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Helmut Schmidhammer

university of innsbruck

31H指数
250论文数
2.8K被引数
收录论文 58
发表时间
Structural and functional basis of antinociceptive action of χ-conotoxin AoIA at the noradrenaline transporterχ-芋螺毒素AoIA在去甲肾上腺素转运蛋白上的镇痛作用的结构和功能基础
err2026-07-21
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errOliver J. V. Belleza; Heng Zhang; Helmut Schmidhammer; Tye I. Gonzalez; Cosmin I. Ciotu; Nataša Tomašević; Carlo Martin M. Ocampo; Jomari C. Fernando; Johannes Koehbach; Paula Schwarz; Mounaf Al Makhlouf; Gabor Tajti; Simon Hasinger; Nina Kastner; Orcun Avsar; Bernhard Retzl; Kathrin Jäntsch; Yi Jiang; Roland Hellinger; Michael J. M. Fischer; K. Johan Rosengren; Christian W. Gruber; Aaron Joseph L. Villaraza; Thomas Stockner; Mariana Spetea; H. Eric Xu; Harald H. Sitte
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Mechanistic Insights into G Protein-Biased κ-Opioid Receptor Signaling Using Dual-Charged Naltrexamine Amides使用双电荷纳曲胺酰胺对g蛋白偏向的 κ 阿片受体信号传导的机理见解
err2026-02-05
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errNiklas Piet Doering; Kristina Puls; Marta Diceglie; Anja Meraner; Axel Hentsch; Siriwat Hongnak; Armin Wurzer; Helmut Schmidhammer; Mariana Spetea; Marc Nazare; Gerhard Wolber
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MACROCYCLIC AND STABILIZED DYNORPHIN PEPTIDES AS POTENT ANALGESICS FOR IBD PAIN MANAGEMENT大环化和稳定化的强啡肽作为IBD疼痛管理的强效镇痛剂
err2026-02-01
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PREAI
errBecker, Elena; Pircher, Claudia; Khatri, Bhavesh; Muratspahic, Edin; Schmidhammer, Helmut; Spetea, Mariana; Craik, David; Gruber, Christian
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Peripheralization Strategies Applied to Morphinans and Implications for Improved Treatment of Pain
err2023-06-14
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errSchmidhammer, Helmut; Al-Khrasani, Mahmoud; Furst, Susanna; Spetea, Mariana
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Development of Diphenethylamines as Selective Kappa Opioid Receptor Ligands and Their Pharmacological Activities
err2020-11-02
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errSchmidhammer, Helmut; Erli, Filippo; Guerrieri, Elena; Spetea, Mariana
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On the Role of Peripheral Sensory and Gut Mu Opioid Receptors: Peripheral Analgesia and Tolerance
err2020-05-26
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errFurst, Susanna; Zadori, Zoltan S.; Zador, Ferenc; Kiraly, Kornel; Balogh, Mihaly; Laszlo, Szilvia B.; Hutka, Barbara; Mohammadzadeh, Amir; Calabrese, Chiara; Galambos, Anna Rita; Riba, Pal; Romualdi, Patrizia; Benyhe, Sandor; Timar, Julia; Schmidhammer, Helmut; Spetea, Mariana; Al-Khrasani, Mahmoud
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N-Phenethyl Substitution in 14-Methoxy-N-methylmorphinan-6-ones Turns Selective μ Opioid Receptor Ligands into Dual μ/δ Opioid Receptor Agonists
err2020-03-27
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errDumitrascuta, Maria; Bermudez, Marcel; Ben Haddou, Tanila; Guerrieri, Elena; Schlaefer, Lea; Ritsch, Andreas; Hosztafi, Sandor; Lantero, Aquilino; Kreutz, Christoph; Massotte, Dominique; Schmidhammer, Helmut; Wolber, Gerhard; Spetea, Mariana
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Synthesis, Biological, and Structural Explorations of New Zwitterionic Derivatives of 14-O-Methyloxymorphone, as Potent μ/δ Opioid Agonists and Peripherally Selective Antinociceptives
err2018-12-20
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errSpetea, Mariana; Rief, Silvia B.; Ben Haddou, Tanila; Fink, Monika; Kristeva, Elka; Mittendorfer, Harald; Haas, Stefanie; Hummer, Nora; Follia, Valeria; Guerrieri, Elena; Asim, Muhammad Faheem; Sturm, Sonja; Schmidhammer, Helmut
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Synthesis, Pharmacology, and Molecular Docking Studies on 6-Desoxo-N-methylmorphinans as Potent μ-Opioid Receptor Agonists
err2017-11-03
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errDumitrascuta, Maria; Ben Haddou, Tanila; Guerrieri, Elena; Noha, Stefan M.; Schlaefer, Lea; Schmidhammer, Helmut; Spetea, Mariana
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Highly Potent and Selective New Diphenethylamines Interacting with the κ-Opioid Receptor: Synthesis, Pharmacology, and Structure-Activity Relationships
err2017-08-30
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errErli, Filippo; Guerrieri, Elena; Ben Haddou, Tanila; Lantero, Aquilino; Mairegger, Michael; Schmidhammer, Helmut; Spetea, Mariana
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Selective κ receptor partial agonist HS666 produces potent antinociception without inducing aversion after i.c.v. administration in mice
err2017-06-27
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errSpetea, Mariana; Eans, Shainnel O.; Ganno, Michelle L.; Lantero, Aquilino; Mairegger, Michael; Toll, Lawrence; Schmidhammer, Helmut; McLaughlin, Jay P.
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μ Opioid receptor: novel antagonists and structural modeling
err2016-02-18
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errKaserer, Teresa; Lantero, Aquilino; Schmidhammer, Helmut; Spetea, Mariana; Schuster, Daniela
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Synthesis and Pharmacological Evaluation of [3H]HS665, a Novel, Highly Selective Radioligand for the Kappa Opioid Receptor
err2014-12-24
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PREAI
errGuerrieri, Elena; Mallareddy, Jayapal Reddy; Toth, Geza; Schmidhammer, Helmut; Spetea, Mariana
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Novel 9′-substituted-noscapines: Synthesis with Suzuki cross-coupling, structure elucidation and biological evaluation
err2014-09-01
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errPorcu, Elena; Sipos, Attila; Basso, Giuseppe; Hamel, Ernest; Bai, Ruoli; Stempfer, Verena; Udvardy, Antal; Benyei, Attila Cs; Schmidhammer, Helmut; Antus, Sandor; Viola, Giampietro
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