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Bruno Melillo

Scripps Research

35H指数
116论文数
3.4K被引数
收录论文 59
发表时间
Tryptoline stereoprobe elaboration identifies inhibitors of the GRPEL1–HSPA9 complex色普利宁立体探针的精制鉴定了GRPEL1–HSPA9复合物的抑制剂
err2026-10-16
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errOAAI
errRachel E. Hayward; Raymond F. Berkeley; Zijian Gao; Maximilian Garhammer; Marc A. Morizono; Evert Njomen; Haoxin Li; Kristen E. DeMeester; Victor Cociorva; Mark A. Herzik; F. Ulrich Hartl; Bruno Melillo; Benjamin F. Cravatt
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An enantioselective covalent inhibitor of BAX confers cytoprotection in vivoBAX的手性选择性共价抑制剂可赋予体内细胞保护作用
err2026-08-28
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errOAAI
errPeiwen Shi; Bruno Melillo; Matthew W. McHenry; Christina M. Camara; Ka Yang; Evert Njomen; Marina Godes; Maria F. Pazyra-Murphy; Mary Rose Branch; Bethany Tesar; Rosalind A. Segal; Lee L. Rubin; Michael D. Cameron; Gregory H. Bird; Thomas E. Wales; Steven P. Gygi; Benjamin F. Cravatt; Loren D. Walensky
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High-throughput ligand diversification to discover chemical inducers of proximity高通量配体多样化以发现邻近性的化学诱导剂
err2026-02-16
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errOAAI
errJames B. Shaum; Miquel Muñoz i Ordoño; Erica A. Steen; Daniela V. Wenge; Hakyung Cheong; Jordan Janowski; Moritz Hunkeler; Eric M. Bilotta; Zoe J. Rutter; Paige A. Barta; Abby M. Thornhill; Natalia Milosevich; Lauren M. Hargis; Timothy R. Bishop; Trever R. Carter; Bryce da Camara; Matthias Hinterndorfer; Lucas Dada; Wen-Ji He; Fabian Offensperger; Hirotake Furihata; Sydney R. Schweber; Charlie Hatton; Yanhe Wen; Benjamin F. Cravatt; Keary M. Engle; Katherine A. Donovan; Bruno Melillo; Seiya Kitamura; Alessio Ciulli; Scott A. Armstrong; Eric S. Fischer; Georg E. Winter; Michael A. Erb
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Correction to “Improved Bicyclic Pyrrolidine Analogues Inhibit Toxoplasma gondii Growth In Vitro and Cure Infection In Vivo”
err2026-02-05
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PREAI
errTaher Uddin; Han Xie; Payal Mittal; Chloe Ence; Anil K. Gupta; Shrushti Patil; Christy Cho; Satavisha Banerjee; Amit Sharma; Bruno Melillo; Arnab K. Chatterjee; L. David Sibley
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Targeting extrachromosomal DNA in human cancers靶向人类癌症中的染色体外DNA
err2026-02-03
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PREAI
errIvy Tsz-Lo Wong; Hyerim Yi; Bruno Melillo; Benjamin F. Cravatt; Howard Y. Chang; Paul S. Mischel
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Cysteine Reactivity Profiling Identifies Host Regulators of Mycobacterium tuberculosis Replication in Human Macrophages
err2026-01-27
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PREAI
errJohn K. Neff; Kristen E. DeMeester; Paola K. Párraga Solórzano; Radu M. Suciu; Melissa M. Dix; Gabriel Simon; Max A. Gianakopoulos; Bruno Melillo; Benjamin F. Cravatt; Michael U. Shiloh
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Structural and mechanistic analysis of covalent ligands targeting the RNA-binding protein NONO共价配体靶向RNA结合蛋白NONO的结构与机制分析
err2026-01-13
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errGarrett L. Lindsey; Thomas K. Hockley; Alejandro Villa Gomez; Andrew C. Marshall; William R. Brothers; Colin T. Finney; Jacob Gross; Archa H. Fox; Gene W. Yeo; Bruno Melillo; Charles S. Bond; Benjamin F. Cravatt
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Complexoform-restricted covalent TRMT112 ligands that allosterically agonize METTL5Complexoform限制性共价TRMT112配体,能够别构激活METTL5
err2026-01-08
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errF. Wieland Goetzke; Steffen M. Bernard; Cheng-Wei Ju; Jonathan Pollock; Kristen E. DeMeester; Jacob Gross; Gabriel M. Simon; Chuan He; Bruno Melillo; Benjamin F. Cravatt
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Proteomic Ligandability Maps of Phosphorus(V) Stereoprobes Identify Covalent TLCD1 Inhibitors磷(V)立体探针的蛋白质组配体可及性图谱鉴定了共价TLCD1抑制剂
err2025-04-23
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PREAI
errSharma, Hayden A.; Bielecki, Michael; Holm, Meredith A.; Thompson, Ty M.; Yin, Yue; Cravatt, Jacob B.; Ware, Timothy B.; Reed, Alex; Nassir, Molhm; Ewing, Tamara El-Hayek; Melillo, Bruno; Bazan, J. Fernando; Baran, Phil S.
