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Theodore M. Kamenecka

State University System of Florida

52H指数
262论文数
1.1W被引数
收录论文 85
发表时间
Myeloid deficiency of RORα exacerbates lipid dysregulation and laser-induced choroidal neovascularizationRORα的髓系缺陷加剧脂质失调和激光诱导的脉络膜新生血管形成
err2026-09-25
err0
errOAAI
errNeetu Kushwah; Chi-Hsiu Liu; Kiran Bora; Meenakshi Maurya; Madeline C. Pavlovich; Zhongjie Fu; Theodore M. Kamenecka; Ye Sun; Laura A. Solt; Jing Chen
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Structural determinants of non-covalent PPARγ inverse agonism and their therapeutic implications非共价PPARγ反向激动作用的结构决定因素及其治疗意义
err2025-12-19
err0
errOAAI
errKuang-Ting Kuo; Bilel Bdiri; Yuanjun He; Ruben D. Garcia-Ordonez; Daniel P. McDougal; Claudia Ruiz; Mi Ra Chang; Michael D. Cameron; John B. Bruning; Theodore M. Kamenecka; Patrick R. Griffin
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The Endo-GeneScreen platform identifies drug-like probes that regulate endogenous protein levels within physiological contextsEndo-GeneScreen平台识别在生理背景下调节内源性蛋白质水平的类药探针
err2025-12-09
err0
errOAAI
errPreston Samowitz; Laszlo Radnai; Thomas Vaissiere; Sheldon D. Michaelson; Camilo Rojas; Ryan Mitchell; Murat Kilinc; Austin Edwards; Justin Shumate; Richard Hawkins; Virneliz Fernandez-Vega; Timothy P. Spicer; Louis Scampavia; Theodore Kamenecka; Courtney A. Miller; Gavin Rumbaugh
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MT-125 Inhibits Non-Muscle Myosin IIA and IIB and Prolongs Survival in GlioblastomaMT-125 抑制非肌性肌球蛋白IIA和IIB并延长胶质母细胞瘤患者的生存期
err2025-11-01
err0
errOAAI
errRosenfeld, Steven; Kenchappa, Rajappa; Radnai, Laszlo; Zarco, Natanael; Canoll, Peter; Dovas, Athanassios; Rumbaugh, Gavin; Griffin, Patrick; Kamenecka, Theodore; Miller, Courtney
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Development of clinically viable non-muscle myosin II small molecule inhibitors开发临床可行的非肌球蛋白II小分子抑制剂
errCell
IF42.5
err2025-07-01
err0
PREAI
errLaszlo Radnai; Erica J. Young; Carlos Kikuti; Katalin Toth; Minghai Zhou; Madalyn Hafenbreidel; Rebecca F. Stremel; Li Lin; Paolo Pasetto; Xiaomin Jin; Aagam Patel; Michael Conlon; Sherri B. Briggs; Leïla Heidsieck; H. Lee Sweeney; James Sellers; Teresa Krieger-Burke; William H. Martin; Jay Sisco; Steven Young; Paul Pearson; Gavin Rumbaugh; Gian Luca Araldi; Steven K. Duddy; Michael D. Cameron; Matthew Surman; Anne Houdusse; Patrick R. Griffin; Theodore M. Kamenecka; Courtney A. Miller
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MT-125 inhibits non-muscle myosin IIA and IIB and prolongs survival in glioblastomaMT-125抑制非肌肉肌球蛋白IIA和IIB并延长胶质母细胞瘤患者的生存期
errCell
IF42.5
err2025-06-10
err0
errOAAI
errRajappa S. Kenchappa; Laszlo Radnai; Erica J. Young; Natanael Zarco; Li Lin; Athanassios Dovas; Christian T. Meyer; Ashley Haddock; Alice Hall; Katalin Toth; Peter Canoll; Naveen K.H. Nagaiah; Gavin Rumbaugh; Michael D. Cameron; Theodore M. Kamenecka; Patrick R. Griffin; Courtney A. Miller; Steven S. Rosenfeld
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Targeting the Glucocorticoid Receptor Solvent Channel for Modulation of Activity靶向糖皮质激素受体溶剂通道以调节活性
err2025-04-21
err0
PREAI
errKobylski, Robin R.; Koenig, Marcel; Nwachukwu, Jerome C.; Kamenecka, Theodore M.; Solt, Laura A.; Nettles, Kendall W.
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Advancing clinical response against glioblastoma: Evaluating SHP1705 CRY2 activator efficacy in preclinical models and safety in phase I trials推进胶质母细胞瘤的临床反应:评估SHP1705 CRY2激活剂在临床前模型中的疗效和I期试验中的安全性
err2025-04-01
err1
errOAAI
errChan, Priscilla; Nagai, Yoshiko; Wu, Qiulian; Hovsepyan, Anahit; Mkhitaryan, Seda; Wang, Jiarui; Karapetyan, Gevorg; Kamenecka, Theodore; Solt, Laura A.; Cope, Jamie; Moats, Rex A.; Hirota, Tsuyoshi; Rich, Jeremy N.; Kay, Steve A.
