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收藏Discovery of Novel Potent and Safe Immunoproteasome Inhibitors with Bridged Ring for Anti-Inflammatory Therapy发现具有桥环结构的强效且安全的免疫蛋白酶体抑制剂,用于抗炎治疗
Wu, Jian; Cai, Shi; Su, Jincai; Ji, Xiaojun; Zhou, Qiuhua; Chen, Zehong; Fan, Yiqing; Li, Xuefei; Liu, Jiang; Dong, Wanting; Ma, Changyou; Xu, Dan; Qian, Hai
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收藏Structure optimization of natural product piperine to obtain novel and potent analogs with anti-inflammation pain and urate-lowering effect天然产物piperine的结构优化,以获得具有抗炎、镇痛和降尿酸作用的全新且高效的类似物
Liu, Chunxia; Wang, Wenxin; Miao, Ruoyang; Chen, Haoyang; Wang, Ning; Cheng, Weiyan; Zheng, Fengxin; Li, Zheng; Pang, Jianxin; Qian, Hai; Tian, Xin
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收藏Design, synthesis and biological activity of novel pyrimidine piperazine ureas as μ-opioid and TRPV1 dual-target ligands for pain management新型嘧啶哌嗪脲类化合物的设计、合成及其作为μ-阿片和TRPV1双靶点配体在疼痛管理中的生物活性
Wang, Yusui; Liu, Shuyu; Zhang, Zhikang; Ma, Yunmeng; Qin, Kexin; Du, Jiahao; Wang, Yu; Wang, Bingxin; Qian, Hai; Pang, Xiaobin; Zhao, Fenqin; Du, Guanhua; Yan, Lin
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收藏Design, Synthesis, and Biological Assessment of Novel Aminobenzidazole Agonists Targeting the Stimulator of Interferon Genes (STING) Receptor Signaling Pathway for Oncology Immunotherapy
Fan, Yiqing; Zeng, Zeqi; Mo, Jiaxian; Wang, Zike; Jiang, Hongyu; Liu, Juanjuan; Qian, Hai; Shi, Wei
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收藏Highly Potent and Intestine Specific P-Glycoprotein Inhibitor to Enable Oral Delivery of Taxol
Zhou, Xianjing; Zhang, Ping; Yang, Yuyan; Shi, Wei; Liu, Lei; Lai, Zhencheng; Zhang, Xing; Pan, Peichen; Li, Lan; Du, Juan; Qian, Hai; Cui, Sunliang
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收藏Development of Peptide Paratope Mimics Derived from the Anti-ROR1 Antibody and Long-Acting Peptide-Drug Conjugates for Targeted Cancer Therapy
Zhang, Yang; Fan, Yiqing; Liu, Shuyu; Guan, Yonghui; Wan, Jiale; Ren, Qiang; Wang, Jialing; Zhong, Li; Hu, Zhipeng; Shi, Wei; Qian, Hai
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收藏Design, synthesis and bioactivity evaluation of novel fusion peptides and their CPT conjugates inducing effective anti-tumor responses on HER2 positive tumors
Zhou, Jiaqi; Xie, Zhancheng; Wang, Jialing; Zeng, Zeqi; Hu, Zhipeng; Zhong, Li; Yang, Qimeng; Shi, Wei; Qian, Hai
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