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Structure-based optimization of TEAD inhibitors: Exploring a novel subpocket near Glu347 for the treatment of NF2-mutant cancer 基于结构的TEAD抑制剂的优化:探索治疗NF2突变型癌症的新型亚口袋(靠近Glu347) Kim, Jin Kwan; Kim, Jinhyuk; Kim, Hadong; Jin, Haiyan; Yoo, Youngki; Fei, Xiang; Maeng, Han-Joo; Seo, Seung-Yong; Han, Gyoonhee; No, Kyoung Tai 分享 收藏
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Interface-aware molecular generative framework for protein-protein interaction modulators 蛋白质-蛋白质相互作用调节剂的界面感知分子生成框架 Wang, Jianmin; Mao, Jiashun; Li, Chunyan; Xiang, Hongxin; Wang, Xun; Wang, Shuang; Wang, Zixu; Chen, Yangyang; Li, Yuquan; No, Kyoung Tai; Song, Tao; Zeng, Xiangxiang 分享 收藏
Pan-Transcriptional Enhanced Associated Domain Palmitoylation Pocket Covalent Inhibitor Kim, Jinhyuk; Kim, Hadong; Kim, Jongwan; Cho, Seon Yeon; Moon, Sungho; Yoo, Youngki; Kim, Hanseong; Kim, Jin Kwan; Jeon, Hyejin; Namkung, Wan; Han, Gyoonhee; No, Kyoung Tai 分享 收藏
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Inhibition of IRP2-dependent reprogramming of iron metabolism suppresses tumor growth in colorectal cancer Hwang, Jieon; Park, Areum; Kim, Chinwoo; Kim, Chang Gon; Kwak, Jaesung; Kim, Byungil; Shin, Hyunjin; Ku, Minhee; Yang, Jaemoon; Baek, Ayoung; Choi, Jiwon; Lim, Hocheol; No, Kyoung Tai; Zhao, Xianghua; Choi, Uyeong; Kim, Tae Il; Jeong, Kyu-Sung; Lee, Hyuk; Shin, Sang Joon 分享 收藏
Identification of novel anti-obesity saponins from the ovary of sea cucumber ( Stichopus japonicus) ) Seo, Hyo-Deok; Lee, Ji-Young; Park, So-Hyun; Lee, Eunyoung; Hahm, Jeong-Hoon; Ahn, Jiyun; Jang, A. Ra; An, So Hee; Ha, Jang Ho; No, Kyoung Tai; Jung, Chang Hwa 分享 收藏
Inhibition of IRP2-dependent reprogramming of iron metabolism suppresses tumor growth in colorectal cancer Hwang, Jieon; Park, Areum; Kim, Chinwoo; Kim, Chang Gon; Kwak, Jaesung; Kim, Byungil; Shin, Hyunjin; Ku, Minhee; Yang, Jaemoon; Baek, Ayoung; Choi, Jiwon; Lim, Hocheol; No, Kyoung Tai; Zhao, Xianghua; Choi, Uyeong; Kim, Tae Il; Jeong, Kyu-Sung; Lee, Hyuk; Shin, Sang Joon 分享 收藏
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Exploring the Conformational Ensembles of Protein-Protein Complex with Transformer-Based Generative Model 基于Transformer的生成模型探索蛋白质-蛋白质复合物的构象集合 Wang, Jianmin; Wang, Xun; Chu, Yanyi; Li, Chunyan; Li, Xue; Meng, Xiangyu; Fang, Yitian; No, Kyoung Tai; Mao, Jiashun; Zeng, Xiangxiang 分享 收藏
KS20226, a first-in-class IRP2 inhibitor, preferentially induces reprogramming of iron metabolism and suppresses tumor growth in colorectal cancer Hwang, Jieon; Park, Areum; Kim, Chinwoo; Kim, Chang Gon; Kwak, Jaesung; Kim, Byungil; Shin, Hyunjin; Ku, Minhee; Yang, Jaemoon; Baek, Ayoung; Choi, Jiwon; Lim, Hocheol; No, Kyoung Tai; Zhao, Xianghua; Choi, Uyeong; Kim, Tae Il; Jeong, Kyu-Sung; Lee, Hyuk; Shin, Sang Joon 分享 收藏
Fragment molecular orbital-based variational quantum eigensolver for quantum chemistry in the age of quantum computing 量子计算时代用于量子化学的基于碎片分子轨道的变分量子本征求解器 Lim, Hocheol; Kang, Doo Hyung; Kim, Jeonghoon; Pellow-Jarman, Aidan; Mcfarthing, Shane; Pellow-Jarman, Rowan; Jeon, Hyeon-Nae; Oh, Byungdu; Rhee, June-Koo Kevin; No, Kyoung Tai 分享 收藏
Discovery of novel and potent TEAD inhibitors, orally available small molecules with anti-tumor activity in hippo pathway-dysregulated cancers Moon, Sungho; Cho, Seon Yeon; Kim, Minhye; Beak, Soojeong; Kim, Jinhyuk; Kim, Yongchan; Park, Sungil; Kim, Jung-In; Kim, Hanseong; Lee, In Sang; No, Kyoung Tai 分享 收藏
Targeting FLT3-TAZ signaling to suppress drug resistance in blast phase chronic myeloid leukemia 靶向FLT3-TAZ信号抑制急变期慢性粒细胞白血病耐药 Shin, Ji Eun; Kim, Soo-Hyun; Kong, Mingyu; Kim, Hwa-Ryeon; Yoon, Sungmin; Kee, Kyung-Mi; Kim, Jung Ah; Kim, Dong Hyeon; Park, So Yeon; Park, Jae Hyung; Kim, Hongtae; No, Kyoung Tai; Lee, Han-Woong; Gee, Heon Yung; Hong, Seunghee; Guan, Kun-Liang; Roe, Jae-Seok; Lee, Hyunbeom; Kim, Dong-Wook; Park, Hyun Woo 分享 收藏
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