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Discovery of MK-4688: an Efficient Inhibitor of the HDM2-p53 Protein-Protein Interaction Reutershan, Michael H.; Machacek, Michelle R.; Altman, Michael D.; Bogen, Stephane; Cai, Mingmei; Cammarano, Carolyn; Chen, Dapeng; Christopher, Matthew; Cryan, John; Daublain, Pierre; Fradera, Xavier; Geda, Prasanthi; Goldenblatt, Peter; Hill, Armetta D.; Kemper, Raymond A.; Kutilek, Victoria; Li, Chaomin; Martinez, Michelle; McCoy, Mark; Nair, Latha; Pan, Weidong; Thompson, Christopher F.; Scapin, Giovanna; Shizuka, Manami; Spatz, Marianne L.; Steinhuebel, Dietrich; Sun, Binyuan; Voss, Matthew E.; Wang, Xiao; Yang, Liping; Yeh, Tammie C.; Dussault, Isabelle; Marshall, C. Gary; Trotter, B. Wesley 分享 收藏
Projected Dose Optimization of Amino- and Hydroxypyrrolidine Purine PI3Kδ Immunomodulators Methot, Joey L.; Zhou, Hua; McGowan, Meredeth A.; Anthony, Neville John; Christopher, Matthew; Garcia, Yudith; Achab, Abdelghani; Lipford, Kathryn; Trotter, Benjamin Wesley; Altman, Michael D.; Fradera, Xavier; Lesburg, Charles A.; Li, Chaomin; Alves, Stephen; Chappell, Craig P.; Jain, Renu; Mangado, Ruban; Pinheiro, Elaine; Williams, Sybill M. G.; Goldenblatt, Peter; Hill, Armetta; Shaffer, Lynsey; Chen, Dapeng; Tong, Vincent; McLeod, Robbie L.; Lee, Hyun-Hee; Yu, Hongshi; Shah, Sanjiv; Katz, Jason D. 分享 收藏
Process Development and Large-Scale Synthesis of BTK Inhibitor BIIB068 Li, Chaomin; Franklin, Lloyd; Chen, Robbie; Mack, Tamera; Humora, Michael; Ma, Bin; Hopkins, Brian T.; Guzowski, John; Zheng, Fengmei; MacPhee, Michael; Lin, Yiqing; Ferguson, Steven; Patience, Daniel; Moniz, George A.; Kiesman, William F.; O'Brien, Erin M. 分享 收藏
Solid tumor activity with a selective PI3Kdelta inhibitor as a single agent and in combination with anti-PD-1 Methot, Joey L.; Zhou, Hua; McGowan, Meredith A.; Trotter, Benjamin W.; Altman, Michael; Fradera, Xavier; Lesburg, Charles; Li, Chaomin; Alves, Stephen; Chappell, Craig P.; Jain, Renu; Mangado, Ruban; Pinheiro, Elaine; Williams, Sybil M.; Goldenblatt, Peter; Hill, Armetta D.; Shaffer, Lynsey; Chen, Dapeng; McLeod, Robbie L.; Lee, Hyun-Hee; Shah, Sanjiv; Katz, Jason D. 分享 收藏
Process Safety Considerations for the Supply of a High-Energy Oxadiazole IDO1-Selective Inhibitor Martinot, Theodore A.; Ardolino, Michael; Chen, Lu; Lam, Yu-hong; Li, Chaomin; Maddess, Matthew L.; Muzzio, Daniel; Qi, Ji; Sauri, Josep; Song, Zhiguo J.; Tan, Lushi; Vickery, Thomas; Yin, Jingjun; Zhao, Ralph 分享 收藏
Structure Overhaul Affords a Potent Purine PI3Kδ Inhibitor with Improved Tolerability Methot, Joey L.; Zhou, Hua; Kattar, Sam D.; McGowan, Meredeth A.; Wilson, Kevin; Garcia, Yudith; Deng, Yongi; Altman, Michael; Fradera, Xavier; Lesburg, Charles; Fischmann, Thierry; Li, Chaomin; Alves, Steve; Shah, Sanjiv; Fernandez, Rafael; Goldenblatt, Peter; Hill, Armetta; Shaffer, Lynsey; Chen, Dapeng; Tong, Vince; McLeod, Robbie L.; Yu, Hongshi; Bass, Alan; Kemper, Ray; Gatto, Nicholas T.; LaFranco-Scheuch, Lisa; Trotter, Benjamin Wesley; Guzi, Timothy; Katz, Jason D. 分享 收藏
Synthesis and evaluation of an N-[18F]fluorodeoxyglycosyl amino acid for PET imaging of tumor metabolism Wu, Zhifang; Ma, Jingxin; Brownell, Anna-Liisa; Wang, Hongliang; Li, Chaomin; Meng, Xiaxia; Yuan, Ling; Liu, Haiyan; Li, Sijin; Xie, Jun 分享 收藏
Discovery of 1-[3-(1-Methyl-1H-pyrazol-4-y1)-5-oxo-5H-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl]-N-(pyridin-2-ylmethyl)methanesulfonamide (MK-8033): A Specific c-Met/Ron Dual Kinase Inhibitor with Preferential Affinity for the Activated State of c-Met Northrup, Alan B.; Katcher, Matthew H.; Altman, Michael D.; Chenard, Melissa; Daniels, Matthew H.; Deshmukh, Sujal V.; Falcone, Danielle; Guerin, David J.; Hatch, Harold; Li, Chaomin; Lu, Wei; Lutterbach, Bart; Allison, Timothy J.; Patel, Sangita B.; Reily, John F.; Reutershan, Michael; Rickert, Keith W.; Rosenstein, Craig; Soisson, Stephen M.; Szewczak, Alexander A.; Walker, Deborah; Wilson, Kevin; Young, Jonathan R.; Pan, Bo-Sheng; Dinsmore, Christopher J. 分享 收藏
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