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SF3B1 thermostability as an assay for splicing inhibitor interactions
err2025-02-01
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errAmorello, Angela N.; Reddy, Guddeti Chandrashekar; Melillo, Bruno; Cravatt, Benjamin F.; Ghosh, Arun K.; Jurica, Melissa S.
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Covalent targeting of splicing in T cells
err2025-01-01
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PREAI
errScott, Kevin A.; Kojima, Hiroyuki; Ropek, Nathalie; Warren, Charles D.; Zhang, Tiffany L.; Hogg, Simon J.; Sanford, Henry; Webster, Caroline; Zhang, Xiaoyu; Rahman, Jahan; Melillo, Bruno; Cravatt, Benjamin F.; Lyu, Jiankun; Abdel-Wahab, Omar; Vinogradova, Ekaterina V.
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Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes
err2024-12-01
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errOAAI
errOgasawara, Daisuke; Konrad, David B.; Tan, Zher Yin; Carey, Kimberly L.; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever R.; DeMeester, Kristen E.; Njomen, Evert; Schreiber, Stuart L.; Xavier, Ramnik J.; Melillo, Bruno; Cravatt, Benjamin F.
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Redirecting the pioneering function of FOXA1 with covalent small molecules
err2024-11-01
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PREAI
errWon, Sang Joon; Zhang, Yuxiang; Reinhardt, Christopher J.; Hargis, Lauren M.; MacRae, Nicole S.; DeMeester, Kristen E.; Njomen, Evert; Remsberg, Jarrett R.; Melillo, Bruno; Cravatt, Benjamin F.; Erb, Michael A.
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An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes
err2024-09-18
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PREAI
errZhang, Yuanjin; Liu, Zhonglin; Hirschi, Marscha; Brodsky, Oleg; Johnson, Eric; Won, Sang Joon; Nagata, Asako; Bezwada, Divya; Petroski, Matthew D.; Majmudar, Jaimeen D.; Niessen, Sherry; Vanarsdale, Todd; Gilbert, Adam M.; Hayward, Matthew M.; Stewart, Al E.; Nager, Andrew R.; Melillo, Bruno; Cravatt, Benjamin F.
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Bicyclic Pyrrolidine Inhibitors of Toxoplasma gondii Phenylalanine t-RNA Synthetase with Antiparasitic Potency In Vitro and Brain Exposure
err2024-05-14
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PREAI
errEnce, Chloe C.; Uddin, Taher; Borrel, Julien; Mittal, Payal; Xie, Han; Zoller, Jochen; Sharma, Amit; Comer, Eamon; Schreiber, Stuart L.; Melillo, Bruno; Sibley, L. David; Chatterjee, Arnab K.
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Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders
err2024-04-03
err6
PREAI
errLiu, Zhonglin; Remsberg, Jarrett R.; Li, Haoxin; Njomen, Evert; Demeester, Kristen E.; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E.; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M.; Schreiber, Stuart L.; Melillo, Bruno; Cravatt, Benjamin F.
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Covalent Targeting As a Common Mechanism for Inhibiting NLRP3 Inflammasome Assembly
err2024-01-10
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errOAAI
errStanton, Caroline; Sun, Jie; Nutsch, Kayla; Rosarda, Jessica D.; Nguyen, Thu; Li-Ma, Chloris; Njomen, Evert; Melillo, Bruno; Kutseikin, Sergei; Saez, Enrique; Cravatt, Benjamin F.; Teijaro, John R.; Wiseman, R. Luke; Bollong, Michael J.
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Genetic crosses within and between species of Cryptosporidium
err2023-12-26
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errShaw, Sebastian; Cohn, Ian S.; Baptista, Rodrigo P.; Xia, Guoqin; Melillo, Bruno; Agyabeng-Dadzie, Fiifi; Kissinger, Jessica C.; Striepen, Boris
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