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José Marco‐Contelles

Institute of Organic Chemistry (CSIC)

56H指数
483论文数
1.2W被引数
收录论文 185
发表时间
Masupirdine; a Selective Serotonin 5-HT6 Receptor Antagonist for Alzheimer’s Disease
err2026-02-06
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PREAI
errMireia Toledano-Pinedo; Isabel Iriepa; M. Mercedes Rodríguez-Fernández; José Marco-Contelles
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Zervimesine, a Small Sigma-2 Receptor Selective Modulator for Alzheimer's Disease
err2025-12-11
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PREAI
errIriepa, Isabel; Contino, Marialessandra; Abate, Carmen; Marco-Contelles, Jose
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First Sustainable One-Pot Tandem Hantzsch Multicomponent Reaction/Click Reaction Approach for Novel Multitarget-Directed Ligands in Alzheimer's Disease
err2025-12-01
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PREAI
errBernard, Paul J.; Wieckowska, Anna; Grosjean, Sylvain; Godyn, Justyna; Salat, Kinga; Detka, Jan; Palacz, Natalia; Tyrybon, Weronika; Jonczyk, Jakub; Szalaj, Natalia; Zareba, Paula; Martin, Helene; Maj, Maciej; Jozwiak, Krzysztof; Marco-Contelles, Jose; Ismaili, Lhassane
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N-Methyl-N-((1-methyl-5-(3-(piperidin-1-yl)propoxy)-1H-benzo[d]imidazol-2-yl)methyl)prop-2-yn-1-amine (MBA-159), a new multitarget small molecule for the therapy of Alzheimer’s diseaseN-Methyl-N-((1-甲基-5-(3-(哌啶-1-基)丙氧基)-1H-苯并[d]咪唑-2-基)甲基)丙-2-炔-1-胺 (MBA-159),一种用于阿尔茨海默病治疗的新型多靶点小分子
err2025-09-27
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errOAAI
errÓscar M. Bautista-Aguilera; Aleksandra Manik; Daniel Diez-Iriepa; Natalia Szałaj; Paula Zaręba; Anna Więckowska; Paweł Żmudzki; Ewelina Honkisz-Orzechowska; Damijan Knez; Stanislav Gobec; Kinga Sałat; Borja Martínez-Alonso; Víctor Guarnizo-Herrero; Guillermo Torrado Durán; Carlos Torrado-Salmerón; Aina Bellver-Sanchis; Inaya Nsiona-Defise; Marta Ribalta-Vilella; Mercè Pallàs; Francisco López-Muñoz; Christian Griñán-Ferré; José Marco-Contelles; Isabel Iriepa
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Generation and validation of a novel multitarget small molecule in glioblastoma胶质母细胞瘤中新型多靶点小分子的生成与验证
err2025-04-04
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errOAAI
errArtetxe-Zurutuza, Aizpea; Iturrioz-Rodriguez, Nerea; Elizazu, Joseba; Toledano-Pinedo, Mireia; Porro-Perez, Alicia; De Goni, Irati; Elua-Pinin, Alejandro; Schaeker-Huebner, Linda; Azkargorta, Mikel; Elortza, Felix; Iriepa, Isabel; Lopez-Munoz, Francisco; Moncho-Amor, Veronica; Hansen, Finn K.; Sampron, Nicolas; Marco-Contelles, Jose Luis; Matheu, Ander
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Phosphorylated Nitrones-Synthesis and Applications
err2025-03-16
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errOAAI
errRozpara, Iwona; Marco-Contelles, Jose; Piotrowska, Dorota G.; Glowacka, Iwona E.
