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Isoform-Selective PAD2/PAD4 Substrates with Unnatural Amino Acids Enable Cellular Peptidylarginine Deiminase Activity Profiling and Reveal Vimentin Citrullination Effects in Macrophages 异构体选择性PAD2/PAD4底物与非常规氨基酸能够实现细胞内肽基精氨酸脱亚胺酶活性分析,并揭示巨噬细胞中波形蛋白瓜氨酸化的效应 Gorzen, Oliwia; Mikolajczyk-Martinez, Agata; Mamun, Abdulla Al.; Horbach, Natalia; Severynovska, Olha; Bereta, Grzegorz; Bielecka, Ewa; Mydel, Piotr; Drag, Marcin; Kantyka, Tomasz; Poreba, Marcin 分享 收藏
Chemical tools to define and manipulate interferon-inducible Ubl protease USP18 化学工具用于定义和操纵干扰素诱导的泛素样蛋白酶USP18 Davis, Griffin J.; Omole, Anthony O.; Jung, Yejin; Rut, Wioletta; Holewinski, Ronald; Suazo, Kiall F.; Kim, Hong-Rae; Yang, Mo; Andresson, Thorkell; Drag, Marcin; Yoo, Euna 分享 收藏
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Thermoprotection by a cell membrane-localized metacaspase in a green alga Zou, Yong; Sabljic, Igor; Horbach, Natalia; Dauphinee, Adrian N.; Asman, Anna; Sancho Temino, Lucia; Minina, Elena A.; Drag, Marcin; Stael, Simon; Poreba, Marcin; Stahlberg, Jerry; Bozhkov, Peter, V 分享 收藏
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Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections Reinke, Patrick Y. A.; de Souza, Edmarcia Elisa; Guenther, Sebastian; Falke, Sven; Lieske, Julia; Ewert, Wiebke; Loboda, Jure; Herrmann, Alexander; Mashhour, Aida Rahmani; Karnicar, Katarina; Usenik, Aleksandra; Lindic, Natasa; Sekirnik, Andreja; Botosso, Viviane Fongaro; Santelli, Glaucia Maria Machado; Kapronezai, Josana; de Araujo, Marcelo Valdemir; Silva-Pereira, Taiana Taina; de Souza Filho, Antonio Francisco; Tavares, Mariana Silva; Florez-Alvarez, Lizdany; de Oliveira, Danielle Bruna Leal; Durigon, Edison Luiz; Giaretta, Paula Roberta; Heinemann, Marcos Bryan; Hauser, Maurice; Seychell, Brandon; Boehler, Hendrik; Rut, Wioletta; Drag, Marcin; Beck, Tobias; Cox, Russell; Chapman, Henry N.; Betzel, Christian; Brehm, Wolfgang; Hinrichs, Winfried; Ebert, Gregor; Latham, Sharissa L.; de Sa Guimaraes, Ana Marcia; Turk, Dusan; Wrenger, Carsten; Meents, Alke 分享 收藏
Ebselen derivatives inhibit SARS-CoV-2 replication by inhibition of its essential proteins: PLpro and Mpro proteases, and nsp14 guanine N7-methyltransferase Zmudzinski, Mikolaj; Rut, Wioletta; Olech, Kamila; Granda, Jaroslaw; Giurg, Miroslaw; Burda-Grabowska, Malgorzata; Kaleta, Rafal; Zgarbova, Michala; Kasprzyk, Renata; Zhang, Linlin; Sun, Xinyuanyuan; Lv, Zongyang; Nayak, Digant; Kesik-Brodacka, Malgorzata; Olsen, Shaun K.; Weber, Jan; Hilgenfeld, Rolf; Jemielity, Jacek; Drag, Marcin 分享 收藏
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SARS-CoV-2 Mpro Protease Variants of Concern Display Altered Viral Substrate and Cell Host Target Galectin-8 Processing but Retain Sensitivity toward Antivirals Chen, Sizhu Amelia; Arutyunova, Elena; Lu, Jimmy; Khan, Muhammad Bashir; Rut, Wioletta; Zmudzinski, Mikolaj; Shahbaz, Shima; Iyyathurai, Jegan; Moussa, Eman W.; Turner, Zoe; Bai, Bing; Lamer, Tess; Nieman, James A.; Vederas, John C.; Julien, Olivier; Drag, Marcin; Elahi, Shokrollah; Young, Howard S.; Lemieux, M. Joanne 分享 收藏
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Evaluation of the anti-SARS-CoV-2 properties of essential oils and aromatic extracts Strub, Daniel Jan; Talma, Michal; Strub, Maria; Rut, Wioletta; Zmudzinski, Mikolaj; Brud, Wladyslaw; Neyts, Johan; Vangeel, Laura; Zhang, Linlin; Sun, Xinyuanyuan; Lv, Zongyang; Nayak, Digant; Olsen, Shaun K.; Hilgenfeld, Rolf; Jochmans, Dirk; Drag, Marcin 分享 收藏
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Parallel imaging of coagulation pathway proteases activated protein C, thrombin, and factor Xa in human plasma Modrzycka, Sylwia; Kolt, Sonia; Polderdijk, Stephanie G., I; Adams, Ty E.; Potoczek, Stanislaw; Huntington, James A.; Kasperkiewicz, Paulina; Drag, Marcin 分享 收藏
Mechanistic insights into COVID-19 by global analysis of the SARS-CoV-2 3CLpro substrate degradome Pablos, Isabel; Machado, Yoan; de Jesus, Hugo C. Ramos; Mohamud, Yasir; Kappelhoff, Reinhild; Lindskog, Cecilia; Vlok, Marli; Bell, Peter A.; Butler, Georgina S.; Grin, Peter M.; Cao, Quynh T.; Nguyen, Jenny P.; Solis, Nestor; Abbina, Srinivas; Rut, Wioletta; Vederas, John C.; Szekely, Laszlo; Szakos, Attila; Drag, Marcin; Kizhakkedathu, Jayachandran N.; Mossman, Karen; Hirota, Jeremy A.; Jan, Eric; Luo, Honglin; Banerjee, Arinjay; Overall, Christopher M. 分享 收藏