未登录Virtual screening-guided repurposing of fluorescent probes to detect EGFR expression in renal cells虚拟筛选指导的荧光探针再利用以检测肾细胞中EGFR表达
Graziano, Giovanni; Trisciuzzi, Daniela; Contino, Marialessandra; Stasi, Alessandra; Laghezza, Antonio; Cimmarusti, Maria Teresa; Campioni, Monica; Mammone, Mariachiara; Fanizzi, Annalisa; Degennaro, Pasquale; Mastrofilippo, Nicola; Fiorentino, Marco; Pontrelli, Paola; Stefanachi, Angela; Colabufo, Nicola Antonio; Gesualdo, Loreto; Nicolotti, Orazio
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收藏4,5-Diazafluorene derivatives and their silver(I) complexes: Synthesis and biological evaluation as antiproliferative agents4,5-二氮芴衍生物及其银(I)配合物:合成与作为抗增殖剂的生物活性评价
Sandin-Mazzondo, Leonardo; Trejo, Angela; Mammone, Mariachiara; Perrone, Maria Grazia; Contino, Marialessandra; Rico-Martinez, Sandra; Alonso, Concepcion; Bartolome, Camino
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收藏Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold
Braconi, Laura; Riganti, Chiara; Parenti, Astrid; Cecchi, Marta; Nocentini, Alessio; Bartolucci, Gianluca; Menicatti, Marta; Contino, Marialessandra; Colabufo, Nicola Antonio; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T.; Teodori, Elisabetta
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收藏N-Adamantyl-1-alkyl-4-oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as Fluorescent Probes to Detect Microglia Activation through the Imaging of Cannabinoid Receptor Subtype 2 (CB2R)
Intranuovo, Francesca; Majellaro, Maria; Mastropasqua, Francesco; Delre, Pietro; Abatematteo, Francesca Serena; Mangiatordi, Giuseppe Felice; Stefanachi, Angela; Brea, Jose; Loza, Maria Isabel; Riganti, Chiara; Ligresti, Alessia; Kumar, Poulami; Esposito, Daniela; Cristino, Luigia; Nicois, Alessandro; Gonzalez, Lucia; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Sotelo, Eddy; Abate, Carmen; Contino, Marialessandra
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收藏Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment
Miciaccia, Morena; Rizzo, Francesca; Centonze, Antonella; Cavallaro, Gianfranco; Contino, Marialessandra; Armenise, Domenico; Baldelli, Olga Maria; Solidoro, Roberta; Ferorelli, Savina; Scarcia, Pasquale; Agrimi, Gennaro; Zingales, Veronica; Cimetta, Elisa; Ronsisvalle, Simone; Sipala, Federica Maria; Polosa, Paola Loguercio; Fortuna, Cosimo Gianluca; Perrone, Maria Grazia; Scilimati, Antonio
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收藏Development of potent isoflavone-based formyl peptide receptor 1 (FPR1) antagonists and their effects in gastric cancer cell models
Francavilla, Fabio; Sarcina, Federica; Schepetkin, Igor A.; Kirpotina, Lilya N.; Contino, Marialessandra; Schirizzi, Annalisa; De Leonardis, Giampiero; Khlebnikov, Andrei I.; D'Alessandro, Rosalba; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello
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收藏Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers
Braconi, Laura; Dei, Silvia; Contino, Marialessandra; Riganti, Chiara; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Guglielmo, Stefano; Teodori, Elisabetta
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收藏Development of Fluorescent 4-[4-(3H-Spiro[isobenzofuran-1,4?- piperidin]-1?-yl)butyl]indolyl Derivatives as High-Affinity Probes to Enable the Study of ? Receptors via Fluorescence-Based Techniques
Abatematteo, Francesca Serena; Majellaro, Maria; Montsch, Bianca; Prieto-Diaz, Ruben; Niso, Mauro; Contino, Marialessandra; Stefanachi, Angela; Riganti, Chiara; Mangiatordi, Giuseppe Felice; Delre, Pietro; Heffeter, Petra; Sotelo, Eddy; Abate, Carmen
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收藏The multiple combination of Paclitaxel, Ramucirumab and Elacridar reverses the paclitaxel-mediated resistance in gastric cancer cell lines
Schirizzi, Annalisa; Contino, Marialessandra; Carrieri, Livianna; Riganti, Chiara; De Leonardis, Giampiero; Scavo, Maria Principia; Perrone, Maria Grazia; Miciaccia, Morena; Kopecka, Joanna; Refolo, Maria Grazia; Lotesoriere, Claudio; Depalo, Nicoletta; Rizzi, Federica; Giannelli, Gianluigi; Messa, Caterina; D'Alessandro, Rosalba
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收藏N-adamantyl-anthranil amide derivatives: New selective ligands for the cannabinoid receptor subtype 2 (CB2R)N-金刚烷基-邻氨基苯甲酰胺衍生物: 大麻素受体亚型2 (CB2R) 的新选择性配体
Graziano, Giovanni; Delre, Pietro; Carofiglio, Francesca; Brea, Jose; Ligresti, Alessia; Kostrzewa, Magdalena; Riganti, Chiara; Gioe-Gallo, Claudia; Majellaro, Maria; Nicolotti, Orazio; Colabufo, Nicola Antonio; Abate, Carmen; Loza, Maria Isabel; Sotelo, Eddy; Mangiatordi, Giuseppe Felice; Contino, Marialessandra; Stefanachi, Angela; Leonetti, Francesco
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收藏Development of N-(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase
Intranuovo, Francesca; Brunetti, Leonardo; DelRe, Pietro; Mangiatordi, Giuseppe Felice; Stefanachi, Angela; Laghezza, Antonio; Niso, Mauro; Leonetti, Francesco; Loiodice, Fulvio; Ligresti, Alessia; Kostrzewa, Magdalena; Brea, Jose; Loza, Maria Isabel; Sotelo, Eddy; Saviano, Michele; Colabufo, Nicola Antonio; Riganti, Chiara; Abate, Carmen; Contino, Marialessandra
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