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收藏Self-Assembly Properties of an Amphiphilic Phosphate Ester Prodrug Designed for the Treatment of COVID-19
Laramy, Matthew N. O'Brien; Bezawada, Padmavani; Horst, Reto; Jaini, Rohit; Lillis, Jonathan; Liu, Yizhou; Luthra, Suman; Nguyen, Bao; Patel, Nandini; Soni, Smita; Sullivan, Bradley P.; Thiel, Andrew; Ticehurst, Martyn D.
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收藏Preclinical characterization of an intravenous coronavirus 3CL protease inhibitor for the potential treatment of COVID19
Boras, Britton; Jones, Rhys M.; Anson, Brandon J.; Arenson, Dan; Aschenbrenner, Lisa; Bakowski, Malina A.; Beutler, Nathan; Binder, Joseph; Chen, Emily; Eng, Heather; Hammond, Holly; Hammond, Jennifer; Haupt, Robert E.; Hoffman, Robert; Kadar, Eugene P.; Kania, Rob; Kimoto, Emi; Kirkpatrick, Melanie G.; Lanyon, Lorraine; Lendy, Emma K.; Lillis, Jonathan R.; Logue, James; Luthra, Suman A.; Ma, Chunlong; Mason, Stephen W.; McGrath, Marisa E.; Noell, Stephen; Obach, R. Scott; O' Brien, Matthew N.; O'Connor, Rebecca; Ogilvie, Kevin; Owen, Dafydd; Pettersson, Martin; Reese, Matthew R.; Rogers, Thomas F.; Rosales, Romel; Rossulek, Michelle I.; Sathish, Jean G.; Shirai, Norimitsu; Steppan, Claire; Ticehurst, Martyn; Updyke, Lawrence W.; Weston, Stuart; Zhu, Yuao; White, Kris M.; Garcia-Sastre, Adolfo; Wang, Jun; Chatterjee, Arnab K.; Mesecar, Andrew D.; Frieman, Matthew B.; Anderson, Annaliesa S.; Allerton, Charlotte
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收藏CK1 δ/ε Inhibitor PF-05006739 Ameliorates Hepatic Steatosis and Hyperinsulinemia in Dio Mice
Peloquin, Matthew; Litchfield, John; Zhang, Bei B.; Chang, Cheng; Miller, Russell A.; Bernardo, Barbara; Luthra, Suman; Cortes, Christian; Li, Xiangping, II; Zou, Chang J.
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收藏Delineating the role of cooperativity in the design of potent PROTACs for BTK
Zorba, Adelajda; Chuong Nguyen; Xu, Yingrong; Starr, Jeremy; Borzilleri, Kris; Smith, James; Zhu, Hongyao; Farley, Kathleen A.; Ding, WeiDong; Schiemer, James; Feng, Xidong; Chang, Jeanne S.; Uccello, Daniel P.; Young, Jennifer A.; Garcia-Irrizary, Carmen N.; Czabaniuk, Lara; Schuff, Brandon; Oliver, Robert; Montgomery, Justin; Hayward, Matthew M.; Coe, Jotham; Chen, Jinshan; Niosi, Mark; Luthra, Suman; Shah, Jaymin C.; El-Kattan, Ayman; Qiu, Xiayang; West, Graham M.; Noe, Mark C.; Shanmugasundaram, Veerabahu; Gilbert, Adam M.; Brown, Matthew F.; Calabrese, Matthew F.
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