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Andrew V. Stachulski

University of Liverpool

32H指数
178论文数
3.0K被引数
收录论文 44
发表时间
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Small but powerful小巧但功能强大
err2025-11-04
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PREAI
errAndrew V. Stachulski; Christopher J. Schofield
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Dynamic kinetic resolution-mediated synthesis of C-3 hydroxylated arginine derivatives动力学拆分介导的C-3羟基化精氨酸衍生物合成
err2025-02-19
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errOAAI
errZheng, Ye; Chen, Zhenyu; Clarkson, Guy J.; Marshall, Stephen A.; Xiao, Jianliang; Schofield, Christopher J.; Wills, Martin; Stachulski, Andrew V.
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Synthetic β-d-Glucuronides: Substrates for Exploring Glucuronide Degradation by Human Gut Bacteria
err2024-12-20
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errOAAI
errGorecka, Aleksandra; Schacht, Heidi; Fraser, Megan K.; Teriosina, Aleksandra; London, James A.; Barsukov, Igor L.; Powell, Andrew K.; Cartmell, Alan; Stachulski, Andrew V.; Yates, Edwin A.
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Cerebrovascular damage caused by the gut microbe/host co-metabolite p-cresol sulfate is prevented by blockade of the EGF receptor
err2024-11-24
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errOAAI
errShah, Sita N.; Knausenberger, Tobias B-A.; Pontifex, Matthew G.; Connell, Emily; Le Gall, Gwenaelle; Hardy, Tom A. J.; Randall, David W.; Mccafferty, Kieran; Yaqoob, Muhammad M.; Solito, Egle; Mueller, Michael; Stachulski, Andrew V.; Glen, Robert C.; Vauzour, David; Hoyles, Lesley; Mcarthur, Simon
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Transacylation and hydrolysis of the acyl glucuronides of ibuprofen and its α-methyl-substituted analogues investigated by 1 H NMR spectroscopy and computational chemistry: Implications for drug design
err2024-08-01
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errOAAI
errRichards, Selena E.; Bradshaw, Peter R.; Johnson, Caroline H.; V. Stachulski, Andrew; Athersuch, Toby J.; Nicholson, Jeremy K.; Lindon, John C.; Wilson, Ian D.
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Thiazolide Prodrug Esters and Derived Peptides: Synthesis and Activity噻唑化物前体酯和衍生肽: 合成和活性
err2023-04-11
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errOAAI
errStachulski, Andrew V.; Rossignol, Jean-Francois; Pate, Sophie; Taujanskas, Joshua; Iggo, Jonathan A.; Aerts, Rudi; Pascal, Etienne; Piacentini, Sara; La Frazia, Simone; Santoro, M. Gabriella; van Vooren, Lieven; Sintubin, Liesje; Cooper, Mark; Swift, Karl; O'Neill, Paul M.
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A host-gut microbial amino acid co-metabolite, p-cresol glucuronide, promotes blood-brain barrier integrity in vivo
err2022-05-20
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errOAAI
errStachulski, Andrew, V; Knausenberger, Tobias B-A; Shah, Sita N.; Hoyles, Lesley; McArthur, Simon
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Synthesis, antiviral activity, preliminary pharmacokinetics and structural parameters of thiazolide amine salts
err2021-08-17
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PREAI
errStachulski, Andrew, V; Rossignol, Jean-Francois; Pate, Sophie; Taujanskas, Joshua; Robertson, Craig M.; Aerts, Rudi; Pascal, Etienne; Piacentini, Sara; Frazia, Simone La; Santoro, M. Gabriella; O'Neill, Paul M.
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Discovery and Optimization of a 4-Aminopiperidine Scaffold for Inhibition of Hepatitis C Virus Assembly
err2021-06-29
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errRolt, Adam; Talley, Daniel C.; Park, Seung Bum; Hu, Zongyi; Dulcey, Andres; Ma, Christopher; Irvin, Parker; Leek, Madeleine; Wang, Amy Q.; Stachulski, Andrew, V; Xu, Xin; Southall, Noel; Ferrer, Marc; Liang, T. Jake; Marugan, Juan J.
