Volodymyr G. Bdzhola - Publications, H-index & Citations

Volodymyr G. Bdzhola

national academy of sciences ukraine

21H指数

86论文数

989被引数

收录论文 29

发表时间

Discovery of new aurone derivatives as submicromolar CK2 inhibitors 新型黄质烯衍生物作为亚微摩尔CK2抑制剂的发现

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2025-12-31

PREAI

Mahdysiuk, Mykhailo V.; Volynets, Galyna P.; Bdzhola, Volodymyr G.; Bieda, Oleksandr A.; Lukashov, Sergiy S.; Sapelkin, Vladislav M.; Karbovskyi, Leonid L.; Yarmoluk, Sergiy M.

Leveraging large language models for literature-driven prioritization of protein binding pockets 利用大型语言模型进行基于文献的蛋白质结合口袋优先级排序

Bioinformatics

IF5.4

2025-08-07

OAAI

Roman Stratiichuk; Mykola Melnychenko; Ihor Koleiev; Taras Voitsitskyi; Vladyslav Husak; Nazar Shevchuk; Zakhar Ostrovsky; Volodymyr Bdzhola; Semen Yesylevskyy; Serhii Starosyla; Alan Nafiiev

Identification of novel Mycobacterium tuberculosis leucyl-tRNA synthetase inhibitors with antibacterial activity 新型分枝杆菌分枝杆菌（Mycobacterium tuberculosis）亮氨酰-tRNA合成酶抑制剂的鉴定及其抗菌活性

FUTURE MEDICINAL CHEMISTRY

IF3.4

2025-04-21

PREAI

Volynets, Galyna P.; Gudzera, Olga I.; Lukashov, Segiy S.; Gorbatiuk, Oksana B.; Usenko, Mariia O.; Ruban, Tetiana P.; Protopopov, Mykola V.; Tarnavskiy, Segiy S.; Kotey, Igor M.; Bdzhola, Volodymyr G.; Prykhod'ko, Andrii O.; Lukash, Lubov L.; Yarmoluk, Sergiy M.; Tukalo, Michael A.

Identification of dual-targeted Mycobacterium tuberculosis aminoacyl-tRNA synthetase inhibitors using machine learning

FUTURE MEDICINAL CHEMISTRY

IF3.4

2022-07-25

PREAI

Volynets, Galyna P.; Usenko, Mariia O.; Gudzera, Olga, I; Starosyla, Segiy A.; Balanda, Anatoliy O.; Syniugin, Anatolii R.; Gorbatiuk, Oksana B.; Prykhod'ko, Andrii O.; Bdzhola, Volodymyr G.; Yarmoluk, Sergiy M.; Tukalo, Michael A.

Identification of Novel Antistaphylococcal Hit Compounds Targeting Sortase A

MOLECULES

IF4.6

2021-11-24

OAAI

Volynets, Galyna; Vyshniakova, Hanna; Nitulescu, Georgiana; Nitulescu, George Mihai; Ungurianu, Anca; Margina, Denisa; Moshynets, Olena; Bdzhola, Volodymyr; Koleiev, Ihor; Iungin, Olga; Tarnavskiy, Sergiy; Yarmoluk, Sergiy

Discovery of novel antituberculosis agents among 3-phenyl-5-(1-phenyl-1H-[1,2,3]triazol-4-yl)-[1,2,4]oxadiazole derivatives targeting aminoacyl-tRNA synthetases

SCIENTIFIC REPORTS

IF3.9

2021-03-30

OAAI

Rybak, Mariia Yu.; Balanda, Anatoliy O.; Yatsyshyna, Anna P.; Kotey, Igor. M.; Starosyla, Sergiy A.; Bdzhola, Volodymyr G.; Lukash, Lubov L.; Yarmoluk, Sergiy M.; Tukalo, Michael A.; Volynets, Galyna P.

Dual-targeted hit identification using pharmacophore screening

JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN

IF3.1

2019-11-06

PREAI

Volynets, Galyna P.; Starosyla, Sergiy A.; Rybak, Mariia Yu; Bdzhola, Volodymyr G.; Kovalenko, Oksana P.; Vdovin, Vasyl S.; Yarmoluk, Sergiy M.; Tukalo, Michail A.

Dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-4-ones as a new class of CK2 inhibitors

MOLECULAR DIVERSITY

IF3.8

2018-05-29

PREAI

Protopopov, Mykola V.; Ostrynska, Olga V.; Starosyla, Sergiy A.; Vodolazhenko, Maria A.; Sirko, Svetlana M.; Gorobets, Nikolay Yu.; Bdzhola, Volodymyr; Desenko, Sergey M.; Yarmoluk, Sergiy M.

Structural Hypervariability of the Two Human Protein Kinase CK2 Catalytic Subunit Paralogs Revealed by Complex Structures with a Flavonol- and a Thieno[2,3-d]pyrimidine-Based Inhibitor

PHARMACEUTICALS

IF4.8

2017-01-11

OAAI

Niefind, Karsten; Bischoff, Nils; Golub, Andriy G.; Bdzhola, Volodymyr G.; Balanda, Anatoliy O.; Prykhod'ko, Andriy O.; Yarmoluk, Sergiy M.

