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Gamal El‐Din A. Abuo‐Rahma

Shaqra University

35H指数
135论文数
3.8K被引数
收录论文 42
发表时间
A review of recent advances in anticancer activity and SAR of pyrazole derivatives近期吡唑衍生物抗肿瘤活性及构效关系研究进展
err2025-03-17
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PREAI
errHofny, Heba A.; Mohamed, Mamdouh F. A.; Hassan, Heba A.; Abdelhafez, El-Shimaa M. N.; Abuo-Rahma, Gamal El-Din A.
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Unveiling the Anticancer Potential of a New Ciprofloxacin-Chalcone Hybrid as an Inhibitor of Topoisomerases I & II and Apoptotic Inducer
err2024-11-15
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errOAAI
errAli, Doaa Mohamed Elroby; Aziz, Hossameldin A.; Brase, Stefan; Al Bahir, Areej; Alkhammash, Abdullah; Abuo-Rahma, Gamal El-Din A.; Elshamsy, Ali M.; Hashem, Hamada; Abdelmagid, Walid M.
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Design, synthesis and mechanistic study of N-4-Piperazinyl Butyryl Thiazolidinedione derivatives of ciprofloxacin with Anticancer Activity via Topoisomerase I/II inhibition
err2024-10-15
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errOAAI
errAziz, Hossameldin A.; El-Saghier, Ahmed M.; Badr, Mohamed; Elsadek, Bakheet E. M.; Abuo-Rahma, Gamal El-Din A.; Shoman, Mai E.
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Synthesis, characterization, molecular docking, and antimicrobial activities of some new sulfur containing norfloxacin analogues
err2024-07-01
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PREAI
errEl-Saghier, Ahmed M. M.; Abosella, Laila; Elakesh, Esmail O.; Abuo-Rahma, Gamal El -Din A.; Abdou, Aly; Hamed, Amany M.
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Design, synthesis and mechanistic study of new dual targeting HDAC/tubulin inhibitors
err2024-03-04
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errEl-Zoghbi, Mona S.; Bass, Amr K. A.; Abuo-Rahma, Gamal El-Din; Mohamed, Mamdouh F. A.; Badr, Mohamed; AL-Ghulikah, Hanan A.; Abdelhafez, El-Shimaa M. N.
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Ciprofloxacin Derivative-Loaded Nanoparticles Synergize with Paclitaxel Against Type II Human Endometrial Cancer环丙沙星衍生物纳米粒与紫杉醇协同治疗II型人子宫内膜癌
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IF12.1
err2023-07-31
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errNaguib, Youssef W.; Alhaj-Suliman, Suhaila O.; Wafa, Emad I.; Saha, Sanjib; Ebeid, Kareem; Mohammed, Hamada H. H.; Abdel-Rahman, Somaya A.; Abuo-Rahma, Gamal El-Din A.; Geary, Sean M.; Salem, Aliasger K.
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A ciprofloxacin derivative with four mechanisms of action overcomes paclitaxel resistance in p53-mutant and MDR1 gene-expressing type II human endometrial cancer具有四种作用机制的环丙沙星衍生物克服了p53-mutant和MDR1基因表达的II型人类子宫内膜癌的紫杉醇耐药性
err2023-05-01
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errAlhaj-Suliman, Suhaila O.; Naguib, Youssef W.; Wafa, Emad I.; Saha, Sanjib; Ebeid, Kareem; Meng, Xiangbing; Mohammed, Hamada H.; Abuo-Rahma, Gamal El-Din A.; Yang, Shujie; Salem, Aliasger K.
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In Vitro Anticancer Activity of Novel Ciprofloxacin Mannich Base in Lung Adenocarcinoma and High-Grade Serous Ovarian Cancer Cell Lines via Attenuating MAPK Signaling Pathway
err2023-01-23
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errFawzy, Michael A.; Abu-baih, Rania H.; Abuo-Rahma, Gamal El-Din A.; Abdel-Rahman, Islam M.; El-Sheikh, Azza A. K.; Nazmy, Maiiada H.
