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Petro Borysko

enamine ltd

19H指数
120论文数
1.1K被引数
收录论文 39
发表时间
Bench-Stable α-Fluoroamines: Synthesis, Properties, and Application in Medicinal Chemistry台架稳定的α-氟代胺:合成、性质及其在药物化学中的应用
err2026-10-07
err0
PREAI
errVadym Levterov; Oleh Shablykin; Oleksandr Stashkevych; Volodymyr Kokhalskyi; Vadym Konashuk; Iryna Sadkova; Olha Shevchuk; Petro Borysko; Henry S. Rzepa; Pavel K. Mykhailiuk
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Bicyclic 1,4-Dioxepanes for Drug Discovery: Multigram Synthesis, Physicochemical, and Structural Characterization
err2025-12-01
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PREAI
errBondarenko, Andrii V.; Kozyriev, Yevhenii; Doroshenko, Illia O.; Lesyk, Dmytro; Borysko, Petro; Shishkina, Svetlana V.; Vashchenko, Bohdan V.; Grygorenko, Oleksandr O.
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Synthesis and Physicochemical Characterization of 5-Trifluoromethyl-Substituted Tetrahydrofurans and Tetrahydrothiophenes5-三氟甲基取代四氢呋喃和四氢噻吩的合成与物理化学表征
err2025-12-01
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errOAAI
errRedka, Mykhailo O.; Dovhaniuk, Nazar; Blahun, Oleksandr; Liashuk, Oleksandr S.; Hurieva, Anastasiia M.; Lesyk, Dmytro; Skrypnik, Daniil; Holota, Yuliia; Durylin, Dmytro; Borysko, Petro; Kondratov, Ivan S.; Grygorenko, Oleksandr O.
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Gram-scale synthesis and physicochemical properties of exo- and endo-5,5-difluorooctahydropentalen-2-amines
err2025-10-01
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PREAI
errVoloshyna, Olena; Moroz, Bohdan; Melnykov, Kostiantyn P.; Holovach, Serhii; Lesyk, Dmytro; Holota, Yuliia; Borysko, Petro; Filatov, Andrey A.; Grygorenko, Oleksandr O.
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Basicity and Lipophilicity of gem-Difluorinated Saturated Bicyclic Amines: Advanced Building Blocks for Drug Discovery碱性和脂溶性:gem-二氟代饱和双环胺:药物发现中的先进构建模块
err2025-09-09
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PREAI
errOleksandr S. Liashuk; Bohdan Moroz; Kostiantyn P. Melnykov; Serhii Holovach; Dmytro Lesyk; Yaroslav Lesyk; Daniil Skrypnik; Yuliia Holota; Petro Borysko; Andrey A. Filatov; Oleksandr O. Grygorenko
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Synthesis and Physicochemical Properties of Functionalized cis–2-((Fluoro)Alkyl)Cyclobutanes功能化顺式-2-((氟)烷基)环丁烷的合成与物理化学性质
err2025-07-09
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PREAI
errAnton V. Chernykh; Oleksandr S. Liashuk; Kyrylo O. Kononenko; Artem Y. Michuda; Oleksandr S. Olifir; Dmytro Lesyk; Karina Turenko; Andrii V. Kozytskyi; Svitlana V. Shishkina; Petro Borysko; Serhiy V. Ryabukhin; Dmytro M. Volochnyuk; Oleksandr O. Grygorenko
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In vitro evaluation of the immunogenic potential of gramicidin S and its photocontrolled analogues体外评价gramicidin S及其光控类似物的免疫原性潜力
err2025-01-01
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errOAAI
errHorbatok, Kateryna; Semchuk, Iryna; Horbach, Oleksandr; Khranovska, Natalia; Kosach, Viktoriia; Borysko, Petro; Koniev, Serhii; Ulrich, Anne S.; Afonin, Sergii; Komarov, Igor V.
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Physicochemical and Biological Evaluation of gem-Difluorinated Saturated Oxygen Heterocycles as Bioisosteres for Drug Discovery
err2024-12-18
err1
PREAI
errMelnykov, Kostiantyn P.; Liashuk, Oleksandr S.; Holovach, Serhii; Shatnia, Valeriia; Horbenko, Artur; Lesyk, Dmytro; Melnyk, Varvara; Skrypnik, Daniil; Beshtynarska, Anna; Borysko, Petro; Viniichuk, Oleksandr; Grygorenko, Oleksandr O.
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Angular Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery
err2024-12-12
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errOAAI
errKirichok, Alexander A.; Tkachuk, Hennadii; Levchenko, Kostiantyn; Granat, Dmitry; Yegorova, Tetyana; Lesyk, Dmytro; Anisiforova, Anna; Holota, Yuliia; Zomchak, Viktoriia; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Korzh, Rodion A.; Al-Maali, Galeb; Kubyshkin, Vladimir; Rzepa, Henry S.; Mykhailiuk, Pavel K.
