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Robert Milne

University of South Australia

42H指数
209论文数
7.4K被引数
收录论文 36
发表时间
A brain-penetrant CDK4/6 inhibitor - AU3-14 shows robust anti-tumor efficacy against glioblastoma一种能够穿透血脑屏障的CDK4/6抑制剂AU3-14显示出对胶质母细胞瘤的显著抗肿瘤效果。
err2025-07-11
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PREAI
errLaychiluh B. Mekonnen; Theodosia Teo; Benjamin Noll; Muhammed H. Rahaman; Jimma Lenjisa; Sunita Basnet; Ramin Hassankhani; Robert Milne; Briony L. Gliddon; Melinda N. Tea; Stuart M. Pitson; Yan Zhou; Lijun Wei; Hui Wang; Jun Liu; Xiang Zhou; Ke Wang; Shudong Wang
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AU2-94: A CDK4-specific inhibitor with the marked anti-tumor efficacy
err2024-03-22
err0
PREAI
errBantie, Laychiluh; Likisa, Jimma; Rahaman, Muhammed; Teo, Theodosia; Safaroghliazar, Ava; Basnet, Sunita K. C.; Hassankhani, Ramin; Noll, Benjamin; Milne, Robert; Wang, Shudong
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Liposomal 5-Fluorouracil Polymer Complexes Facilitate Tumor-Specific Delivery: Pharmaco-Distribution Kinetics Using Microdialysis
err2022-01-18
err7
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errWang, Wen; Joyce, Paul; Bremmell, Kristen; Milne, Robert; Prestidge, Clive A.
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CDK9: A Comprehensive Review of Its Biology, and Its Role as a Potential Target for Anti-Cancer Agents
err2021-05-10
err96
errOAAI
errAnshabo, Abel Tesfaye; Milne, Robert; Wang, Shudong; Albrecht, Hugo
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Potent and orally bioavailable CDK8 inhibitors: Design, synthesis, structure-activity relationship analysis and biological evaluation有效和口服可生物利用的CDK8抑制剂: 设计,合成,构效关系分析和生物学评估
err2021-03-01
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PREAI
errYu, Mingfeng; Teo, Theodosia; Yang, Yuchao; Li, Manjun; Long, Yi; Philip, Stephen; Noll, Benjamin; Heinemann, Gary K.; Diab, Sarah; Eldi, Preethi; Mekonnen, Laychiluh; Anshabo, Abel T.; Rahaman, Muhammed H.; Milne, Robert; Hayball, John D.; Wang, Shudong
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Targeting CDK9 for treatment of colorectal cancer
err2019-08-21
err40
errOAAI
errRahaman, Muhammed H.; Lam, Frankie; Zhong, Longjin; Teo, Theodosia; Adams, Julian; Yu, Mingfeng; Milne, Robert W.; Pepper, Chris; Lokman, Noor A.; Ricciardelli, Carmela; Oehler, Martin K.; Wang, Shudong
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Sulfonamide-Based Inhibitors of Biotin Protein Ligase as New Antibiotic Leads
err2019-08-13
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PREAI
errLee, Kwang Jun; Tieu, William; Blanco-Rodriguez, Beatriz; Paparella, Ashleigh S.; Yu, Jingxian; Hayes, Andrew; Feng, Jiage; Marshall, Andrew C.; Noll, Benjamin; Milne, Robert; Cini, Danielle; Wilce, Matthew C. J.; Booker, Grant W.; Bruning, John B.; Polyak, Steven W.; Abell, Andrew D.
