREAI

Collet, Alvaro; Chuang, Ming; Sweeney, Pat; Gillett, Don; Evseev, Dennis; Calabrese, David; Hoppe, Hugues; Kirk, Adam; Sullivan, Steve

Epigenetic regulatory elements: Recent advances in understanding their mode of action and use for recombinant protein production in mammalian cells

BIOTECHNOLOGY JOURNAL

IF3.1

2015-06-23

PREAI

Harraghy, Niamh; Calabrese, David; Fisch, Igor; Girod, Pierre-Alain; LeFourn, Valerie; Regamey, Alexandre; Mermod, Nicolas

Amphiphilic oligopeptides grafted to PDMS-based diblock copolymers for use in antifouling and fouling release coatings

POLYMERS FOR ADVANCED TECHNOLOGIES

IF3.4

2015-04-30

PREAI

Calabrese, David R.; Wenning, Brandon; Finlay, John A.; Callow, Maureen E.; Callow, James A.; Fischer, Daniel; Ober, Christopher K.

Efficient Synthesis of Thiopyrans Using a Sulfur-Enabled Anionic Cascade 使用硫使能的阴离子级联有效合成硫代吡喃

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2012-01-10

PREAI

Li, Fang; Calabrese, David; Brichacek, Matthew; Lin, Ivy; Njardarson, Jon T.

High-level transgene expression by homologous recombination-mediated gene transfer

NUCLEIC ACIDS RESEARCH

IF13.1

2011-06-06

OAAI

Grandjean, Melanie; Girod, Pierre-Alain; Calabrese, David; Kostyrko, Kaja; Wicht, Marianne; Yerly, Florence; Mazza, Christian; Beckmann, Jacques S.; Martinet, Danielle; Mermod, Nicolas

Gain of Function Mutations in CgPDR1 of Candida glabrata Not Only Mediate Antifungal Resistance but Also Enhance Virulence

PLOS PATHOGENS

IF4.9

2009-01-16

258

OAAI

Ferrari, Selene; Ischer, Francoise; Calabrese, David; Posteraro, Brunella; Sanguinetti, Maurizio; Fadda, Giovanni; Rohde, Bettina; Bauser, Christopher; Bader, Oliver; Sanglard, Dominique

Syntheses of α- and β-C-Glucopyranosyl Serines from a Common Intermediate

ORGANIC LETTERS

IF5

2008-09-27

PREAI

Nolen, Ernest G.; Donahue, Laurence A.; Greaves, Rebecca; Daly, Trevor A.; Calabrese, David R.

Genome-wide prediction of matrix attachment regions that increase gene expression in mammalian cells

NATURE METHODS

IF32.1

2007-08-05

158

PREAI

Girod, Pierre-Alain; Nguyen, Duc-Quang; Calabrese, David; Puttini, Stefania; Grandjean, Melanie; Martinet, Danielle; Regamey, Alexandre; Saugy, Damien; Beckmann, Jacques S.; Bucher, Philipp; Mermod, Nicolas

研究方向