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Francisco Gamarro

consejo superior de investigaciones cientificas (csic)

43H指数
165论文数
6.6K被引数
收录论文 78
发表时间
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei
err2024-08-13
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errOAAI
errFerrins, Lori; Diaz, Rosario; Cordon-Obras, Carlos; Rojas-Barros, Domingo; Quotadamo, Antonio; Oehme, Daniel P.; Ceballos-Perez, Gloria; Swaminathan, Uma; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Garcia-Hernandez, Raquel; Gomez-Linan, Claudia; Saura, Andreu; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Martinez-Martinez, Maria Santos; Manzano, Pilar; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Pollastri, Michael P.
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Deciphering Host-Parasite Interplay in Leishmania Infection through a One Health View of Proteomics Studies on Drug Resistance
err2024-08-01
err0
PREAI
errTagliazucchi, Lorenzo; Pinetti, Diego; Genovese, Filippo; Malpezzi, Giulia; Martinez, Ana Perea; Manzano, Jose, I; Garcia-Hernandez, Raquel; Cole, Alexander R.; Kwon, Ba Reum; Aiello, Daniele; Brooks, Bryan W.; Thore, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola
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Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes (vol 14, 1149145, 2023)
err2023-10-25
err0
errOAAI
errFerrins, Lori; Buskes, Melissa J.; Kapteyn, Madison M.; Engels, Hannah N.; Enos, Suzanne E.; Lu, Chenyang; Klug, Dana M.; Singh, Baljinder; Quotadamo, Antonio; Bachovchin, Kelly; Tear, Westley F.; Spaulding, Andrew E.; Forbes, Katherine C.; Bag, Seema; Rivers, Mitch; Leblanc, Catherine; Burchfield, Erin; Armand, Jeremy R.; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Gomez-Linan, Claudia; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Mensa-Wilmot, Kojo; Pollastri, Michael P.; Kyle, Dennis E.; Rice, Christopher A.
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Synthesis and Biophysical and Biological Studies of N-Phenylbenzamide Derivatives Targeting Kinetoplastid Parasites
err2023-09-20
err4
errOAAI
errNue-Martinez, J. Jonathan; Cisneros, David; Moreno-Blazquez, Maria del Valle; Fonseca-Berzal, Cristina; Manzano, Jose Ignacio; Kraeutler, Damien; Ungogo, Marzuq A.; Aloraini, Maha A.; Elati, Hamza A. A.; Ibanez-Escribano, Alexandra; Lagartera, Laura; Herraiz, Tomas; Gamarro, Francisco; de Koning, Harry P.; Gomez-Barrio, Alicia; Dardonville, Christophe
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Strasseriolides display in vitro and in vivo activity against trypanosomal parasites and cause morphological and size defects in Trypanosoma cruzi
err2023-09-15
err2
errOAAI
errBosch-Navarrete, Cristina; Perez-Moreno, Guiomar; Annang, Frederick; Diaz-Gonzalez, Rosario; Garcia-Hernandez, Raquel; Rocha, Hedy; Gamarro, Francisco; Cordon-Obras, Carlos; Navarro, Miguel; Rodriguez, Ana; Genilloud, Olga; Reyes, Fernando; Vicente, Francisca; Ruiz-Perez, Luis M.; Gonzalez-Pacanowska, Dolores
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Label-Free Mass Spectrometry Proteomics Reveals Different Pathways Modulated in THP-1 Cells Infected with Therapeutic Failure and Drug Resistance Leishmania infantum Clinical Isolates
err2023-02-10
err2
errOAAI
errTagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Manzano, Jose Ignacio; Genovese, Filippo; Garcia-Hernandez, Raquel; Pinetti, Diego; Gamarro, Francisco; Costi, Maria Paola
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Transcriptome Analysis of Intracellular Amastigotes of Clinical Leishmania infantum Lines from Therapeutic Failure Patients after Infection of Human Macrophages
err2022-06-27
err3
errOAAI
errGarcia-Hernandez, Raquel; Perea-Martinez, Ana; Ignacio Manzano, Jose; Terron-Camero, Laura C.; Andres-Leon, Eduardo; Gamarro, Francisco
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Transcriptomic Analysis in Human Macrophages Infected with Therapeutic Failure Clinical Isolates of Leishmania infantum
err2022-03-30
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errPerea-Martinez, Ana; Garcia-Hernandez, Raquel; Ignacio Manzano, Jose; Gamarro, Francisco
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Synthesis of sp2-Iminosugar Selenoglycolipids as Multitarget Drug Candidates with Antiproliferative, Leishmanicidal and Anti-Inflammatory Properties
err2021-12-11
err5
errOAAI
errSanchez-Fernandez, Elena M.; Garcia-Hernandez, Raquel; Gamarro, Francisco; Arroba, Ana I.; Aguilar-Diosdado, Manuel; Padron, Jose M.; Garcia Fernandez, Jose M.; Ortiz Mellet, Carmen
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Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis
err2021-06-22
err5
errOAAI
errKlug, Dana M.; Mavrogiannaki, Eftychia M.; Forbes, Katherine C.; Silva, Lisseth; Diaz-Gonzalez, Rosario; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Bosch-Navarrete, Cristina; Cordon-Obras, Carlos; Gomez-Linan, Claudia; Saura, Andreu; Momper, Jeremiah D.; Santos Martinez-Martinez, Maria; Manzano, Pilar; Syed, Ali; El-Sakkary, Nelly; Caffrey, Conor R.; Gamarro, Francisco; Miguel Ruiz-Perez, Luis; Gonzalez Pacanowska, Dolores; Ferrins, Lori; Navarro, Miguel; Pollastri, Michael P.
