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Michel O. Steinmetz

psi

82H指数
388论文数
2.3W被引数
收录论文 156
发表时间
An integrated experimental and computational pipeline for crystallographic fragment screening of membrane protein in the lipid cubic phase膜蛋白在脂质立方相中的晶体学片段筛选集成实验与计算流程
err2026-05-13
err0
errOAAI
errChia-Ying Huang; Robert Cheng; Alexander Metz; Denis Bucher; Fabio Andres; Arianna Bacchin; Hannah Glover; Christoph P. Sager; Meitian Wang; Michel O. Steinmetz; Michael Hennig; May Sharpe
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Structural basis of microtubule-mediated signal transduction微管介导的信号转导的结构基础
errCell
IF42.5
err2025-12-08
err0
errOAAI
errSung Ryul Choi; Thorsten B. Blum; Matteo Giono; Bibhas Roy; Ioannis Vakonakis; Dominic Schmid; Nicole Oelgarth; Apisha Ranganathan; Alvar D. Gossert; G.V. Shivashankar; Alfred Zippelius; Michel O. Steinmetz
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Asymmetric Total Synthesis of (−)-Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding(−)-Glycybridin B的不对称全合成,一种用于微管结合的药效基筛选候选物
err2025-08-06
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errOAAI
errDr. Alice Maiocchi; Dr. Maxim Shevelev; Dr. Zlata Boiarska; Dr. Juan Estévez-Gallego; Dr. Francesca Bonato; Dr. Paolo Orlando; Alessandra Chinosi; Emanuele Marcone; Dr. Andrea Citarella; Dr. Dragos Horvath; Prof. Dr. Michel O. Steinmetz; Dr. Andrea E. Prota; Dr. Alexandre Varnek; Dr. Valerio Fasano; Prof. Dr. Daniele Passarella
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Hydrolysis-deficient mosaic microtubules as faithful mimics of the GTP cap水解缺陷型镶嵌微管作为GTP帽的忠实模拟物
err2025-03-10
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errOAAI
errEstevez-Gallego, Juan; Blum, Thorsten B.; Ruhnow, Felix; Gili, Maria; Speroni, Silvia; Garcia-Castellanos, Raquel; Steinmetz, Michel O.
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Centriolar cap proteins CP110 and CPAP control slow elongation of microtubule plus ends中心粒帽蛋白CP110和CPAP调控微管正极的缓慢延长
err2025-01-23
err0
errOAAI
errIyer, Saishree S.; Chen, Fangrui; Ogunmolu, Funso E.; Moradi, Shoeib; Volkov, Vladimir A.; van Grinsven, Emma J.; van Hoorn, Chris; Wu, Jingchao; Andrea, Nemo; Hua, Shasha; Jiang, Kai; Vakonakis, Ioannis; Potocnjak, Mia; Herzog, Franz; Gigant, Benoit; Gudimchuk, Nikita; Stecker, Kelly E.; Dogterom, Marileen; Steinmetz, Michel O.; Akhmanova, Anna
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Bridging the maytansine and vinca sites: Cryptophycins target β-tubulin ' s T5-loop
err2024-06-01
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errOAAI
errAbel, Anne-Catherine; Muhlethaler, Tobias; Dessin, Cedric; Schachtsiek, Thomas; Sammet, Benedikt; Sharpe, Timothy; Steinmetz, Michel O.; Sewald, Norbert; Prota, Andrea E.
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The novel microtubule-destabilizing compound AUS_001 maintains unique binding to the colchicine site of tubulin and elicits reversible cellular effects relative to other anti-tubulin agents
err2024-03-22
err0
PREAI
errLelie, Herman; Chou, Yao-Chieh; King, Alastair J.; Boiarska, Zlata; Prota, Andrea E.; Steinmetz, Michel O.; Koutsioumpa, Marina
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Modular synthesis of functional libraries by accelerated SuFEx click chemistry
err2024-01-01
err3
errOAAI
errHomer, Joshua A.; Koelln, Rebecca A.; Barrow, Andrew S.; Gialelis, Timothy L.; Boiarska, Zlata; Steinohrt, Nikita S.; Lee, Erinna F.; Yang, Wen-Hsuan; Johnson, Robert M.; Chung, Taemoon; Habowski, Amber N.; Vishwakarma, Dharmendra S.; Bhunia, Debmalya; Avanzi, Charlotte; Moorhouse, Adam D.; Jackson, Mary; Tuveson, David A.; Lyons, Scott K.; Lukey, Michael J.; Fairlie, W. Douglas; Haider, Shozeb M.; Steinmetz, Michel O.; Prota, Andrea E.; Moses, John E.
