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Michael E. Kopach

Eli Lilly and Company

27H指数
86论文数
3.2K被引数
收录论文 54
发表时间
Perspectives on Sustainability in the Pharmaceutical Industry制药行业的可持续发展展望
err2026-04-27
err0
errOAAI
errHarrison B. Rose; Huey Shann Sue; Martin D. Eastgate; Michael E. Kopach; Nima Yazdanpanah; Moiz Diwan; Andreas S. Bommarius
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A Convergent Hybrid Gram-Scale Synthesis of Tirzepatide: Tangential Flow Filtration Assisted Native Chemical Ligation-Desulfurization Approach
err2025-12-01
err0
PREAI
errJalan, Ankur; Murzinski, Emily S.; Jansen, Patrick J.; Miller, Richard D.; Embry, Matthew C.; Scherer, Roger B.; Moomaw, John F.; Williams, Katerina M.; Fisher, Cyrus A.; James, Jinju; Arbour, Christine A.; Guinn, Emily J.; Teng, Jing; Kopach, Michael E.
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Quality by design of solid-phase peptide/protein coupling reaction via mechanistic reaction kinetics modeling approach
err2024-04-12
err1
PREAI
errWang, Jingyao; Agrawal, Paridhi; Berglund, Mark R.; Groh, Jennifer McClary; Kopach, Michael E.; Seibert, Kevin D.; Viswanath, Shekhar K.
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Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in Peptide Synthesis过程质量强度 (PMI): 对当前肽制造过程的整体分析为肽合成的可持续性提供了信息
err2024-03-20
err28
errOAAI
errKekessie, Ivy; Wegner, Katarzyna; Martinez, Isamir; Kopach, Michael E.; White, Timothy D.; Tom, Janine K.; Kenworthy, Martin N.; Gallou, Fabrice; Lopez, John; Koenig, Stefan G.; Payne, Philippa R.; Eissler, Stefan; Arumugam, Balasubramanian; Li, Changfeng; Mukherjee, Subha; Isidro-Llobet, Albert; Ludemann-Hombourger, Olivier; Richardson, Paul; Kittelmann, Jorg; Pedersen, Daniel Sejer; van den Bos, Leendert J.
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Phosphine-Dependent Photoinitiation of Alkyl Thiols under Near-UV Light Facilitates User-Friendly Peptide Desulfurization
err2023-01-05
err19
PREAI
errVenneti, Naresh M.; Samala, Ganesh; Morsy, Rana M. I.; Mendoza, Lawrence G.; Isidro-Llobet, Albert; Tom, Janine K.; Mukherjee, Subha; Kopach, Michael E.; Stockdill, Jennifer L.
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Metal-free reductive desulfurization of C-sp3-substituted thiols using phosphite catalysis
err2023-01-01
err4
errOAAI
errMorsy, Rana M. I.; Samala, Ganesh; Jalan, Ankur; Kopach, Michael E.; Venneti, Naresh M.; Stockdill, Jennifer L.
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Mechanistic Study of Diketopiperazine Formation during Solid- Phase Peptide Synthesis of Tirzepatide
err2022-12-06
err14
errOAAI
errWang, Jingyao; Berglund, Mark R.; Braden, Timothy; Embry, Matthew C.; Johnson, Martin D.; Groskreutz, Stephen R.; Sayyed, Fareed Bhasha; Tsukanov, Sergey Vladimirovich; White, Timothy D.; Jalan, Ankur; Seibert, Kevin D.; Kopach, Michael E.
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Improved iGAL 2.0 Metric Empowers Pharmaceutical Scientists to Make Meaningful Contributions to United Nations Sustainable Development Goal 12
err2021-08-12
err34
errOAAI
errRoschangar, Frank; Li, Jun; Zhou, Yanyan; Aelterman, Wim; Borovika, Alina; Colberg, Juan; Dickson, David P.; Gallou, Fabrice; Hayler, John D.; Koenig, Stefan G.; Kopach, Michael E.; Kosjek, Birgit; Leahy, David K.; O'Brien, Erin; Smith, Austin G.; Henry, Manuel; Cook, Jutta; Sheldon, Roger A.
