未登录 Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei Ferrins, Lori; Diaz, Rosario; Cordon-Obras, Carlos; Rojas-Barros, Domingo; Quotadamo, Antonio; Oehme, Daniel P.; Ceballos-Perez, Gloria; Swaminathan, Uma; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Garcia-Hernandez, Raquel; Gomez-Linan, Claudia; Saura, Andreu; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Martinez-Martinez, Maria Santos; Manzano, Pilar; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Pollastri, Michael P. 分享 收藏
Deciphering Host-Parasite Interplay in Leishmania Infection through a One Health View of Proteomics Studies on Drug Resistance Tagliazucchi, Lorenzo; Pinetti, Diego; Genovese, Filippo; Malpezzi, Giulia; Martinez, Ana Perea; Manzano, Jose, I; Garcia-Hernandez, Raquel; Cole, Alexander R.; Kwon, Ba Reum; Aiello, Daniele; Brooks, Bryan W.; Thore, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola 分享 收藏
Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes (vol 14, 1149145, 2023) Ferrins, Lori; Buskes, Melissa J.; Kapteyn, Madison M.; Engels, Hannah N.; Enos, Suzanne E.; Lu, Chenyang; Klug, Dana M.; Singh, Baljinder; Quotadamo, Antonio; Bachovchin, Kelly; Tear, Westley F.; Spaulding, Andrew E.; Forbes, Katherine C.; Bag, Seema; Rivers, Mitch; Leblanc, Catherine; Burchfield, Erin; Armand, Jeremy R.; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Gomez-Linan, Claudia; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Mensa-Wilmot, Kojo; Pollastri, Michael P.; Kyle, Dennis E.; Rice, Christopher A. 分享 收藏
Synthesis and Biophysical and Biological Studies of N-Phenylbenzamide Derivatives Targeting Kinetoplastid Parasites Nue-Martinez, J. Jonathan; Cisneros, David; Moreno-Blazquez, Maria del Valle; Fonseca-Berzal, Cristina; Manzano, Jose Ignacio; Kraeutler, Damien; Ungogo, Marzuq A.; Aloraini, Maha A.; Elati, Hamza A. A.; Ibanez-Escribano, Alexandra; Lagartera, Laura; Herraiz, Tomas; Gamarro, Francisco; de Koning, Harry P.; Gomez-Barrio, Alicia; Dardonville, Christophe 分享 收藏
Strasseriolides display in vitro and in vivo activity against trypanosomal parasites and cause morphological and size defects in Trypanosoma cruzi Bosch-Navarrete, Cristina; Perez-Moreno, Guiomar; Annang, Frederick; Diaz-Gonzalez, Rosario; Garcia-Hernandez, Raquel; Rocha, Hedy; Gamarro, Francisco; Cordon-Obras, Carlos; Navarro, Miguel; Rodriguez, Ana; Genilloud, Olga; Reyes, Fernando; Vicente, Francisca; Ruiz-Perez, Luis M.; Gonzalez-Pacanowska, Dolores 分享 收藏
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Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis Klug, Dana M.; Mavrogiannaki, Eftychia M.; Forbes, Katherine C.; Silva, Lisseth; Diaz-Gonzalez, Rosario; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Bosch-Navarrete, Cristina; Cordon-Obras, Carlos; Gomez-Linan, Claudia; Saura, Andreu; Momper, Jeremiah D.; Santos Martinez-Martinez, Maria; Manzano, Pilar; Syed, Ali; El-Sakkary, Nelly; Caffrey, Conor R.; Gamarro, Francisco; Miguel Ruiz-Perez, Luis; Gonzalez Pacanowska, Dolores; Ferrins, Lori; Navarro, Miguel; Pollastri, Michael P. 分享 收藏
Structure-property studies of an imidazoquinoline chemotype with antitrypanosomal activity Klug, Dana M.; Diaz-Gonzalez, Rosario; DeLano, Travis J.; Mavrogiannaki, Eftychia M.; Buskes, Melissa J.; Dalton, Raeann M.; Fisher, John K.; Schneider, Katherine M.; Hilborne, Vivian; Fritsche, Melanie G.; Simpson, Quillon J.; Tear, Westley F.; Devine, William G.; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Bosch-Navarrete, Cristina; Miguel Ruiz-Perez, Luis; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Santos Martinez-Martinez, Maria; Manzano-Chinchon, Pilar; Navarro, Miguel; Pollastri, Michael P.; Ferrins, Lori 分享 收藏
Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5-b]pyridazines for the Treatment of Human African Trypanosomiasis Tear, Westley F.; Bag, Seema; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; Rojas-Barros, Domingo I.; Cordon-Obras, Carlos; Perez-Moreno, Guiomar; Garcia-Hernandez, Raquel; Santos Martinez-Martinez, Maria; Miguel Ruiz-Perez, Luis; Gamarro, Francisco; Gonzalez Pacanowska, Dolores; Caffrey, Conor R.; Ferrins, Lori; Manzano, Pilar; Navarro, Miguel; Pollastri, Michael P. 分享 收藏
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Synthesis of polyfluoroalkyl sp2-iminosugar glycolipids and evaluation of their immunomodulatory properties towards anti-tumor, anti-leishmanial and anti-inflammatory therapies Sanchez-Fernandez, Elena M.; Isabel Garcia-Moreno, Ma; Arroba, Ana I.; Aguilar-Diosdado, Manuel; Padron, Jose M.; Garcia-Hernandez, Raquel; Gamarro, Francisco; Fustero, Santos; Sanchez-Aparicio, Jose-Emilio; Masgrau, Laura; Garcia Fernandez, Jose Manuel; Ortiz Mellet, Carmen 分享 收藏
Imidazo[2,1-a]isoindole scaffold as an uncharted structure active on Leishmania donovani Arsene, Sobinson; Gomez-Perez, Veronica; Escarcena, Ricardo; Angeles Abengozar, Maria; Garcia-Hernandez, Raquel; Nacher-Vazquez, Montserrat; San Feliciano, Arturo; Gamarro, Francisco; Rivas, Luis; del Olmo, Esther 分享 收藏
Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics Klug, Dana M.; Tschiegg, Laura; Diaz, Rosario; Rojas-Barros, Domingo; Perez-Moreno, Guiomar; Ceballos, Gloria; Garcia-Hernandez, Raquel; Santos Martinez-Martinez, Maria; Manzano, Pilar; Miguel Ruiz, Luis; Caffrey, Conor R.; Gamarro, Francisco; Gonzalez Pacanowska, Dolores; Ferrins, Lori; Navarro, Miguel; Pollastri, Michael P. 分享 收藏
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Complete assembly of the Leishmania donovani (HU3 strain) genome and transcriptome annotation Camacho, Esther; Gonzalez-de La Fuent, Sandra; Rastrojo, Alberto; Peiro-Pastor, Ramon; Solana, Jose Carlos; Tabera, Laura; Gamarro, Francisco; Carrasco-Ramiro, Fernando; Requen, Jose M.; Aguado, Begoiia 分享 收藏
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents Klug, Dana M.; Diaz-Gonzalez, Rosario; Perez-Moreno, Guiomar; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Gomez-Perez, Veronica; Ruiz-Perez, Luis Miguel; Rojas-Barros, Domingo I.; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Martinez-Martinez, Maria S.; Manzano, Pilar; Ferrins, Lori; Caffrey, Conor R.; Navarro, Miguel; Pollastri, Michael P. 分享 收藏