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Identification of furo[2,3-d]pyrimidin-4-ylsulfanyl-1,3,4-thiadiazole derivatives as novel FLT3-ITD inhibitors Moradi, Mahfam; Mousavi, Alireza; Reznickova, Eva; Peytam, Fariba; Perina, Miroslav; Vojackova, Veronika; Firoozpour, Loghman; Jorda, Radek; Gruz, Jiri; Emamgholipour, Zahra; Sadat-Ebrahimi, Seyed Esmaeil; Krystof, Vladimir; Foroumadi, Alireza 分享 收藏
Synthesis and photo-induced anticancer activity of new 2-phenylethenyl-1H-benzo[e]indole dyes Varvuolyte, Gabriele; Reznickova, Eva; Krikstole, Sonata; Tamuliene, Rasa; Bieliauskas, Aurimas; Malina, Lukas; Vojackova, Veronika; Duben, Zdenko; Kolarova, Hana; Kleiziene, Neringa; Arbaciauskiene, Egle; Zukauskaite, Asta; Krystof, Vladimir; Sackus, Algirdas 分享 收藏
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New Inhibitors of Bcr-Abl Based on 2,6,9-Trisubstituted Purine Scaffold Elicit Cytotoxicity in Chronic Myeloid Leukemia-Derived Cell Lines Sensitive and Resistant to TKIs 基于2,6,9-三取代嘌呤支架的新型bcr-abl抑制剂在对TKIs敏感和耐药的慢性粒细胞白血病衍生细胞系中引起细胞毒性 Delgado, Thalia; Vesela, Denisa; Dostalova, Hana; Krystof, Vladimir; Vojackova, Veronika; Jorda, Radek; Castro, Alejandro; Bertrand, Jeanluc; Rivera, Gildardo; Faundez, Mario; Strnad, Miroslav; Espinosa-Bustos, Christian; Salas, Cristian O. 分享 收藏
Cyclin dependent kinase 4/6 inhibitor palbociclib synergizes with BCL2 inhibitor venetoclax in experimental models of mantle cell lymphoma without RB1 deletion 细胞周期蛋白依赖性激酶4/6抑制剂palbociclib与BCL2抑制剂venetoclax在无RB1缺失的套细胞淋巴瘤实验模型中协同作用 Malarikova, Diana; Jorda, Radek; Kupcova, Kristyna; Senavova, Jana; Dolnikova, Alexandra; Pokorna, Eva; Kazantsev, Dmitry; Nozickova, Kristina; Sovilj, Dana; Bellanger, Celine; Chiron, David; Andera, Ladislav; Krystof, Vladimir; Strnad, Miroslav; Helman, Karel; Klanova, Magdalena; Trneny, Marek; Havranek, Ondrej; Klener, Pavel 分享 收藏
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Design and synthesis of novel 1,2,4-triazolo[4,3-b]pyridazine derivatives with anti-cancer activity 具有抗癌活性的新型1,2,4-三唑并 [4,3-b] 哒嗪衍生物的设计与合成 Ganai, Ab Majeed; Pathan, Tabasum Khan; Mohite, Sachin Balaso; Vojackova, Veronika; Reznickova, Eva; Kozlanska, Karolina; Krystof, Vladimir; Govender, Katya; Mokoena, Sithabile; Merugu, Srinivas Reddy; Palkar, Mahesh; Moodley, Kimeshni; Karpoormath, Rajshekhar 分享 收藏
2,4-Diaryl-pyrimido[1,2-a]benzimidazole derivatives as novel anticancer agents endowed with potent anti-leukemia activity: Synthesis, biological evaluation and kinase profiling 2,4-二芳基-嘧啶并 [1,2-a] 苯并咪唑衍生物作为具有有效抗白血病活性的新型抗癌剂: 合成,生物学评估和激酶谱 Shaldam, Moataz A.; Hendrychov, Denisa; El-Haggar, Radwan; Voj, Veronika; Majrashi, Taghreed A.; Elkaeed, Eslam B.; Masurier, Nicolas; Krystof, Vladimir; Tawfik, Haytham O.; Eldehna, Wagdy M. 分享 收藏
Inhibition of FLT3-ITD Kinase in Acute Myeloid Leukemia by New Imidazo[1,2-b]pyridazine Derivatives Identified by Scaffold Hopping Brehova, Petra; Reznickova, Eva; Skach, Krystof; Jorda, Radek; Dejmek, Milan; Vojackova, Veronika; Sala, Michal; Kovalova, Marketa; Dracinsky, Martin; Dolnikova, Alexandra; Strmen, Timotej; Kinnertova, Monika; Chalupsky, Karel; Dvorakova, Alexandra; Gucky, Tomas; Kaiserova, Helena Mertlikova; Klener, Pavel; Nencka, Radim; Krystoy, Vladimir 分享 收藏
Characterization of new highly selective pyrazolo[4,3-d]pyrimidine inhibitor of CDK7 Kovalova, Marketa; Havlicek, Libor; Djukic, Stefan; Skerlova, Jana; Perina, Miroslav; Pospisil, Tomas; Reznickova, Eva; Rezacova, Pavlina; Jorda, Radek; Krystof, Vladimir 分享 收藏
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