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收藏Identification of Novel β-Lactam Derivatives as Proteasome Inhibitors for Antitumor Therapy新型β-内酰胺衍生物作为蛋白酶体抑制剂在抗肿瘤治疗中的鉴定
Cao, Yu; Xu, Gaoya; Gao, Lixin; Sun, Jingjing; Zhang, Lu; Tong, Qiao; Kong, Limin; Zhang, Jiankang; Zhou, Yubo; Liao, Li; Fu, Liping; Xi, Jianjun
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收藏Synthesis, photophysical properties and fluorescent application of novel [1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one derivatives
Gan, Suya; Gao, Li-Xin; Cao, Zitong; Zhang, Chun; Fu, Yiqiu; Wang, Wen-Long
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收藏Insights into the fluorescence and bio-activity of 2-quinolone derivatives against SHP2 from simulated and experimental aspects
Zhang, Chun; Yang, Yuting; Gao, Li-Xin; Gan, Suya; Zhao, Tian-Tian; Gao, Wenran; Li, Jia; Zhu, Yun-Long; Zhou, Yu-Bo; Wang, Wen-Long
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收藏Synthesis, fluorescence properties of novel thiazolo[3,2-b][1,2,4]triazol derivatives as potent SHP2 inhibitors and its uses in sensing for Fe3+and cell imaging
Yan, Xue; Zhang, Chun; Gao, Li-Xin; Cao, Zi-Tong; Gan, Su-Ya; Li, Jia; Xiang, Da-Jun; Zhou, Yu-Bo; Wang, Wen-Long
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收藏pH-Responsive DNA-Functionalized Liquid Metal-Organic Frameworks (L-MOFs) as Molecular Sponges for Ultrasensitive and Label-Free SERS Detection of Folic AcidpH响应性DNA功能化液态金属有机框架(L-MOFs)作为分子海绵,用于叶酸的超灵敏和无标签SERS检测
Liu, Xu; Glazutdinova, Liliia; Wu, Guangrun; Yang, Wenxu; Liu, Hongbo; Shen, Yifu; Zhang, Siyao; Wu, Jing; Ji, Haoyu; Gao, Lixin; Gao, Xinlu; Zhao, Jiayi
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收藏Novel functionalized benzimidazole-salicylic acid derivatives: synthesis, photophysical characteristics and biological applications
Yan, Xue; Gao, Li-Xin; Cao, Zi-Tong; Gan, Su-Ya; Fu, Yi-Qiu; Li, Jia; Xiang, Da-Jun; Zhou, Yu-Bo; Wang, Wen-Long
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收藏DiPTAC: A degradation platform via directly targeting proteasomeDiPTAC:一种通过直接靶向蛋白酶体实现降解的平台
Tu, YT; Yu, Q; Li, MN; Gao, LX; Mao, JL; Ma, JK; Dong, XW; Che, JX; Zhang, C; Zeng, LH; Zhu, HJ; Shao, JA; Hou, JL; Hu, LM; Wan, BB; Li, J; Zhou, YB; Zhang, JK
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收藏Exploration of novel 20S proteasome activators featuring anthraquinone structures and their application in hypoxic cardiomyocyte protection
Yu, Qian; Gao, Lixin; Xu, Linhao; Han, Yubing; Cao, Yu; Xi, Jianjun; Zhong, Yigang; Li, Linjie; Shen, Liteng; Che, Jinxin; Dong, Xiaowu; Zhang, Chong; Zeng, Linghui; Zhu, Huajian; Shao, Jiaan; Xu, Yizhou; Li, Jia; Zhou, Yubo; Zhang, Jiankang
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收藏Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
Wang, Wen-Jing; Gao, Lixin; Wang, Simei; Huang, Wensi; Meng, Xin-Yu; Hu, Hao; Chen, Ziqiang; Sun, Jingya; Yuan, Yali; Zhou, Yubo; Diao, Xingxing; Huang, Ruimin; Li, Jia; Chen, Xiao-Hua
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收藏Discovery and Optimization of Novel Nonbile Acid FXR Agonists as Preclinical Candidates for the Treatment of Inflammatory Bowel Disease
Li, Yuan; Xu, Tingting; Zhao, Yue; Zhang, Hui; Liu, Zesheng; Wang, Hao; Huang, Chaoying; Shu, Zhihao; Gao, Lixin; Xie, Rongrong; Jiao, Tingying; Zhang, Dan; Zhang, Dong; Liang, Xuewu; Zang, Yi; Sun, Yili; Liu, Hong; Li, Jia; Zhou, Yu
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收藏Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
Yan, Xue; Zhang, Chun; Gao, Li-Xin; Liu, Min -Min; Yang, Yu-Ting; Yu, Li-Jie; Zhou, Yu-Bo; Milaneh, Slieman; Zhu, Yun-Long; Li, Jia; Wang, Wen-Long
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收藏Synthesis and Biological Evaluation of 3-Amino-4,4-Dimethyl Lithocholic Acid Derivatives as Novel, Selective, and Cellularly Active Allosteric SHP1 Activators
Chen, Huiqing; Liu, Zekun; Gao, Lixin; Yu, Li-Fang; Zhou, Yubo; Tang, Jie; Li, Jia; Yang, Fan
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收藏High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitorsSARS-CoV-2主要和木瓜蛋白酶类蛋白酶抑制剂的高通量筛选
Zang, Yi; Su, Mingbo; Wang, Qingxing; Cheng, Xi; Zhang, Wenru; Zhao, Yao; Chen, Tong; Jiang, Yingyan; Shen, Qiang; Du, Juan; Tan, Qiuxiang; Wang, Peipei; Gao, Lixin; Jin, Zhenming; Zhang, Mengmeng; Li, Cong; Zhu, Ya; Feng, Bo; Tang, Bixi; Xie, Han; Wang, Ming-Wei; Zheng, Mingyue; Pan, Xiaoyan; Yang, Haitao; Xu, Yechun; Wu, Beili; Zhang, Leike; Rao, Zihe; Yang, Xiuna; Jiang, Hualiang; Xiao, Gengfu; Zhao, Qiang; Li, Jia
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