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收藏Anticancer Activities of Novel Nicotinamide Phosphoribosyltransferase Inhibitors in Hematological Malignancies新型烟酰胺磷酸核糖转移酶抑制剂在血液系统恶性肿瘤中的抗癌活性
Biniecka, Paulina; Matsumoto, Saki; Belotti, Axel; Joussot, Jessie; Bai, Jian Fei; Majjigapu, Somi Reddy; Thoueille, Paul; Spaggiari, Dany; Desfontaine, Vincent; Piacente, Francesco; Bruzzone, Santina; Cea, Michele; Decosterd, Laurent A. A.; Vogel, Pierre; Nencioni, Alessio; Duchosal, Michel A. A.; Nahimana, Aimable
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收藏Identification of new FK866 analogues with potent anticancer activity against pancreatic cancer
Bai, Jian-Fei; Majjigapu, Somi Reddy; Sordat, Bernard; Poty, Sophie; Vogel, Pierre; Elias-Rodriguez, Pilar; Moreno-Vargas, Antonio J.; Carmona, Ana T.; Caffa, Irene; Ghanem, Moustafa; Khalifa, Amr; Monacelli, Fiammetta; Cea, Michele; Robina, Inmaculada; Gajate, Consuelo; Mollinedo, Faustino; Bellotti, Axel; Nahimana, Aimable; Duchosal, Michel; Nencioni, Alessio
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收藏Structure-based optimization of type III indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors
Roehrig, Ute F.; Majjigapu, Somi Reddy; Vogel, Pierre; Reynaud, Aline; Pojer, Florence; Dilek, Nahzli; Reichenbach, Patrick; Ascencao, Kelly; Irving, Melita; Coukos, George; Michielin, Olivier; Zoete, Vincent
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收藏Azole-Based Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors唑类吲哚胺2,3-双加氧酶1 (IDO1) 抑制剂
Rohrig, Ute F.; Majjigapu, Somi Reddy; Reynaud, Aline; Pojer, Florence; Dilek, Nahzli; Reichenbach, Patrick; Ascencao, Kelly; Irving, Melita; Coukos, George; Vogel, Pierre; Michielin, Olivier; Zoete, Vincent
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收藏Induction of cell killing and autophagy by amphiphilic pyrrolidine derivatives on human pancreatic cancer cells
Bello, Claudia; Bai, Jianfei; Zambron, Bartosz K.; Elias-Rodriguez, Pilar; Gajate, Consuelo; Robina, Inmaculada; Caffa, Irene; Cea, Michele; Montecucco, Fabrizio; Nencioni, Alessio; Nahimana, Aimable; Aubry, Dominique; Breton, Caroline; Duchosal, Michel A.; Mollinedo, Faustino; Vogel, Pierre
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收藏Detailed analysis and follow-up studies of a high-throughput screening for indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors吲哚胺2,3-双加氧酶1 (IDO1) 抑制剂高通量筛选的详细分析和后续研究
Roehrig, Ute F.; Majjigapu, Somi Reddy; Chambon, Marc; Bron, Sylvian; Pilotte, Luc; Colau, Didier; Van den Eynde, Benoit J.; Turcatti, Gerardo; Vogel, Pierre; Zoete, Vincent; Michielin, Olivier
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收藏A critical role of autophagy in antileukemia/lymphoma effects of APO866, an inhibitor of NAD biosynthesis
Ginet, Vanessa; Puyal, Julien; Rummel, Coralie; Aubry, Dominique; Breton, Caroline; Cloux, Anne-Julie; Majjigapu, Somi R.; Sordat, Bernard; Vogel, Pierre; Bruzzone, Santina; Nencioni, Alessio; Duchosal, Michel A.; Nahimana, Aimable
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收藏Rational Design of 4-Aryl-1,2,3-Triazoles for Indoleamine 2,3-Dioxygenase 1 Inhibition
Roehrig, Ute F.; Majjigapu, Somi Reddy; Grosdidier, Aurelien; Bron, Sylvian; Stroobant, Vincent; Pilotte, Luc; Colau, Didier; Vogel, Pierre; Van den Eynde, Benoit J.; Zoete, Vincent; Michielin, Olivier
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收藏Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols
Bello, Claudia; Dal Bello, Giovanna; Cea, Michele; Nahimana, Aimable; Aubry, Dominique; Garuti, Anna; Motta, Giulia; Moran, Eva; Fruscione, Floriana; Pronzato, Paolo; Grossi, Francesco; Patrone, Franco; Ballestrero, Alberto; Dupuis, Marc; Sordat, Bernard; Zimmermann, Kaspar; Loretan, Jacqueline; Wartmann, Markus; Duchosal, Michel A.; Nencioni, Alessio; Vogel, Pierre
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