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Marián Hajdúch

palacky university and university hospital olomouc

58H指数
745论文数
1.5W被引数
收录论文 268
发表时间
Synthesis and Biological Activity of 2,6-Disubstituted and 2,6,9-Trisubstituted 7-Deazapurine Nucleobases2,6-二取代和2,6,9-三取代7-脱氮嘌呤碱基的合成与生物活性
err2026-09-07
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errOAAI
errUgnė Šinkevičiūtė; Kateřina Burgetová Ječmeňová; Soňa Gurská; Lenka Poštová Slavětínská; Vincent Baran; Pavel Polishchuk; Petr Džubák; Michal Hocek; Marián Hajdúch; Michal Tichý
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New 1,2,3-Triazole Hybrids as Anticancer Agents: Design, Synthesis, Characterization, and In Silico Studies新型1,2,3-三唑杂化物作为抗癌药物:设计、合成、表征及计算机模拟研究
err2026-09-07
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PREAI
errAlirica I. Suárez; Katiuska E. Chávez; Pablo Martínez; José Bubis; Zuleyma Blanco; Hegira Ramírez; Jenny Valentina Garmendia; Juan Bautista De Sanctis; Soňa Gurská; Petr Džubák; Marián Hajdúch; Jaime E. Charris
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Optimization of Azaspirooxindolinone-based PROTACs targeting BTK: Synthesis, kinase profiling, and degradation analysis氮杂螺恶唑啉酮基PROTACs靶向BTK的优化:合成、激酶谱分析及降解分析
err2026-05-01
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PREAI
errRampeesa, Naveen Kumar; Gundla, Rambabu; Gurska, Sona; Yadam, Sabitha; Tangallapalli, Sudhakar; Anugu, Sreenivasa Reddy; De Sanctis, Juan Bautista; Dzubak, Petr; Hajduch, Marian; Katari, Naresh Kumar; Das, Viswanath; Jonnalagadda, Sreekantha Babu
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Design; synthesis; and biological evaluation of novel 3-oxo-2; 3-dihydropyridazine derivatives as interleukin-2-inducible T-cell kinase (ITK) inhibitors设计、合成及新型3-氧代-2,3-二氢吡啶azine衍生物的生物活性评价,作为白细胞介素-2诱导的T细胞激酶(ITK)抑制剂
err2025-12-03
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errOAAI
errSudhakar Tangallapalli; Rambabu Gundla; Kalyani Paidikondala; Soňa Gurská; Naveen Kumar Rampeesa; Sreenivasa Reddy Anugu; Petr Džubák; Marián Hajdúch; Viswanath Das; Naresh Kumar Katari
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May the target be with you: polysaccharide-coated upconverting nanoparticles for macrophage targeting愿靶标与你同在:聚糖涂层上转换纳米颗粒用于巨噬细胞靶向
err2025-10-23
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errOAAI
errKarolina Zajdel †; Volodymyr Lobaz †; Martin Ondra †; Rafal Konefał; Oliver Moravec; Ognen Pop-Georgievski; Jiří Pánek; Damian Kalita; Bożena Sikora-Dobrowolska; Lukáš Lenart; Marián Hajdúch; Martin Hrubý; Marek Pruszyński
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Paving the way for future PSMA inhibitors: insights from comparative preclinical evaluations of structure modifications为未来PSMA抑制剂铺平道路:结构修饰比较性临床前评估的见解
err2025-09-26
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errOAAI
errKatarína Hajduová; Kateřina Dvořáková Bendová; Miloš Petřík; Martina Benešová-Schäfer; Martin Schäfer; Marián Hajdúch; Zbyněk Nový
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Hydrophobic residues in the α-synuclein NAC domain drive seed-competent fibril formation and are targeted by peptide inhibitorsα-突触核蛋白NAC结构域中的疏水残基驱动具有种子能力的原纤维形成,并被肽抑制剂靶向。
err2025-08-17
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errOAAI
errViswanath Das; Sayed Mostafa Modarres Mousavi; Narendran Annadurai; Sunčica Sukur; Faramarz Mehrnejad; Sajad Moradi; Lukáš Malina; Markéta Kolaříková; Vaclav Ranc; Ivo Frydrych; Roman Kouřil; Saman Hosseinkhani; Marián Hajdúch; Maryam Nikkhah
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Triterpenoid derivatives inhibit Gli-mediated transcription in human glioblastoma cell line via direct interaction with Gli1三萜类衍生物通过直接与Gli1相互作用,抑制人胶质母细胞瘤细胞系中的Gli介导的转录。
err2025-07-10
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errOAAI
errIvo Frydrych; Jiří Řehulka; Lucie Slavíková; Jiří Hodoň; Jan Pokorný; Veronika Šidová; Martina Medvedíková; Hanuš Slavík; Pavel Polishchuk; Tomáš Oždian; Jana Vrbková; Jan Šarek; Petr Džubák; Marián Hajdúch; Milan Urban
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Morphological profiling data resource enables prediction of chemical compound properties形态学分析数据资源能够预测化学化合物的性质
err2025-05-01
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errOAAI
errWolff, Christopher; Neuenschwander, Martin; Beese, Carsten Jorn; Sitani, Divya; Ramos, Maria C.; Srovnalova, Alzbeta; Varela, Maria Jose; Polishchuk, Pavel; Skopelitou, Katholiki E.; Skuta, Ctibor; Stechmann, Bahne; Brea, Jose; Clausen, Mads Hartvig; Dzubak, Petr; Fernandez-Godino, Rosario; Genilloud, Olga; Hajduch, Marian; Loza, Maria Isabel; Lehmann, Martin; von Kries, Jens Peter; Sun, Han; Schmied, Christopher
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In vitro and in vivo evaluation of anti-HER2 antibody conjugates labelled with 225Ac体外和体内评价标记有225Ac的抗HER2抗体偶联物
err2025-04-04
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errOAAI
errOndrak Fialova, Katerina; Ondrak, Lukas; Vlk, Martin; Kozempel, Jan; Novakova, Katerina; Novy, Zbynek; Hajduova, Katarina; Hajduch, Marian; Petrik, Milos; Pruszynski, Marek; Bruchertseifer, Frank; Morgenstern, Alfred
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Design, synthesis, and biological evaluation of novel azaspirooxindolinone derivatives as potent inhibitors of ITK and BTK-dependent cancers
err2025-04-01
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PREAI
errMudasani, Gopal; Rampeesa, Naveen Kumar; Anugu, Sreenivasa Reddy; Muddasani, Pullareddy; Gurska, Sona; Dzubak, Petr; Hajduch, Marian; Das, Viswanath; Gundla, Rambabu
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