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Bicyclic 1,4-Dioxepanes for Drug Discovery: Multigram Synthesis, Physicochemical, and Structural Characterization Bondarenko, Andrii V.; Kozyriev, Yevhenii; Doroshenko, Illia O.; Lesyk, Dmytro; Borysko, Petro; Shishkina, Svetlana V.; Vashchenko, Bohdan V.; Grygorenko, Oleksandr O. 分享 收藏
Synthesis and Physicochemical Characterization of 5-Trifluoromethyl-Substituted Tetrahydrofurans and Tetrahydrothiophenes 5-三氟甲基取代四氢呋喃和四氢噻吩的合成与物理化学表征 Redka, Mykhailo O.; Dovhaniuk, Nazar; Blahun, Oleksandr; Liashuk, Oleksandr S.; Hurieva, Anastasiia M.; Lesyk, Dmytro; Skrypnik, Daniil; Holota, Yuliia; Durylin, Dmytro; Borysko, Petro; Kondratov, Ivan S.; Grygorenko, Oleksandr O. 分享 收藏
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Gram-scale synthesis and physicochemical properties of exo- and endo-5,5-difluorooctahydropentalen-2-amines Voloshyna, Olena; Moroz, Bohdan; Melnykov, Kostiantyn P.; Holovach, Serhii; Lesyk, Dmytro; Holota, Yuliia; Borysko, Petro; Filatov, Andrey A.; Grygorenko, Oleksandr O. 分享 收藏
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In vitro evaluation of the immunogenic potential of gramicidin S and its photocontrolled analogues 体外评价gramicidin S及其光控类似物的免疫原性潜力 Horbatok, Kateryna; Semchuk, Iryna; Horbach, Oleksandr; Khranovska, Natalia; Kosach, Viktoriia; Borysko, Petro; Koniev, Serhii; Ulrich, Anne S.; Afonin, Sergii; Komarov, Igor V. 分享 收藏
Physicochemical and Biological Evaluation of gem-Difluorinated Saturated Oxygen Heterocycles as Bioisosteres for Drug Discovery Melnykov, Kostiantyn P.; Liashuk, Oleksandr S.; Holovach, Serhii; Shatnia, Valeriia; Horbenko, Artur; Lesyk, Dmytro; Melnyk, Varvara; Skrypnik, Daniil; Beshtynarska, Anna; Borysko, Petro; Viniichuk, Oleksandr; Grygorenko, Oleksandr O. 分享 收藏
Angular Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery Kirichok, Alexander A.; Tkachuk, Hennadii; Levchenko, Kostiantyn; Granat, Dmitry; Yegorova, Tetyana; Lesyk, Dmytro; Anisiforova, Anna; Holota, Yuliia; Zomchak, Viktoriia; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Korzh, Rodion A.; Al-Maali, Galeb; Kubyshkin, Vladimir; Rzepa, Henry S.; Mykhailiuk, Pavel K. 分享 收藏
CF3-Cyclobutanes: Synthesis, Properties, and Evaluation as a Unique tert-Butyl Group Analogue CF3-Cyclobutanes: 独特的叔丁基类似物的合成,性质和评价 Ahunovych, Volodymyr; Klipkov, Anton A.; Bugera, Maksym; Tarasenko, Karen; Trofymchuk, Serhii; Razhyk, Bohdan; Boretskyi, Andrii; Stanko, Oleh; Panasiuk, Yaroslav; Shablykin, Oleh; Al-Maali, Galeb; Lesyk, Dmytro; Klymenko-Ulianov, Oleksii; Horbatok, Kateryna; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Kubyshkin, Vladimir; Mykhailiuk, Pavel K. 分享 收藏
3,3-Difluorooxetane-A Versatile Functional Group for Bioisosteric Replacements in Drug Discovery Liashuk, Oleksandr S.; Fedinchyk, Anastasiya; Melnykov, Kostiantyn P.; Herasymchuk, Maksym; Alieksieieva, Diana; Lesyk, Dmytro; Bas, Yuliia P.; Keda, Tetiana Ye.; Yatsymyrskiy, Andriy V.; Holota, Yuliia; Borysko, Petro; Yarmolchuk, Volodymyr S.; Grygorenko, Oleksandr O. 分享 收藏
2-Oxabicyclo[2.1.1]hexanes: Synthesis, Properties, and Validation as Bioisosteres of ortho- and meta-Benzenes 2-氧杂双环 [2.1.1] 己烷: 邻苯和间苯的生物电子等排体的合成,性质和验证 Levterov, Vadym V.; Panasiuk, Yaroslav; Shablykin, Oleh; Stashkevych, Oleksandr; Sahun, Kateryna; Rassokhin, Artur; Sadkova, Iryna; Lesyk, Dmytro; Anisiforova, Anna; Holota, Yuliia; Borysko, Petro; Bodenchuk, Iryna; Voloshchuk, Nataliya M.; Mykhailiuk, Pavel K. 分享 收藏
Anticancer activity features of imidazole-based ionic liquids and lysosomotropic detergents: in silico and in vitro studies Gryniukova, Anastasiia; Borysko, Petro; Myziuk, Iryna; Alieksieieva, Diana; Hodyna, Diana; Semenyuta, Ivan; Kovalishyn, Vasyl; Metelytsia, Larysa; Rogalsky, Sergiy; Tcherniuk, Sergey 分享 收藏
Spiro[3.3]heptane as a Saturated Benzene Bioisostere 螺 [3.3] 庚烷作为饱和苯生物电子等排物 Prysiazhniuk, Kateryna; Datsenko, Oleksandr P.; Polishchuk, Oleksandr; Shulha, Stanislav; Shablykin, Oleh; Nikandrova, Yelyzaveta; Horbatok, Kateryna; Bodenchuk, Iryna; Borysko, Petro; Shepilov, Dmytro; Pishel, Iryna; Kubyshkin, Vladimir; Mykhailiuk, Pavel K. 分享 收藏
2-Oxabicyclo[2.2.2]octane as a new bioisostere of the phenyl ring Levterov, Vadym V.; Panasiuk, Yaroslav; Sahun, Kateryna; Stashkevych, Oleksandr; Badlo, Valentyn; Shablykin, Oleh; Sadkova, Iryna; Bortnichuk, Lina; Klymenko-Ulianov, Oleksii; Holota, Yuliia; Lachmann, Leonid; Borysko, Petro; Horbatok, Kateryna; Bodenchuk, Iryna; Bas, Yuliia; Dudenko, Dmytro; Mykhailiuk, Pavel K. 分享 收藏
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AI-Powered Virtual Screening of Large Compound Libraries Leads to the Discovery of Novel Inhibitors of Sirtuin-1 Gryniukova, Anastasiia; Kaiser, Florian; Myziuk, Iryna; Alieksieieva, Diana; Leberecht, Christoph; Heym, Peter P.; Tarkhanova, Olga O.; Moroz, Yurii S.; Borysko, Petro; Haupt, V. Joachim 分享 收藏
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