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LS007, a potent and orally bioavailable CDK9 inhibitor, suppresses the growth of triple-negative and estrogen receptor-positive breast cancer
err2019-07-01
err0
PREAI
errRahaman, Muhammed Hamidur; Zhang, Yinghui; Islam, Md Saiful; Heinemann, Gary; Anshabo, Abel Tesfaye; Albrecht, Hugo; Milne, Robert; Wang, Shudong
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Discovery of CDK5 Inhibitors through Structure-Guided Approach
err2019-03-20
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errKhair, Nishat Z.; Lenjisa, Jimma L.; Tadesse, Solomon; Kumarasiri, Malika; Basnet, Sunita K. C.; Mekonnen, Laychiluh B.; Li, Manjun; Diab, Sarah; Sykes, Matthew J.; Albrecht, Hugo; Milne, Robert; Wang, Shudong
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CDKI-73: an orally bioavailable and highly efficacious CDK9 inhibitor against acute myeloid leukemia
err2018-09-08
err30
PREAI
errRahaman, Muhammed H.; Yu, Yingyi; Zhong, Longjin; Adams, Julian; Lam, Frankie; Li, Peng; Noll, Ben; Milne, Robert; Peng, Jun; Wang, Shudong
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A first-in-class CDK4 inhibitor shows excellent in vitro and in vivo efficacy against ovarian cancer
err2018-07-01
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PREAI
errMekonnen, Laychiluh B.; Zeleke, Solomon; Lenjisa, Jimma; Yu, Mingfeng; Noll, Benjamin; Heinemann, Gary; Milne, Robert; Albrecht, Hugo; Oehler, Martin K.; Wang, Shudong
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Preclinical development of a highly potent and selective dual inhibitor of CDK4/6 for the treatment of cancer
err2018-07-01
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PREAI
errBantie, Laychiluh; Tadesse, Solomon; Likisa, Jimma; Yu, Mingfeng; Noll, Benjamin; Albrecht, Hugo; Milne, Robert; Wang, Shudong
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Discovery and pharmacological characterization of a novel series of highly selective inhibitors of cyclin-dependent kinases 4 and 6 as anticancer agents
err2018-05-08
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errTadesse, Solomon; Bantie, Laychiluh; Tomusange, Khamis; Yu, Mingfeng; Islam, Saiful; Bykovska, Nataliya; Noll, Benjamin; Zhu, Ge; Li, Peng; Lam, Frankie; Kumarasiri, Malika; Milne, Robert; Wang, Shudong
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CDK5 in oncology: recent advances and future prospects
err2017-10-27
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errLenjisa, Jimma Likisa; Tadesse, Solomon; Khair, Nishat Zareen; Kumarasiri, Malika; Yu, Mingfeng; Albrecht, Hugo; Milne, Robert; Wang, Shudong
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Dual Inhibition of Mnk2 and FLT3 for potential treatment of acute myeloid leukaemia
err2017-10-01
err22
PREAI
errDiab, Sarah; Abdelaziz, Ahmad M.; Li, Peng; Teo, Theodosia; Basnet, Sunita K. C.; Noll, Ben; Rahaman, Muhammed H.; Lu, Jingfeng; Hou, Jinqiang; Yu, Mingfeng; Le, Bich T.; Albrecht, Hugo; Milne, Robert W.; Wang, Shudong
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The association between total phthalate concentration and non-communicable diseases and chronic inflammation in South Australian urban dwelling men
err2017-10-01
err41
PREAI
errBai, Peter Y.; Wittert, Gary; Taylor, Anne W.; Martin, Sean A.; Milne, Robert W.; Jenkins, Alicia J.; Januszewski, Andrzej S.; Shi, Zumin
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Highly Potent, Selective, and Orally Bioavailable 4-Thiazol-N-(pyridin-2-yl)pyrimidin-2-amine Cyclin-Dependent Kinases 4 and 6 Inhibitors as Anticancer Drug Candidates: Design, Synthesis, and Evaluation
err2017-02-16
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errOAAI
errTadesse, Solomon; Yu, Mingfeng; Mekonnen, Laychiluh B.; Lam, Frankie; Islam, Saiful; Tomusange, Khamis; Rahaman, Muhammed H.; Noll, Benjamin; Basnet, Sunita K. C.; Teo, Theodosia; Albrecht, Hugo; Milne, Robert; Wang, Shudong
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Targeting CDK9: a promising therapeutic opportunity in prostate cancer靶向CDK9: 前列腺癌的一个有希望的治疗机会
err2016-12-01
err59
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errRahaman, Muhammed H.; Kumarasiri, Malika; Mekonnen, Laychiluh B.; Yu, Mingfeng; Diab, Sarah; Albrecht, Hugo; Milne, Robert W.; Wang, Shudong
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Unveiling new chemical scaffolds as Mnk inhibitors
err2016-02-24
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PREAI
errDiab, Sarah; Li, Peng; Basnet, Sunita K. C.; Lu, Jingfeng; Yu, Mingfeng; Albrecht, Hugo; Milne, Robert W.; Wang, Shudong
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Targeting Pim kinases for cancer treatment: opportunities and challenges
err2015-01-13
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PREAI
errLe, Bich Thuy; Kumarasiri, Malika; Adams, Julian R. J.; Yu, Mingfeng; Milne, Robert; Sykes, Matthew J.; Wang, Shudong
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