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Structure-property studies of an imidazoquinoline chemotype with antitrypanosomal activity
err2020-01-01
err3
errOAAI
errKlug, Dana M.; Diaz-Gonzalez, Rosario; DeLano, Travis J.; Mavrogiannaki, Eftychia M.; Buskes, Melissa J.; Dalton, Raeann M.; Fisher, John K.; Schneider, Katherine M.; Hilborne, Vivian; Fritsche, Melanie G.; Simpson, Quillon J.; Tear, Westley F.; Devine, William G.; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Bosch-Navarrete, Cristina; Miguel Ruiz-Perez, Luis; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Santos Martinez-Martinez, Maria; Manzano-Chinchon, Pilar; Navarro, Miguel; Pollastri, Michael P.; Ferrins, Lori
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Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5-b]pyridazines for the Treatment of Human African Trypanosomiasis
err2019-12-17
err14
errOAAI
errTear, Westley F.; Bag, Seema; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; Rojas-Barros, Domingo I.; Cordon-Obras, Carlos; Perez-Moreno, Guiomar; Garcia-Hernandez, Raquel; Santos Martinez-Martinez, Maria; Miguel Ruiz-Perez, Luis; Gamarro, Francisco; Gonzalez Pacanowska, Dolores; Caffrey, Conor R.; Ferrins, Lori; Manzano, Pilar; Navarro, Miguel; Pollastri, Michael P.
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Discovery and Pharmacological Studies of 4-Hydroxyphenyl-Derived Phosphonium Salts Active in a Mouse Model of Visceral Leishmaniasis
err2019-11-08
err14
errOAAI
errIgnacio Manzano, Jose; Cueto-Diaz, Eduardo J.; Isabel Olias-Molero, Ana; Perea, Ana; Herraiz, Tomas; Torrado, Juan J.; Maria Alunda, Jose; Gamarro, Francisco; Dardonville, Christophe
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Synthesis of polyfluoroalkyl sp2-iminosugar glycolipids and evaluation of their immunomodulatory properties towards anti-tumor, anti-leishmanial and anti-inflammatory therapies
err2019-11-01
err18
PREAI
errSanchez-Fernandez, Elena M.; Isabel Garcia-Moreno, Ma; Arroba, Ana I.; Aguilar-Diosdado, Manuel; Padron, Jose M.; Garcia-Hernandez, Raquel; Gamarro, Francisco; Fustero, Santos; Sanchez-Aparicio, Jose-Emilio; Masgrau, Laura; Garcia Fernandez, Jose Manuel; Ortiz Mellet, Carmen
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Imidazo[2,1-a]isoindole scaffold as an uncharted structure active on Leishmania donovani
err2019-11-01
err4
errOAAI
errArsene, Sobinson; Gomez-Perez, Veronica; Escarcena, Ricardo; Angeles Abengozar, Maria; Garcia-Hernandez, Raquel; Nacher-Vazquez, Montserrat; San Feliciano, Arturo; Gamarro, Francisco; Rivas, Luis; del Olmo, Esther
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Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics
err2019-10-31
err17
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errKlug, Dana M.; Tschiegg, Laura; Diaz, Rosario; Rojas-Barros, Domingo; Perez-Moreno, Guiomar; Ceballos, Gloria; Garcia-Hernandez, Raquel; Santos Martinez-Martinez, Maria; Manzano, Pilar; Miguel Ruiz, Luis; Caffrey, Conor R.; Gamarro, Francisco; Gonzalez Pacanowska, Dolores; Ferrins, Lori; Navarro, Miguel; Pollastri, Michael P.
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4-Aminoquinoline-based compounds as antileishmanial agents that inhibit the energy metabolism of Leishmania基于4-氨基喹啉的化合物作为抑制利什曼原虫能量代谢的抗利什曼原药
err2019-10-01
err13
PREAI
errManzano, Jose Ignacio; Konstantinovic, Jelena; Scaccabarozzi, Diletta; Perea, Ana; Pavic, Aleksandar; Cavicchini, Loredana; Basilico, Nicoletta; Gamarro, Francisco; Solaja, Bogdan A.
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Thiol-ene Click Synthesis and Pharmacological Evaluation of C-Glycoside sp2-Iminosugar Glycolipids
err2019-08-08
err9
errOAAI
errSanchez-Fernandez, Elena M.; Isabel Garcia-Moreno, M.; Garcia-Hernandez, Raquel; Padron, Jose M.; Garcia Fernandez, Jose M.; Gamarro, Francisco; Ortiz Mellet, Carmen
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Complete assembly of the Leishmania donovani (HU3 strain) genome and transcriptome annotation
err2019-04-16
err24
errOAAI
errCamacho, Esther; Gonzalez-de La Fuent, Sandra; Rastrojo, Alberto; Peiro-Pastor, Ramon; Solana, Jose Carlos; Tabera, Laura; Gamarro, Francisco; Carrasco-Ramiro, Fernando; Requen, Jose M.; Aguado, Begoiia
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Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents
err2019-02-08
err3
errOAAI
errKlug, Dana M.; Diaz-Gonzalez, Rosario; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Gomez-Perez, Veronica; Ruiz-Perez, Luis Miguel; Rojas-Barros, Domingo I.; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Martinez-Martinez, Maria S.; Manzano, Pilar; Ferrins, Lori; Caffrey, Conor R.; Navarro, Miguel; Pollastri, Michael P.
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