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Small molecules targeting selective PCK1 and PGC-1α lysine acetylation cause anti-diabetic action through increased lactate oxidation (vol 31, pg 1772, 2024)
err2025-02-01
err0
PREAI
errMutlu, Beste; Sharabi, Kfir; Sohn, Jee Hyung; Yuan, Bo; Latorre-Muro, Pedro; Qin, Xin; Yook, Jin-Seon; Lin, Hua; Yu, Deyang; Camporez, Joao Paulo G.; Kajimura, Shingo; Shulman, Gerald I.; Hui, Sheng; Kamenecka, Theodore M.; Griffin, Patrick R.; Puigserver, Pere
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MT-125 INHIBITS NON-MUSCLE MYOSIN IIA AND IIB, SYNERGIZES WITH ONCOGENIC KINASE INHIBITORS, AND PROLONGS SURVIVAL IN GLIOBLASTOMA
err2024-11-11
err0
PREAI
errRosenfeld, Steven; Kenchappa, Rajappa; Radnai, Laszlo; Zarco, Natanael; Dovas, Athanassios; Haddock, Ashley; Canoll, Peter; Rumbaugh, Gavin; Griffin, Patrick; Kamenecka, Theodore; Miller, Courtney
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Interrogating circadian clock compounds as an adjuvant to chemoradiation against GBM询问昼夜节律钟化合物作为针对GBM的化学辐射的佐剂
err2024-03-22
err0
PREAI
errChan, Priscilla; Wu, Qiulian; Hovsepyan, Anahit; Mkhitaryan, Seda; Karapetyan, Gevorg; Shah, Khalid; Wakimoto, Hiroaki; Kamenecka, Theodore; Solt, Laura A.; Cope, Jamie; Hirota, Tsuyoshi; Moats, Rex A.; Rich, Jeremy N.; Kay, Steve A.
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Senotherapeutic drug treatment ameliorates chemotherapy-induced cachexia
err2024-01-23
err13
errOAAI
errEnglund, Davis A.; Jolliffe, Alyssa M.; Hanson, Gabriel J.; Aversa, Zaira; Zhang, Xu; Jiang, Xinyi; White, Thomas A.; Zhang, Lei; Monroe, David G.; Robbins, Paul D.; Niedernhofer, Laura J.; Kamenecka, Theodore M.; Khosla, Sundeep; LeBrasseur, Nathan K.
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Structure-Activity Relationship and Biological Investigation of a REV-ERBα-Selective Agonist SR-29065 (34) for Autoimmune Disorders
err2023-10-27
err0
PREAI
errHe, Yuanjun; Zhu, Di; Greenman, Kevin; Ruiz, Claudia; Shang, Jinsai; Lu, Qun; Kojetin, Douglas J.; Drakas, Robert; Cameron, Michael D.; Lizarzaburu, Mike; Solt, Laura A.; Kamenecka, Theodore M.
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PPARγ Corepression Involves Alternate Ligand Conformation and Inflation of H12 Ensembles
err2023-05-05
err3
PREAI
errFrkic, Rebecca L.; Pederick, Jordan L.; Horsfall, Aimee J.; Jovcevski, Blagojce; Crame, Elise E.; Kowalczyk, Wioleta; Pukala, Tara L.; Chang, Mi Ra; Zheng, Jie; Blayo, Anne-Laure; Abell, Andrew D.; Kamenecka, Theodore M.; Harbort, Joshua S.; Harmer, Jeffrey R.; Griffin, Patrick R.; Bruning, John B.
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Small molecule circadian clock compounds display therapeutic potential in targeting glioblastoma stem cells小分子生物钟化合物在靶向胶质母细胞瘤干细胞方面显示出治疗潜力
err2023-04-04
err0
PREAI
errChan, Priscilla; Wu, Lian; Hovsepyan, Anahit; Mkhitaryan, Seda; Karapetyan, Gevorg; Shah, Khalid; Wakimoto, Hiroaki; Kamenecka, Theodore; Solt, Laura A.; Cope, Jamie; Moats, Rex A.; Hirota, Tsuyoshi; Rich, Jeremy N.; Kay, Steve A.
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Defining the transcriptional regulation of NR2F6 in CD4+ T helper cell responses
err2022-05-01
err0
PREAI
errWilson, Adrianna N.; Campbell, Sean; Lu, Qun; Mosure, Sarah A.; He, Yuanjun; Bdiri, Bilel; Kamenecka, Theodore M.; Solt, Laura A.
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Novel small molecule inhibition of IKK/NF-κB activation reduces markers of senescence and improves healthspan in mouse models of aging
err2021-11-03
err33
errOAAI
errZhang, Lei; Zhao, Jing; Mu, Xiaodong; McGowan, Sara J.; Angelini, Luise; O'Kelly, Ryan D.; Yousefzadeh, Matthew J.; Sakamoto, Ayumi; Aversa, Zaira; LeBrasseur, Nathan K.; Suh, Yousin; Huard, Johnny; Kamenecka, Theodore M.; Niedernhofer, Laura J.; Robbins, Paul D.
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Discovery of Selective Inhibitors for In Vitro and In Vivo Interrogation of Skeletal Myosin II
err2021-09-24
err4
PREAI
errRadnai, Laszlo; Surman, Matthew; Hafenbreidel, Madalyn; Young, Erica J.; Stremel, Rebecca F.; Lin, Li; Bdiri, Bilel; Pasetto, Paolo; Jin, Xiaomin; Geedy, Mackenzie; Partridge, Joni-Rae; Patel, Aagam; Conlon, Michael; Sellers, James R.; Cameron, Michael D.; Rumbaugh, Gavin; Griffin, Patrick R.; Kamenecka, Theodore M.; Miller, Courtney A.
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Assessment of NR4A Ligands That Directly Bind and Modulate the Orphan Nuclear Receptor Nurr1 (vol 63, pg 15639, 2020)
err2021-04-12
err0
PREAI
errMunoz-Tello, Paola; Lin, Hua; Khan, Pasha; de Vera, Ian Mitchelle S.; Kamenecka, Theodore M.; Kojetin, Douglas J.
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