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Drug discovery of N-methyl-pyrazole derivatives as potent selective estrogen receptor degrader (SERD) for the treatment of breast cancer N-甲基-吡唑衍生物作为有效的选择性雌激素受体降解剂 (SERD) 用于治疗乳腺癌的药物发现 Dai, Rupeng; Bao, Xueting; Liu, Chao; Yin, Xunkai; Zhu, Zhenzhen; Zheng, Zhe; Wang, Bo; Yang, Kundi; Wen, Hongmei; Li, Wei; Zhu, Haohao; Du, Qianming; Liu, Jian 分享 收藏
Hot-Spot Residue-Based Virtual Screening of Novel Selective Estrogen-Receptor Degraders for Breast Cancer Treatment Dai, Rupeng; Bao, Xueting; Zhang, Ying; Huang, Yan; Zhu, Haohao; Yang, Kundi; Wang, Bo; Wen, Hongmei; Li, Wei; Liu, Jian 分享 收藏
Profiling bourbons based on congener concentrations Zhang, Huan; Johnson, Eric C.; Carroll, Anne; Pryor, Cecily; Howe, Kenneth; Kramer, Ryan; Rajesh, Naik; Meyer, Emily; Shurina, Ben; Kumarage, Nuwanthika; Yang, Kundi; Kennedy, Michael A.; Crowder, Michael W. 分享 收藏
Synthesis of Isoquinolone, 1,2-Benzothiazine, and Naphtho[1',2':4,5]imidazo[1,2-a]pyridine Derivatives via Rhodium(III)-Catalyzed (4+2) Annulation Zhu, Yueyue; Dai, Rupeng; Huang, Chaoqun; Zhou, Wang; Zhang, Xiaoyuan; Yang, Kundi; Wen, Hongmei; Li, Wei; Liu, Jian 分享 收藏
Spectroscopic and biochemical characterization of metallo-8-lactamase IMP-1 with dicarboxylic, sulfonyl, and thiol inhibitors Zhang, Huan; Yang, Kundi; Cheng, Zishuo; Thomas, Caitlyn; Steinbrunner, Abbie; Pryor, Cecily; Vulcan, Maya; Kemp, Claire; Orea, Diego; Paththamperuma, Chathura; Chen, Allie Y.; Cohen, Seth M.; Page, Richard C.; Tierney, David L.; Crowder, Michael W. 分享 收藏
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Carbapenem Use Is Driving the Evolution of Imipenemase 1 Variants Cheng, Zishuo; Bethel, Christopher R.; Thomas, Pei W.; Shurina, Ben A.; Alao, John-Paul; Thomas, Caitlyn A.; Yang, Kundi; Marshall, Steven H.; Zhang, Huan; Sturgill, Aidan M.; Kravats, Andrea N.; Page, Richard C.; Fast, Walter; Bonomo, Robert A.; Crowder, Michael W. 分享 收藏
A Multi-Omics Study Revealing the Metabolic Effects of Estrogen in Liver Cancer Cells HepG2 Shen, Minqian; Xu, Mengyang; Zhong, Fanyi; Crist, McKenzie C.; Prior, Anjali B.; Yang, Kundi; Allaire, Danielle M.; Choueiry, Fouad; Zhu, Jiangjiang; Shi, Haifei 分享 收藏
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Probing the mechanisms of inhibition for various inhibitors of metallo-β-lactamases VIM-2 and NDM-1 Thomas, Caitlyn A.; Cheng, Zishuo; Yang, Kundi; Hellwarth, Elle; Yurkiewicz, Cole J.; Baxter, Faith M.; Fullington, Sarah A.; Klinsky, Spencer A.; Otto, Jen L.; Chen, Allie Y.; Cohen, Seth M.; Crowder, Michael W. 分享 收藏
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Rhodium(III)-Catalyzed Oxidative Annulation of 4-Aminoquinolines and Acrylate through Two Consecutive C(sp2)-H Activations Liu, Jian; Gao, Yi; Zhu, Yehua; Zhu, Junru; Wang, Chao; Rui, Xiyan; Yang, Kundi; Si, Dongjuan; Lin, Jiamin; Yuan, Dandan; Wen, Hongmei; Li, Wei 分享 收藏
A Single Salt Bridge in VIM-20 Increases Protein Stability and Antibiotic Resistance under Low-Zinc Conditions Cheng, Zishuo; Shurina, Ben A.; Bethel, Christopher R.; Thomas, Pei W.; Marshall, Steven H.; Thomas, Caitlyn A.; Yang, Kundi; Kimble, Robert L.; Montgomery, Jonathan S.; Orischak, Matthew G.; Miller, Callie M.; Tennenbaum, Jordan L.; Nix, Jay C.; Tierney, David L.; Fast, Walter; Bonomo, Robert A.; Page, Richard C.; Crowder, Michael W. 分享 收藏
Copper-Catalyzed, Chloroamide-Directed Benzylic C-H Difluoromethylation Zeng, Xiaojun; Yang, Wenhao; Paeth, Matthew; Zacate, Samson B.; Hong, Pei-Hsun; Wang, Yufei; Yang, Dongqi; Yang, Kundi; Yan, Tao; Song, Chang; Cao, Zhi; Cheng, Mu-Jeng; Liu, Wei 分享 收藏
Copper-Catalyzed Decarboxylative Difluoromethylation Zeng, Xiaojun; Yan, Wenhao; Zacate, Samson B.; Chao, Tzu-Hsuan; Sun, Xiaodong; Cao, Zhi; Bradford, Kate G. E.; Paeth, Matthew; Tyndall, Sam B.; Yang, Kundi; Kuo, Tung-Chun; Cheng, Mu-Jeng; Liu, Wei 分享 收藏
Csp3-Csp3 Bond-Forming Reductive Elimination from Well-Defined Copper(III) Complexes 从定义明确的铜 (III) 配合物中Csp3-Csp3形成键的还原消除 Paeth, Matthew; Tyndall, Sam B.; Chen, Liang-Yu; Hong, Jia-Cheng; Carson, William P.; Liu, Xingwu; Sun, Xiaodong; Liu, Jinjia; Yang, Kundi; Hale, Elizabeth M.; Tierney, David L.; Liu, Bin; Cao, Zhi; Cheng, Mu-Jeng; Goddard, William A., III; Liu, Wei 分享 收藏
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