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Therapeutic Potential of Nitazoxanide: An Appropriate Choice for Repurposing versus SARS-CoV-2?硝唑尼特的治疗潜力: 再利用与SARS-CoV-2的合适选择?
err2020-12-22
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errStachulski, Andrew, V; Taujanskas, Joshua; Pate, Sophie L.; Rajoli, Rajith K. R.; Aljayyoussi, Ghaith; Pennington, Shaun H.; Ward, Stephen A.; Hong, Weiqian David; Biagini, Giancarlo A.; Owen, Andrew; Nixon, Gemma L.; Leung, Suet C.; O'Neill, Paul M.
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Acyl glucuronide reactivity in perspective
err2020-09-01
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errOAAI
errBradshaw, Peter R.; Athersuch, Toby J.; Stachulski, Andrew, V; Wilson, Ian D.
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Second-generation nitazoxanide derivatives: thiazolides are effective inhibitors of the influenza A virus
err2018-04-09
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errStachulski, Andrew V.; Santoro, M. Gabriella; Piacentini, Sara; Belardo, Giuseppe; La Frazia, Simone; Pidathala, Chandrakala; Row, Eleanor C.; Berry, Neil G.; Iqbal, Mazhar; Allman, Sarah A.; Semple, J. Edward; Eklov, Brian M.; O'Neill, Paul M.; Rossignol, Jean-Francois
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Rational Design, Synthesis, and Biological Evaluation of Heterocyclic Quinolones Targeting the Respiratory Chain of Mycobacterium tuberculosis
err2017-04-25
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errHong, W. David; Gibbons, Peter D.; Leung, Suet C.; Amewu, Richard; Stocks, Paul A.; Stachulski, Andrew; Horta, Pedro; Cristiano, Maria L. S.; Shone, Alison E.; Moss, Darren; Ardrey, Alison; Sharma, Raman; Warman, Ashley J.; Bedingfield, Paul T. P.; Fisher, Nicholas E.; Aljayyoussi, Ghaith; Mead, Sally; Caws, Maxine; Berry, Neil G.; Ward, Stephen A.; Biagini, Giancarlo A.; O'Neill, Paul M.; Nixon, Gemma L.
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Synthesis and pre-clinical studies of new amino-acid ester thiazolide prodrugs
err2017-01-01
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errOAAI
errStachulski, Andrew V.; Swift, Karl; Cooper, Mark; Reynolds, Stephen; Norton, Daniel; Slonecker, Steven D.; Rossignol, Jean-Francois
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Mass Spectrometric Characterization of Circulating Covalent Protein Adducts Derived from a Drug Acyl Glucuronide Metabolite: Multiple Albumin Adductions in Diclofenac Patients
err2014-06-01
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errOAAI
errHammond, Thomas G.; Meng, Xiaoli; Jenkins, Rosalind E.; Maggs, James L.; Castelazo, Anahi Santoyo; Regan, Sophie L.; Bennett, Stuart N. L.; Earnshaw, Caroline J.; Aithal, Guruprasad P.; Pande, Ira; Kenna, J. Gerry; Stachulski, Andrew V.; Park, B. Kevin; Williams, Dominic P.
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Dissecting the reaction of Phase II metabolites of ibuprofen and other NSAIDS with human plasma protein
err2014-01-01
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PREAI
errMonrad, Rune Nygaard; Errey, James C.; Barry, Conor S.; Iqbal, Mazhar; Meng, Xiaoli; Iddon, Lisa; Perrie, Jennifer A.; Harding, John R.; Wilson, Ian D.; Stachulski, Andrew V.; Davis, Benjamin G.
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Activation of carbamazepine-responsive T-cell clones with metabolically inert halogenated derivatives
err2013-08-01
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PREAI
errFarrell, John; Lichtenfels, Maike; Sullivan, Andrew; Elliott, Emma C.; Alfirevic, Ana; Stachulski, Andrew V.; Pirmohamed, Munir; Naisbitt, Dean J.; Park, B. Kevin
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