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A photo-SAR study of photoswitchable azobenzene tubulin-inhibiting antimitotics identifying a general method for near-quantitative photocontrol
err2024-01-01
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errOAAI
errReynders, Martin; Garscia, Malgorzata; Mueller-Deku, Adrian; Wranik, Maximilian; Krauskopf, Kristina; de la Rosa, Luis de la Osa; Schaffer, Konstantin; Joetten, Anna; Rode, Alexander; Stierle, Valentin; Kraus, Yvonne; Baumgartner, Benedikt; Ali, Ahmed; Bubeneck, Andrei; Seal, Trina; Steinmetz, Michel O.; Paulitschke, Philipp; Thorn-Seshold, Oliver
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A multi-reservoir extruder for time-resolved serial protein crystallography and compound screening at X-ray free-electron lasers用于x射线自由电子激光器的时间分辨系列蛋白质晶体学和化合物筛选的多储层挤出机
err2023-12-02
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errOAAI
errWranik, Maximilian; Kepa, Michal W.; Beale, Emma V.; James, Daniel; Bertrand, Quentin; Weinert, Tobias; Furrer, Antonia; Glover, Hannah; Gashi, Dardan; Carrillo, Melissa; Kondo, Yasushi; Stipp, Robin T.; Khusainov, Georgii; Nass, Karol; Ozerov, Dmitry; Cirelli, Claudio; Johnson, Philip J. M.; Dworkowski, Florian; Beale, John H.; Stubbs, Scott; Zamofing, Thierry; Schneider, Marco; Krauskopf, Kristina; Gao, Li; Thorn-Seshold, Oliver; Bostedt, Christoph; Bacellar, Camila; Steinmetz, Michel O.; Milne, Christopher; Standfuss, Jorg
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The motor domain of the kinesin Kip2 promotes microtubule polymerization at microtubule tips
err2023-04-24
err2
errOAAI
errChen, Xiuzhen; Portran, Didier; Widmer, Lukas A. A.; Stangier, Marcel M. M.; Czub, Mateusz P. P.; Liakopoulos, Dimitris; Stelling, Jorg; Steinmetz, Michel O. O.; Barral, Yves
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Structural insight into the stabilization of microtubules by taxanes紫杉烷类化合物对微管稳定的结构见解
err2023-03-06
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errOAAI
errProta, Andrea E.; Lucena-Agell, Daniel; Ma, Yuntao; Estevez-Gallego, Juan; Li, Shuo; Bargsten, Katja; Josa-Prado, Fernando; Altmann, Karl-Heinz; Gaillard, Natacha; Kamimura, Shinji; Muhlethaler, Tobias; Gago, Federico; Oliva, Maria A.; Steinmetz, Michel O.; Fang, Wei-Shuo; Diaz, J. Fernando
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Watching the release of a photopharmacological drug from tubulin using time-resolved serial crystallography
err2023-02-17
err16
errOAAI
errWranik, Maximilian; Weinert, Tobias; Slavov, Chavdar; Masini, Tiziana; Furrer, Antonia; Gaillard, Natacha; Gioia, Dario; Ferrarotti, Marco; James, Daniel; Glover, Hannah; Carrillo, Melissa; Kekilli, Demet; Stipp, Robin; Skopintsev, Petr; Brunle, Steffen; Muhlethaler, Tobias; Beale, John; Gashi, Dardan; Nass, Karol; Ozerov, Dmitry; Johnson, Philip J. M.; Cirelli, Claudio; Bacellar, Camila; Braun, Markus; Wang, Meitian; Dworkowski, Florian; Milne, Chris; Cavalli, Andrea; Wachtveitl, Josef; Steinmetz, Michel O. O.; Standfuss, Jorg
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Multivalency ensures persistence of a plus TIP body at specialized microtubule ends
err2022-12-19
err22
errOAAI
errMeier, Sandro M.; Farcas, Ana-Maria; Kumar, Anil; Ijavi, Mahdiye; Bill, Robert T.; Stelling, Joerg; Dufresne, Eric R.; Steinmetz, Michel O.; Barral, Yves
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VASH1-SVBP and VASH2-SVBP generate different detyrosination profiles on microtubules
err2022-12-13
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errOAAI
errRamirez-Rios, Sacnicte; Choi, Sung Ryul; Sanyal, Chadni; Blum, Thorsten B. B.; Bosc, Christophe; Krichen, Fatma; Denarier, Eric; Soleilhac, Jean-Marc; Blot, Beatrice; Janke, Carsten; Stoppin-Mellet, Virginie; Magiera, Maria M. M.; Arnal, Isabelle; Steinmetz, Michel O. O.; Moutin, Marie-Jo
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Changes in seam number and location induce holes within microtubules assembled from porcine brain tubulin and in Xenopus egg cytoplasmic extracts
err2022-12-12
err8
errOAAI
errGuyomar, Charlotte; Bousquet, Clement; Ku, Siou; Heumann, John M.; Guilloux, Gabriel; Gaillard, Natacha; Heichette, Claire; Duchesne, Laurence; Steinmetz, Michel O.; Gibeaux, Romain; Chretien, Denis; Welburn, Julie P., I
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Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas
err2022-12-01
err33
PREAI
errBarreca, Marilia; Span, Virginia; Rocca, Roberta; Bivacqua, Roberta; Abel, Anne -Catherine; Maruca, Annalisa; Montalbano, Alessandra; Raimondi, Maria Valeria; Tarantelli, Chiara; Gaudio, Eugenio; Cascione, Luciano; Rinaldi, Andrea; Bai, Ruoli; Steinmetz, Michel O.; Prota, Andrea E.; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Barraja, Paola
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Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents
err2022-11-01
err19
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errde la Roche, Noelia Montel; Muehlethaler, Tobias; Di Martino, Rita Maria Concetta; Ortega, Jose Antonio; Gioia, Dario; Roy, Bibhas; Prota, Andrea E.; Steinmetz, Michel O.; Cavalli, Andrea
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Rational Design of a Novel Tubulin Inhibitor with a Unique Mechanism of Action具有独特作用机制的新型微管蛋白抑制剂的合理设计
err2022-04-25
err14
errOAAI
errMuhlethaler, Tobias; Milanos, Lampros; Ortega, Jose Antonio; Blum, Thorsten B.; Gioia, Dario; Roy, Bibhas; Prota, Andrea E.; Cavalli, Andrea; Steinmetz, Michel O.
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