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Kilogram-Scale GMP Manufacture of Tirzepatide Using a Hybrid SPPS/LPPS Approach with Continuous Manufacturing
err2021-06-17
err37
PREAI
errFrederick, Michael O.; Boyse, Raymond A.; Braden, Timothy M.; Calvin, Joel R.; Campbell, Bradley M.; Changi, Shujauddin M.; Coffin, Stephanie R.; Condon, Carmel; Gowran, Olivia; Groh, Jennifer McClary; Groskreutz, Stephen R.; Harms, Zachary D.; Humenik, Ashley A.; Kallman, Neil J.; Klitzing, Nicholas D.; Kopach, Michael E.; Kretsinger, Juliana K.; Lambertus, Gordon R.; Lampert, Jeffrey T.; Maguire, Laura M.; Moynihan, Humphrey A.; Mullane, Nessa S.; Murphy, John D.; O'Mahony, Marie E.; Richey, Rachel N.; Seibert, Kevin D.; Spencer, Richard D.; Strege, Mark A.; Tandogan, Nil; Torres, Frank L. Torres; Tsukanov, Sergey, V; Xia, Han
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Liquid Phase Peptide Synthesis via One-Pot Nanostar Sieving (PEPSTAR)通过一锅Nanostar筛分 (PEPSTAR) 进行液相肽合成
err2021-02-24
err25
errOAAI
errYeo, Jet; Peeva, Ludmila; Chung, Seoyeon; Gaffney, Piers; Kim, Daeok; Luciani, Carla; Tsukanov, Sergey; Seibert, Kevin; Kopach, Michael; Albericio, Fernando; Livingston, Andrew
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Sustainability Challenges and Opportunities in Oligonucleotide Manufacturing
err2020-11-30
err71
errOAAI
errAndrews, Benjamin, I; Antia, Firoz D.; Brueggemeier, Shawn B.; Diorazio, Louis J.; Koenig, Stefan G.; Kopach, Michael E.; Lee, Heewon; Olbrich, Martin; Watson, Anna L.
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The PMI Predictor app to enable green-by-design chemical synthesis
err2019-10-28
err35
PREAI
errBorovika, Alina; Albrecht, Jacob; Li, Jun; Wells, Andrew S.; Briddell, Christiana; Dillon, Barry R.; Diorazio, Louis J.; Gage, James R.; Gallou, Fabrice; Koenig, Stefan G.; Kopach, Michael E.; Leahy, David K.; Martinez, Isamir; Olbrich, Martin; Piper, Jared L.; Roschangar, Frank; Sherer, Edward C.; Eastgate, Martin D.
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Sodium Butylated Hydroxytoluene (NaBHT) as a New and Efficient Hydride Source for Pd-Catalysed Reduction Reactions
err2019-09-19
err4
PREAI
errSharif, Sepideh; Rodriguez, Michael J.; Lu, Yu; Kopach, Michael E.; Mitchell, David; Hunter, Howard N.; Organ, Michael G.
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A Green Chemistry Continuum for a Robust and Sustainable Active Pharmaceutical Ingredient Supply Chain
err2019-09-19
err42
PREAI
errKoenig, Stefan G.; Bee, Cisco; Boroyika, Alina; Briddell, Christiana; Colberg, Juan; Humphrey, Guy R.; Kopach, Michael E.; Martinez, Isamir; Nambiar, Sudhir; Plummer, Scott V.; Ribe, Seth D.; Roschangar, Frank; Scott, Jeremy P.; Sneddon, Helen F.
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Sustainability Challenges in Peptide Synthesis and Purification: From R&D to Production
err2019-03-22
err311
errOAAI
errIsidro-Llobet, Albert; Kenworthy, Martin N.; Mukherjee, Subha; Kojach, Michael E.; Wegner, Katarzyna; Gallou, Fabrice; Smith, Austin G.; Roschangar, Frank
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Bringing Macrolactamization Full Circle: Self-Cleaving Head-to-Tail Macrocyclization of Unprotected Peptides via Mild N-Acyl Urea Activation
err2018-12-19
err22
PREAI
errArbour, Christine A.; Belavek, Kayla J.; Tariq, Rooha; Mukherjee, Subha; Tom, Janine K.; Isidro-Llobet, Albert; Kopach, Michael E.; Stockdill, Jennifer L.
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