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CF3-Cyclobutanes: Synthesis, Properties, and Evaluation as a Unique tert-Butyl Group AnalogueCF3-Cyclobutanes: 独特的叔丁基类似物的合成,性质和评价
errJACS AU
IF8.7
err2024-11-11
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errOAAI
errAhunovych, Volodymyr; Klipkov, Anton A.; Bugera, Maksym; Tarasenko, Karen; Trofymchuk, Serhii; Razhyk, Bohdan; Boretskyi, Andrii; Stanko, Oleh; Panasiuk, Yaroslav; Shablykin, Oleh; Al-Maali, Galeb; Lesyk, Dmytro; Klymenko-Ulianov, Oleksii; Horbatok, Kateryna; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Kubyshkin, Vladimir; Mykhailiuk, Pavel K.
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3,3-Difluorooxetane-A Versatile Functional Group for Bioisosteric Replacements in Drug Discovery
err2024-10-31
err1
PREAI
errLiashuk, Oleksandr S.; Fedinchyk, Anastasiya; Melnykov, Kostiantyn P.; Herasymchuk, Maksym; Alieksieieva, Diana; Lesyk, Dmytro; Bas, Yuliia P.; Keda, Tetiana Ye.; Yatsymyrskiy, Andriy V.; Holota, Yuliia; Borysko, Petro; Yarmolchuk, Volodymyr S.; Grygorenko, Oleksandr O.
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2-Oxabicyclo[2.1.1]hexanes: Synthesis, Properties, and Validation as Bioisosteres of ortho- and meta-Benzenes2-氧杂双环 [2.1.1] 己烷: 邻苯和间苯的生物电子等排体的合成,性质和验证
err2024-04-03
err13
errOAAI
errLevterov, Vadym V.; Panasiuk, Yaroslav; Shablykin, Oleh; Stashkevych, Oleksandr; Sahun, Kateryna; Rassokhin, Artur; Sadkova, Iryna; Lesyk, Dmytro; Anisiforova, Anna; Holota, Yuliia; Borysko, Petro; Bodenchuk, Iryna; Voloshchuk, Nataliya M.; Mykhailiuk, Pavel K.
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Anticancer activity features of imidazole-based ionic liquids and lysosomotropic detergents: in silico and in vitro studies
err2024-01-22
err1
PREAI
errGryniukova, Anastasiia; Borysko, Petro; Myziuk, Iryna; Alieksieieva, Diana; Hodyna, Diana; Semenyuta, Ivan; Kovalishyn, Vasyl; Metelytsia, Larysa; Rogalsky, Sergiy; Tcherniuk, Sergey
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Spiro[3.3]heptane as a Saturated Benzene Bioisostere螺 [3.3] 庚烷作为饱和苯生物电子等排物
err2024-01-22
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errOAAI
errPrysiazhniuk, Kateryna; Datsenko, Oleksandr P.; Polishchuk, Oleksandr; Shulha, Stanislav; Shablykin, Oleh; Nikandrova, Yelyzaveta; Horbatok, Kateryna; Bodenchuk, Iryna; Borysko, Petro; Shepilov, Dmytro; Pishel, Iryna; Kubyshkin, Vladimir; Mykhailiuk, Pavel K.
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2-Oxabicyclo[2.2.2]octane as a new bioisostere of the phenyl ring
err2023-10-02
err18
errOAAI
errLevterov, Vadym V.; Panasiuk, Yaroslav; Sahun, Kateryna; Stashkevych, Oleksandr; Badlo, Valentyn; Shablykin, Oleh; Sadkova, Iryna; Bortnichuk, Lina; Klymenko-Ulianov, Oleksii; Holota, Yuliia; Lachmann, Leonid; Borysko, Petro; Horbatok, Kateryna; Bodenchuk, Iryna; Bas, Yuliia; Dudenko, Dmytro; Mykhailiuk, Pavel K.
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Hydroaminoalkyl Functionalization of Pyrimidin-2(1H)-ones by Visible Light Organophotocatalysis: A Radical Approach to Biginelli-Type Dihydropyrimidines
err2023-09-06
err2
PREAI
errLukianov, Oleh; Tkachuk, Viktor; Shishkina, Svitlana; Lachmann, Leonid; Vadzyuk, Olga; Borysko, Petro; Kovalskyy, Dmytro; Gillaizeau, Isabelle; Sukach, Volodymyr
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AI-Powered Virtual Screening of Large Compound Libraries Leads to the Discovery of Novel Inhibitors of Sirtuin-1
err2023-07-27
err12
PREAI
errGryniukova, Anastasiia; Kaiser, Florian; Myziuk, Iryna; Alieksieieva, Diana; Leberecht, Christoph; Heym, Peter P.; Tarkhanova, Olga O.; Moroz, Yurii S.; Borysko, Petro; Haupt, V. Joachim
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Anionic amphiphilic calixarenes for peptide assembly and delivery
err2022-10-01
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errOAAI
errRodik, Roman V.; Cherenok, Sergiy O.; Postupalenko, Viktoriia Y.; Oncul, Sule; Brusianska, Vladyslava; Borysko, Petro; Kalchenko, Vitaly I.; Mely, Yves; Klymchenko, Andrey S.
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