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1-[(Imidazolidin-2-yl)imino]-1H-indoles as new hypotensive agents: synthesis and in vitro and in vivo biological studies Kornicka, Anita; Wasilewska, Aleksandra; Saczewski, Jaroslaw; Hudson, Alan L.; Boblewski, Konrad; Lehmann, Artur; Gzella, Karol; Belka, Mariusz; Saczewski, Franciszek; Gdaniec, Maria; Rybczynska, Apolonia; Baczek, Tomasz 分享 收藏
Combined Interactions with I1-, I2-Imidazoline Binding Sites and α2-Adrenoceptors To Manage Opioid Addiction Giusepponi, Maria Elena; Cifani, Carlo; Di Bonaventura, Maria Vittoria Micioni; Mattioli, Laura; Hudson, Alan; Diamanti, Eleonora; Del Bello, Fabio; Giannella, Mario; Mammoli, Valerio; Paoletti, Corinne Dalila; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma 分享 收藏
Transfer of SAR information from hypotensive indazole to indole derivatives acting at α-adrenergic receptors: In vitro and in vivo studies Saczewski, Jaroslaw; Hudson, Alan; Scheinin, Mika; Wasilewska, Aleksandra; Saczewski, Franciszek; Rybczynska, Apolonia; Ferdousi, Mehnaz; Laurila, Jonne M.; Boblewski, Konrad; Lehmann, Artur; Watts, Helena; Ma, Daqing 分享 收藏
EVERSUN: a phase 2 trial of alternating sunitinib and everolimus as first-line therapy for advanced renal cell carcinoma Davis, I. D.; Long, A.; Yip, S.; Espinoza, D.; Thompson, J. F.; Kichenadasse, G.; Harrison, M.; Lowenthal, R. M.; Pavlakis, N.; Azad, A.; Kannourakis, G.; Steer, C.; Goldstein, D.; Shapiro, J.; Harvie, R.; Jovanovic, L.; Hudson, A. L.; Nelson, C. C.; Stockler, M. R.; Martin, A. 分享 收藏
Fluorinated analogues of marsanidine, a highly α2-AR/imidazoline I1 binding site-selective hypotensive agent. Synthesis and biological activities Wasilewska, Aleksandra; Saczewski, Franciszek; Hudson, Alan L.; Ferdousi, Mehnaz; Scheinin, Mika; Laurila, Jonne M.; Rybczynska, Apolonia; Boblewski, Konrad; Lehmann, Artur 分享 收藏
Modulation of Resistance Artery Tone by the Trace Amine β-Phenylethylamine: Dual Indirect Sympathomimetic and α1-Adrenoceptor Blocking Actions Narang, Deepak; Kerr, Paul M.; Lunn, Stephanie E.; Beaudry, Rhys; Sigurdson, Julie; Lalies, Margaret D.; Hudson, Alan L.; Light, Peter E.; Holt, Andrew; Plane, Frances 分享 收藏
Discovery and Structure-Activity Relationships of Pyrrolone Antimalarials Murugesan, Dinakaran; Mital, Alka; Kaiser, Marcel; Shackleford, David M.; Morizzi, Julia; Katneni, Kasiram; Campbell, Michael; Hudson, Alan; Charman, Susan A.; Yeates, Clive; Gilbert, Ian H. 分享 收藏
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Favourable involvement of α2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancement Mammoli, Valerio; Bonifazi, Alessandro; Del Bello, Fabio; Diamanti, Eleonora; Giannella, Mario; Hudson, Alan L.; Mattioli, Laura; Perfumi, Marina; Piergentili, Alessandro; Quaglia, Wilma; Titomanlio, Federica; Pigini, Maria 分享 收藏
Synthesis and biological activities of 2-[(heteroaryl)methyl]imidazolines Saczewski, Jaroslaw; Hudson, Alan; Scheinin, Mika; Rybczynska, Apolonia; Ma, Daqing; Saczewski, Franciszek; Laird, Shayna; Laurila, Jonne M.; Boblewski, Konrad; Lehmann, Artur; Gu, Jianteng; Watts, Helena 分享 收藏
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Antimalarial Pyrido[1,2-a]benzimidazoles Ndakala, Albert J.; Gessner, Richard K.; Gitari, Patricia W.; October, Natasha; White, Karen L.; Hudson, Alan; Fakorede, Foluke; Shackleford, David M.; Kaiser, Marcel; Yeates, Clive; Charman, Susan A.; Chibale, Kelly 分享 收藏
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3-[(Imidazolidin-2-yl)imino]indazole ligands with selectivity for the α2-adrenoceptor compared to the imidazoline I1 receptor Saczewski, Franciszek; Kornicka, Anita; Hudson, Alan L.; Laird, Shayna; Scheinin, Mika; Laurila, Jonne M.; Rybczynska, Apolonia; Boblewski, Konrad; Lehmann, Artur; Gdaniec, Maria 分享 收藏
Novel imidazoline compounds as partial or full agonists of D2-like dopamine receptors inspired by I2-imidazoline binding sites ligand 2-BFI 新型咪唑啉化合物作为D2-like多巴胺受体的部分或完全激动剂,受I2-imidazoline结合位点配体2-BFI启发 Giorgioni, Gianfabio; Ambrosini, Dario; Vesprini, Cristian; Hudson, Alan; Nasuti, Cinzia; Di Stefano, Antonio; Sozio, Piera; Ciampi, Osele; Costa, Barbara; Martini, Claudia; Carrieri, Antonio; Carbonara, Giuseppe; Enzensperger, Christoph; Pigini, Maria 分享 收藏
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