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New s-Triazine/Tetrazole conjugates as potent antifungal and antibacterial agents: Design, molecular docking and mechanistic study
err2022-11-01
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PREAI
errMekheimer, Ramadan Ahmed; Abuo-Rahma, Gamal El -Din A.; Abd-Elmonem, Mohamed; Yahia, Ramadan; Hisham, Mohamed; Hayallah, Alaa M.; Mostafa, Sara M.; Abo-Elsoud, Fatma A.; Sadek, Kamal Usef
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Synthesis and molecular docking of new N4-piperazinyl ciprofloxacin hybrids as antimicrobial DNA gyrase inhibitors
err2022-09-24
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errOAAI
errMohammed, Hamada H. H.; Ali, Doaa Mohamed Elroby; Badr, Mohamed; Habib, Ahmed G. K.; Mahmoud, Abobakr Mohamed; Farhan, Sarah M.; Gany, Shimaa Salah Hassan Abd El; Mohamad, Soad A.; Hayallah, Alaa M.; Abbas, Samar H.; Abuo-Rahma, Gamal El-Din A.
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New 1,2,3-triazole linked ciprofloxacin-chalcones induce DNA damage by inhibiting human topoisomerase I& II and tubulin polymerization
err2022-05-11
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errMohammed, Hamada H. H.; Abd El-Hafeez, Amer Ali; Ebeid, Kareem; Mekkawy, Aml, I; Abourehab, Mohammed A. S.; Wafa, Emad, I; Alhaj-Suliman, Suhaila O.; Salem, Aliasger K.; Ghosh, Pradipta; Abuo-Rahma, Gamal El-Din A.; Hayallah, Alaa M.; Abbas, Samar H.
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Solulan C24- and Bile Salts-Modified Niosomes for New Ciprofloxacin Mannich Base for Combatting Pseudomonas-Infected Corneal Ulcer in Rabbits
err2021-12-29
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errMohamed, Soad A.; Abdelgawad, Mohamed A.; Alaaeldin, Rania; Fathalla, Zeinab; Moharram, Hossam; Abdallah, Raafat M. A.; Abdel-Rahman, Islam M.; Abdel-Aziz, Mohamed; Abuo-Rahma, Gamal El-Din A.; Ghoneim, Mohammed M.; Hayallah, Alaa M.; Elrehany, Mahmoud; Abdelkader, Hamdy
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New 4-thiazolidinone/quinoline-2-ones scaffold: Design, synthesis, docking studies and biological evaluation as potential urease inhibitors
err2021-11-01
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PREAI
errElbastawesy, Mohammed A., I; Aly, Ashraf A.; El-Shaier, Yaseen A. M. M.; Brown, Alan B.; Abuo-Rahma, Gamal El-Din A.; Ramadan, Mohamed
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New Multi-Targeted Antiproliferative Agents: Design and Synthesis of IC261-Based Oxindoles as Potential Tubulin, CK1 and EGFR Inhibitors
err2021-10-30
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errFareed, Momen R.; Shoman, Mai E.; Hamed, Mohammed I. A.; Badr, Mohamed; Bogari, Hanin A.; Elhady, Sameh S.; Ibrahim, Tarek S.; Abuo-Rahma, Gamal El-Din A.; Ali, Taha F. S.
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A first-in-class anticancer dual HDAC2/FAK inhibitors bearing hydroxamates/benzamides capped by pyridinyl-1,2,4-triazoles
err2021-10-01
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errMustafa, Muhamad; Abd El-Hafeez, Amer Ali; Abdelhamid, Dalia; Katkar, Gajanan D.; Mostafa, Yaser A.; Ghosh, Pradipta; Hayallah, Alaa M.; Abuo-Rahma, Gamal El-Din A.
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Thiazolidine-2,4-dione-linked ciprofloxacin derivatives with broad-spectrum antibacterial, MRSA and topoisomerase inhibitory activities
err2021-08-29
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PREAI
errAziz, Hossameldin A.; El-Saghier, Ahmed M. M.; Badr, Mohamed; Abuo-Rahma, Gamal El-Din A.; Shoman, Mai E.
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FAK inhibitors as promising anticancer targets: present and future directions
err2021-08-03
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errMustafa, Muhamad; Abd El-Hafeez, Amer Ali; Abdelhafeez, Dalia A.; Abdelhamid, Dalia; Mostafa, Yaser A.; Ghosh, Pradipta; Hayallah, Alaa M.; Abuo-Rahma, Gamal El-Din
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Novel 4-(piperazin-1-yl)quinolin-2(1H)-one bearing thiazoles with antiproliferative activity through VEGFR-2-TK inhibition
err2021-06-01
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PREAI
errHassan, Abdelfattah; Badr, Mohamed; Hassan, Heba A.; Abdelhamid, Dalia; Abuo-Rahma, Gamal El-Din A.
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