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收藏Fused in silico and bioactivity evaluation method for drug discovery: T001-10027877 was identified as an antiproliferative agent that targets EGFRT790M/C797S/L858R and EGFRT790M/L858R
Wang, Linxiao; Huang, Xiaoling; Xu, Shidi; An, Yufeng; Lv, Xinya; Zhu, Wufu; Xu, Shan; Tu, Yuanbiao; Chen, Shuhui; Lv, Qiaoli; Zheng, Pengwu
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收藏In silico method and bioactivity evaluation to discover novel antimicrobial agents targeting FtsZ protein: Machine learning, virtual screening and antibacterial mechanism study
Wang, Linxiao; Xie, Zhouling; Ruan, Wei; Lan, Feixiang; Qin, Qi; Tu, Yuanbiao; Zhu, Wufu; Zhao, Jing; Zheng, Pengwu
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收藏Space-confined nanozyme with cascade reaction based on PCN-224 for synergistic bacterial infection treatment and NIR fluorescence imaging of wound bacterial infections
Lai, Luogen; Guo, Qiuyan; Zou, Wanqing; Huang, Liangxiao; Xu, Shan; Qiao, Dan; Wang, Linxiao; Zheng, Pengwu; Pan, Qingshan; Zhu, Wufu
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收藏Based on virtual screening methods and biological activity assessment, AK-968/13030056 has been identified as a potential mTOR inhibitor
Yang, Yang; Peng, Rujue; Cheng, Zhenjie; Yu, Mengting; Fu, Li; Zhang, Xufei; Zheng, Pengwu; Zhu, Wufu; Wang, Linxiao; Xu, Shan
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收藏Design, synthesis, and biological evaluation of 4-(2-fluorophenoxy)-7-methoxyquinazoline derivatives as dual EGFR/ c-Met inhibitors for the treatment of NSCLC
Tang, Sheng; Sun, Chuanchuan; He, Xintao; Gan, Wenhui; Wang, Linxiao; Qiao, Dan; Guan, Xinyu; Xu, Shan; Zheng, Pengwu; Zhu, Wufu
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收藏Design, synthesis and biological evaluation of 4-(4-aminophenoxy) picolinamide derivatives as potential antitumor agents
Dai, Jintian; Zhang, Jianqing; Fu, Dongxue; Liu, Meng; Zhang, Han; Tang, Sheng; Wang, Linxiao; Xu, Shan; Zhu, Wufu; Tang, Qidong; Zheng, Pengwu; Chen, Ting
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收藏Synthesis and antiproliferative activity of 6,7-disubstituted-4-phenoxyquinoline derivatives bearing the 1,8-naphthyridin-2-one moiety
Tang, Qidong; Duan, Yongli; Xiong, Hehua; Chen, Ting; Xiao, Zhen; Wang, Linxiao; Xiao, Yueyue; Huang, Shunmin; Xiong, Yinhua; Zhu, Wufu; Gong, Ping; Zheng, Pengwu
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收藏Discovery of novel pyrrolopyrimidine/pyrazolopyrimidine derivatives bearing 1,2,3-triazole moiety as c-Met kinase inhibitors
Wang, Linxiao; Liu, Xiaobo; Duan, Yongli; Li, Xiaojing; Zhao, Bingbing; Wang, Caolin; Xiao, Zhen; Zheng, Pengwu; Tang, Qidong; Zhu, Wufu
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收藏Synthesis and bioevaluation study of novel N-methylpicolinamide and thienopyrimidine derivatives as selectivity c-Met kinase inhibitors
Wang, Linxiao; Xu, Shan; Chen, Xiuying; Liu, Xiaobo; Duan, Yongli; Kong, Dejia; Zhao, Dandan; Zheng, Pengwu; Tang, Qidong; Zhu, Wufu
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收藏Synthesis and antiproliferative activity of pyrrolo[2,3-b]pyridine derivatives bearing the 1,8-naphthyridin-2-one moiety
Tang, Qidong; Duan, Yongli; Wang, Linxiao; Wang, Min; Ouyang, Yiqiang; Wang, Caolin; Mei, Han; Tang, Sheng; Xiong, Yinhua; Zheng, Pengwu; Gong, Ping; Zhu, Wufu
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