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Contilisant-Belinostat Hybrids: Polyfunctionalized Indole Derivatives as Multineurotarget Drugs for the Potential Treatment of Alzheimer's DiseaseContilisant-Belinostat 杂合体:多官能化吲哚衍生物作为多神经靶点药物用于阿尔茨海默病潜在治疗
err2025-02-07
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PREAI
errSchäker-Hübner, L; Toledano-Pinedo, M; Eimermacher, S; Krasniqi, V; Porro-Perez, A; Tan, K; Horn, G; Stegen, P; Elsinghorst, PW; Wille, T; Pietsch, M; Gütschow, M; Marco-Contelles, J; Hansen, FK
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Contilisant plus Tubastatin A Hybrids: Polyfunctionalized Indole Derivatives as New HDAC Inhibitor-Based Multitarget Small Molecules with In Vitro and In Vivo Activity in Neurodegenerative Diseases
err2024-09-10
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PREAI
errToledano-Pinedo, Mireia; Porro-Perez, Alicia; Schaeker-Huebner, Linda; Romero, Fernando; Dong, Min; Samadi, Abdelouahid; Almendros, Pedro; Iriepa, Isabel; Bautista-Aguilera, Oscar M.; Rodriguez-Fernandez, M. Mercedes; Solana-Manrique, Cristina; Sanchis, Inmaculada; Mora-Morell, Alba; Rodriguez, Ania Canseco; Sanchez-Perez, Ana M.; Knez, Damijan; Gobec, Stanislav; Bellver-Sanchis, Aina; Perez, Belen; Dobrydnev, Alexey V.; Artetxe-Zurutuza, Aizpea; Matheu, Ander; Siwek, Agata; Wolak, Malgorzata; Satala, Grzegorz; Bojarski, Andrzej J.; Doroz-Plonka, Agata; Handzlik, Jadwiga; Godyn, Justyna; Wieckowska, Anna; Paricio, Nuria; Grinan-Ferre, Christian; Hansen, Finn K.; Marco-Contelles, Jose
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Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors
err2024-08-29
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PREAI
errMalek, Rim; Salat, Kinga; Totoson, Perle; Karcz, Tadeusz; Refouvelet, Bernard; Skrzypczak-Wiercioch, Anna; Maj, Maciej; Simakov, Alexey; Martin, Helene; Siwek, Agata; Szalaj, Natalia; Godyn, Justyna; Panek, Dawid; Wieckowska, Anna; Jozwiak, Krzysztof; Demougeot, Celine; Kiec-Kononowicz, Katarzyna; Chabchoub, Fakher; Iriepa, Isabel; Marco-Contelles, Jose; Ismaili, Lhassane
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Hydrazides as Inhibitors of Histone Deacetylases
err2024-08-02
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PREAI
errCarreiras, Maria do Carmo; Marco-Contelles, Jose
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Synthesis, antioxidant and neuroprotective analysis of diversely functionalized α-aryl-N-alkyl nitrones as potential agents for ischemic stroke therapy
err2024-02-01
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PREAI
errEscobar-Peso, Alejandro; Martinez-Alonso, Emma; Hadjipavlou-Litina, Dimitra; Alcazar, Alberto; Marco-Contelles, Jose
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Neuroprotective and Antioxidant Properties of CholesteroNitrone ChN2 and QuinolylNitrone QN23 in an Experimental Model of Cerebral Ischemia: Involvement of Necrotic and Apoptotic Cell Death
err2023-06-29
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errOAAI
errChamorro, Beatriz; Izquierdo-Bermejo, Sara; Martin-de-Saavedra, Maria Dolores; Lopez-Munoz, Francisco; Chioua, Mourad; Marco-Contelles, Jose; Oset-Gasque, Maria Jesus
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Neuroprotective and antioxidant properties of new quinolylnitrones in in vitro and in vivo cerebral ischemia models
err2023-02-17
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errOAAI
errChamorro, Beatriz; Izquierdo-Bermejo, Sara; Serrano, Julia; Hadjipavlou-Litina, Dimitra; Chioua, Mourad; Lopez-Munoz, Francisco; Marco-Contelles, Jose; Martinez-Murillo, Ricardo; Oset-Gasque, Maria Jesus
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Synthesis and Antioxidant Properties of Novel 1,2,3-Triazole-Containing Nitrones
err2022-12-24
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errOAAI
errHadjipavlou-Litina, Dimitra; Glowacka, Iwona E.; Marco-Contelles, Jose; Piotrowska, Dorota G.
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Biginelli Reaction Synthesis of Novel Multitarget-Directed Ligands with Ca2+ Channel Blocking Ability, Cholinesterase Inhibition, Antioxidant Capacity, and Nrf2 Activation
err2022-12-22
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errOAAI
errMalek, Rim; Simakov, Alexey; Davis, Audrey; Maj, Maciej; Bernard, Paul J.; Wnorowski, Artur; Martin, Helene; Marco-Contelles, Jose; Chabchoub, Fakher; Dallemagne, Patrick; Rochais, Christophe; Jozwiak, Krzysztof; Ismaili, Lhassane
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Benzochromenopyrimidines: Synthesis, Antiproliferative Activity against Colorectal Cancer and Physicochemical Properties
err2022-11-15
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errOAAI
errChoura, Emna; Elghali, Fares; Bernard, Paul J.; Msalbi, Dhouha; Marco-Contelles, Jose; Aifa, Sami; Ismaili, Lhassane; Chabchoub, Fakher
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