未登录 Synthesis of Nirmatrelvir: Development of an Efficient, Scalable Process to Generate the Western Fragment Algera, Russell F.; Allais, Christophe; Baldwin, Aaron F.; Becirovic, Husein; Bowles, Paul; Brown, Adam R.; Buske, Jamie M.; Clarke, Hugh J.; Do, Nga M.; Doyle, Kevin; Fifer, Jonathan; Gray, Kaitlyn; Happe, Alan; Hardink, Mark; Hubbell, Aran K.; James, Chintelle; Khadamkar, Hrushikesh P.; Magano, Javier; McInturff, Emma L.; Mustakis, Jason; Ozbuyukkaya, Gizem; Piper, Jared L.; Place, David W.; Ragan, John A.; Rauschenberger, Blake; Reyes, Giselle; Shehadeh, Rawan; Stanchina, Corey; Stanley, Michael; Weekly, R. Matthew; Weinstein, Ethan; Weisenburger, Gerald A.; Wood, Ethan; Yayla, Hatice G.; Yu, Shu 分享 收藏
Synthesis of Nirmatrelvir: Design and Optimization of an Efficient Telescoped Amidation-Dehydration Sequence Algera, Russell F.; Baldwin, Aaron F.; Bowles, Paul; Clarke, Hugh J.; Connor, Christina G.; Cordi, Eric M.; Do, Nga M.; Nicholson, Lindsay D.; Georgian, William; Happe, Alan; Herman, Madeline I.; Hilou, Elaa; James, Chintelle; Johnson, Amber M.; Kalinowski, Maciej; Kulkarni, Samir A.; Launer-Felty, Katherine D.; Lee, Johnny W.; Lee, Taegyo; Lopez, Jorge; Mcinturff, Emma L.; Piper, Jared L.; Place, David W.; Ragan, John A.; Rauschenberger, Blake; Ryder, Katherine; Stanley, Michael; Weisenburger, Gerald A.; Weekly, R. Matthew; Allais, Christophe 分享 收藏
Application of Biocatalytic Reductive Amination for the Synthesis of a Key Intermediate to a CDK 2/4/6 Inhibitor Duan, Shengquan; Widlicka, Daniel W.; Burns, Michael P.; Kumar, Rajesh; Hotham, Ian; Desrosiers, Jean-Nicolas; Bowles, Paul; Jones, Kris N.; Nicholson, Lindsay D.; Buetti-Weekly, Michele T.; Han, Lu; Steflik, Jeremy; Hansen, Eric; Hayward, Cheryl M.; Strohmeyer, Holly; Monfette, Sebastien; Sutton, Scott C.; Morris, Christopher 分享 收藏
分享 收藏
分享 收藏
Commercial Route Research and Development for SGLT2 Inhibitor Candidate Ertugliflozin Bowles, Paul; Brenek, Steven J.; Caron, Stephane; Do, Nga M.; Drexler, Michele T.; Duan, Shengquan; Dube, Pascal; Hansen, Eric C.; Jones, Brian P.; Jones, Kris N.; Ljubicic, Tomislav A.; Makowski, Teresa W.; Mustakis, Jason; Nelson, Jade D.; Olivier, Mark; Peng, Zhihui; Perfect, Handi H.; Place, David W.; Ragan, John A.; Salisbury, John J.; Stanchina, Corey L.; Vanderplas, Brian C.; Webster, Mark E.; Weekly, R. Matt 分享 收藏
Synthesis of Filibuvir. Part I. Diastereoselective Preparation of a β-Hydroxy Alkynyl Oxazolidinone and Conversion to a 6,6-Disubstituted 2H-Pyranone Singer, Robert A.; Ragan, John A.; Bowles, Paul; Chisowa, Esmort; Conway, Brian G.; Cordi, Eric M.; Leeman, Kyle R.; Letendre, Leo J.; Sieser, Janice E.; Sluggett, Gregory W.; Stanchina, Corey L.; Strohmeyer, Holly; Blunt, Jon; Taylor, Stuart; Byrne, Ciaran; Lynch, Denis; Mullane, Sandra; O'Sullivan, Maria M.; Whelan, Marcella 分享 收藏
分享 收藏
分享 收藏
分享 收藏
分享 收藏
分享 收藏
分享 收藏
Synthesis and purification of 6-ethoxy-4-oxo-1,4-dihydro-[1,5]naphthyridine-3-carboxylic acid benzylamide Beaudin, J; Bourassa, DE; Bowles, P; Castaldi, MJ; Clay, R; Couturier, MA; Karrick, G; Makowski, TW; McDermott, RE; Meltz, CN; Meltz, M; Phillips, JE; Ragan, JA; Ripin, DHB; Singer, RA; Tucker, JL; Wei, LL 分享 收藏
分享 收藏
分享 收藏
分享 收藏