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Structure-Metabolism Relationships of Benzimidazole Derivatives with anti-Trypanosoma cruzi Activity for Chagas Disease 具有抗锥虫活性的苯并咪唑衍生物对查加斯病的结构代谢关系 Espinoza-Chavez, Rocio Marisol; Rezende Junior, Celso de Oliveira; de Souza, Mariana Laureano; Chelucci, Rafael Consolin; Michelan-Duarte, Simone; Krogh, Renata; Ferreira, Leonardo Luiz Gomes; Valli, Marilia; de Oliveira, Aldo Sena; Andricopulo, Adriano D.; Dias, Luiz Carlos 分享 收藏
New Chalcogen-Functionalized Naphthoquinones: Design, Synthesis, and Evaluation, In Vitro and In Silico, against Squamous Cell Carcinoma Gomes, Luana da Silva; Costa, Erica de Oliveira; Duarte, Thuany G.; Charret, Thiago S.; Castiglione, Raquel C.; Simoes, Rafael L.; Pascoal, Vinicius D. B.; Doring, Thiago H.; da Silva, Fernando de C.; Ferreira, Vitor F.; de Oliveira, Aldo S.; Pascoal, Aislan C. R. F.; Cruz, Andre L. S.; Nascimento, Vanessa 分享 收藏
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Structure-activity relationships of novel N-imidazoylpiperazines with potent anti-Trypanosoma cruzi activity Espinoza-Chavez, Rocio Marisol; de Oliveira Rezende Jr, Celso; de Souza, Mariana Laureano; Pauli, Ivani; Valli, Marilia; Ferreira, Leonardo Luiz Gomes; Chelucci, Rafael Consolin; Michelan-Duarte, Simone; Krogh, Renata; da Silva, Fernando Bezerra Romualdo; Cruz, Fabio Cardoso; de Oliveira, Aldo Sena; Andricopulo, Adriano Defini; Dias, Luiz Carlos 分享 收藏
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DYRK1A Inhibitors and Perspectives for the Treatment of Alzheimer's Disease de Souza, Marcia Maria; Cenci, Arthur Ribeiro; Teixeira, Kerolain Faoro; Machado, Valkiria; Schuler, Majory Christina Garcia Mendes; Goncalves, Ana Elisa; Dalmagro, Ana Paula; Cazarin, Camila Andre; Gomes Ferreira, Leonardo Luiz; de Oliveira, Aldo Sena; Andricopulo, Adriano Defini 分享 收藏
Synthesis and investigation of the trypanocidal potential of novel 1,2,3-triazole-selenide hybrids Chipoline, Ingrid C.; Brasil, Beatrice F. A. B.; Neto, Jose S. S.; Valli, Marilia; Krogh, Renata; Cenci, Arthur R.; Teixeira, Kerolain F.; Zapp, Eduardo; Brondani, Daniela; Ferreira, Leonardo L. G.; Andricopulo, Adriano D.; Oliveira, Aldo S. de; Nascimento, Vanessa 分享 收藏
Phomoxanthone A, Compound of Endophytic Fungi Paecilomyces sp. and Its Potential Antimicrobial and Antiparasitic Ramos, Gisele da Costa; Silva-Silva, Joao Victor; Watanabe, Luciano Almeida; de Sousa Siqueira, Jose Edson; Almeida-Souza, Fernando; Calabrese, Katia S.; do Rosario Marinho, Andrey Moacir; Barbosa Marinho, Patricia Santana; de Oliveira, Aldo Sena 分享 收藏
Novel trypanocidal thiophen-chalcone cruzain inhibitors: structure- and ligand-based studies de Oliveira, Aldo S.; Valli, Marilia; Ferreira, Leonardo L. G.; Souza, Julia M.; Krogh, Renata; Meier, Lidiane; Abreu, Heitor R.; Voltolini, Bruna G.; Llanes, Luana C.; Nunes, Ricardo J.; Braga, Antonio L.; Andricopulo, Adriano D. 分享 收藏
Carajurin Induces Apoptosis in Leishmania amazonensis Promastigotes through Reactive Oxygen Species Production and Mitochondrial Dysfunction Silva-Silva, Joao Victor; Moragas-Tellis, Carla J.; Chagas, Maria S. S.; Souza, Paulo Victor R.; Moreira, Davyson L.; Hardoim, Daiana J.; Taniwaki, Noemi N.; Costa, Vanessa F. A.; Bertho, Alvaro L.; Brondani, Daniela; Zapp, Eduardo; de Oliveira, Aldo Sena; Calabrese, Katia S.; Behrens, Maria D.; Almeida-Souza, Fernando 分享 收藏
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Pyrazolines as potential anti-Alzheimer's agents: DFT, molecular docking, enzyme inhibition and pharmacokinetic studies Machado, Valkiria; Cenci, Arthur R.; Teixeira, Kerolain F.; Sens, Larissa; Tizziani, Tiago; Nunes, Ricardo J.; Ferreira, Leonardo L. G.; Yunes, Rosendo A.; Sandjo, Louis P.; Andricopulo, Adriano D.; de Oliveira, Aldo S. 分享 收藏
Diaminomaleonitrile derivatives as new potential antichagasic compounds: a study of structure-activity relationships de Oliveira, Aldo S.; Mello, Lucas dos S.; Ogihara, Camila H.; Doring, Thiago H.; Palomino-Salcedo, David L.; Michelan-Duarte, Simone; Ferreira, Leonardo L. G.; Souza, Julia M.; Davila-Rodriguez, Maria Jose; da Cruz Junior, Jose W.; Dockal, Edward R.; Andricopulo, Adriano D. 分享 收藏
Carajurin: a anthocyanidin from Arrabidaea chica as a potential biological marker of antileishmanial activity Silva-Silva, Joao Victor; Moragas-Tellis, Carla J.; Chagas, Maria S. S.; Souza, Paulo Victor R.; Moreira, Davyson L.; de Souza, Celeste S. F.; Teixeira, Kerolain F.; Cenci, Arthur R.; de Oliveira, Aldo S.; Almeida-Souza, Fernando; Behrens, Maria D.; Calabrese, Katia S. 分享 收藏
Structure-activity relationships of sulfonamides derived from carvacrol and their potential for the treatment of Alzheimer's disease de Souza, Marcia Maria; Andreolla, Marina Correa; Ribeiro, Thais Cecilia; Goncalves, Ana Elisa; Medeiros, Alex Rogerio; de Souza, Anacleto Silva; Gomes Ferreira, Leonardo Luiz; Andricopulo, Adriano Defini; Yunes, Rosendo Augusto; de Oliveira, Aldo Sena 分享 收藏
Antinociceptive effect of hydroalcoholic extract and isoflavone isolated from Polygala molluginifolia in mice: evidence for the involvement of opioid receptors and TRPV1 and TRPA1 channels Nucci-Martins, Catharina; Nascimento, Leandro F.; Venzke, Dalila; Brethanha, Lizandra C.; Sako, Alysson V. F.; Oliveira, Aldo S.; Brighente, Ines M. C.; Micke, Gustavo A.; Pizzolatti, Moacir G.; Santos, Adair R. S. 分享 收藏