Design, synthesis and evaluation of 3-quinoline carboxylic acids as new inhibitors of protein kinase CK2

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2016-09-02

OAAI

Syniugin, Anatolii R.; Ostrynska, Olga V.; Chekanov, Maksym O.; Volynets, Galyna P.; Starosyla, Sergiy A.; Bdzhola, Volodymyr G.; Yarmoluk, Sergiy M.

Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno[2,3-d]pyrimidines

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-06-01

PREAI

Ostrynska, Olga V.; Balanda, Anatoliy O.; Bdzhola, Volodymyr G.; Golub, Andriy G.; Kotey, Igor M.; Kukharenko, Olexander P.; Gryshchenko, Andrii A.; Briukhovetska, Nadiia V.; Yarmoluk, Sergiy M.

Identification of Mycobacterium tuberculosis leucyl-tRNA synthetase (LeuRS) inhibitors among the derivatives of 5-phenylamino-2H-[1,2,4]triazin-3-one

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2016-05-31

OAAI

Gudzera, Olga I.; Golub, Andriy G.; Bdzhola, Volodymyr G.; Volynets, Galyna P.; Kovalenko, Oksana P.; Boyarshin, Konstantin S.; Yaremchuk, Anna D.; Protopopov, Mykola V.; Yarmoluk, Sergiy M.; Tukalo, Michail A.

Design, synthesis and biological evaluation of 5-amino-4-(1H-benzoimidazol-2-yl)-phenyl-1,2-dihydro-pyrrol-3-ones as inhibitors of protein kinase FGFR1

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2016-05-01

PREAI

Gryshchenko, A. A.; Tarnavskiy, S. S.; Levchenko, K. V.; Bdzhola, V. G.; Volynets, G. P.; Golub, A. G.; Ruban, T. P.; Vygranenko, K. V.; Lukash, L. L.; Yarmoluk, S. M.

Discovery of potent anti-tuberculosis agents targeting leucyl-tRNA synthetase 发现靶向亮氨酰-tRNA合成酶的有效抗结核药物

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2016-03-01

PREAI

Gudzera, Olga I.; Golub, Andriy G.; Bdzhola, Volodymyr G.; Volynets, Galyna P.; Lukashov, Sergiy S.; Kovalenko, Oksana P.; Kriklivyi, Ivan A.; Yaremchuk, Anna D.; Starosyla, Sergiy A.; Yarmoluk, Sergiy M.; Tukalo, Michail A.

A Note of Caution on the Role of Halogen Bonds for Protein Kinase/Inhibitor Recognition Suggested by High- And Low-Salt CK2α Complex Structures

ACS CHEMICAL BIOLOGY

IF3.8

2015-05-15

PREAI

Guerra, Barbara; Bischoff, Nils; Bdzhola, Volodymyr G.; Yarmoluk, Sergiy M.; Issinger, Olaf-Georg; Golub, Andriy G.; Niefind, Karsten

Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1,5-dihydro-pyrrol-2-one benzothiazol-2-yl-3-hydroxy-5-phenyl-1，5-二氢-吡咯-2-酮衍生物中凋亡信号调节激酶1 (ASK1) 抑制剂的鉴定

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-05-01

PREAI

Starosyla, Sergiy A.; Volynets, Galyna P.; Lukashov, Sergiy S.; Gorbatiuk, Oksana B.; Golub, Andriy G.; Bdzhola, Volodymyr G.; Yarmoluk, Sergiy M.

Design, synthesis and biological evaluation of N-phenylthieno[2,3-d]pyrimidin-4-amines as inhibitors of FGFR1 FGFR1抑制剂N-苯基噻吩并 [2，3-d]pyrimidin-4-amines的设计、合成及生物活性评价

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-05-01

PREAI

Gryshchenko, A. A.; Bdzhola, V. G.; Balanda, A. O.; Briukhovetska, N. V.; Kotey, I. M.; Golub, A. G.; Ruban, T. P.; Lukash, L. L.; Yarmoluk, S. M.

Design, synthesis and biological evaluation of naphthostyril derivatives as novel protein kinase FGFR1 inhibitors 新型蛋白激酶FGFR1抑制剂萘苯普利衍生物的设计、合成及生物活性评价

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2014-06-18

OAAI

Gryshchenko, Andrii Anatoliyovych; Levchenko, Kostiantyn Vasyliovych; Bdzhola, Volodymyr Grygorovich; Ruban, Tatiana Panasivna; Lukash, Lyubov Leonidovna; Yarmoluk, Sergiy Mikolayovych

Discovery and characterization of synthetic 4′-hydroxyflavones-New CK2 inhibitors from flavone family

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2013-11-01

PREAI

Golub, Andriy G.; Bdzhola, Volodymyr G.; Ostrynska, Olga V.; Kyshenia, Iaroslav V.; Sapelkin, Vladislav M.; Prykhod'ko, Andriy O.; Kukharenko, Olexander P.; Yarmoluk, Sergiy M.

Design, synthesis and biological evaluation of 2-aminopyrimidinones and their 6-aza-analogs as a new class of CK2 inhibitors

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2013-10-03

PREAI

Chekanov, Maksym O.; Ostrynska, Olga V.; Tarnavskyi, Sergii S.; Synyugin, Anatoliy R.; Briukhovetska, Nadiia V.; Bdzhola, Volodymyr G.; Pashenko, Alexander E.; Fokin, Andrey A.; Yarmoluk, Sergiy M.

研究方向