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Cardiac human bitter taste receptors contain naturally occurring variants that alter function Bloxham, Conor J.; Hulme, Katina D.; Fierro, Fabrizio; Fercher, Christian; Pegg, Cassandra L.; O'Brien, Shannon L.; Foster, Simon R.; Short, Kirsty R.; Furness, Sebastian G. B.; Reichelt, Melissa E.; Niv, Masha Y.; Thomas, Walter G. 分享 收藏
Acid-sensing ion channel 1a blockade reduces myocardial injury in rodent models of myocardial infarction 酸敏感离子通道1a阻断可减轻啮齿动物心肌梗死模型的心肌损伤 Redd, Meredith A.; Yoshikawa, Yusuke; Khan, Nemat; Waqar, Maleeha; Saez, Natalie J.; Outhwaite, Jennifer E.; Russell, Jake S.; Hanna, Amy D.; Chiu, Han S.; Er, Sing Yan; Butcher, Neville J.; Mardon, Karine; Fraser, John F.; Smythe, Mark L.; Rash, Lachlan D.; Thomas, Walter G.; King, Glenn F.; Reichelt, Melissa E.; Palpant, Nathan J. 分享 收藏
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A peptide toxin in ant venom mimics vertebrate EGF-like hormones to cause long-lasting in mammals 蚂蚁毒液中的肽毒素模仿脊椎动物EGF样激素,在哺乳动物中引起持久 Eagles, David A.; Saez, Natalie J.; Krishnarjuna, Bankala; Bradford, Julia J.; Chin, Yanni K. -Y.; Starobova, Hana; Mueller, Alexander; Reichelt, Melissa E.; Undheim, Eivind A. B.; Norton, Raymond S.; Thomas, Walter G.; Vetter, Irina; King, Glenn F.; Robinson, Samuel D. 分享 收藏
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BRET-based assay to monitor EGFR transactivation by the AT1R reveals Gq/11 protein-independent activation and AT1R-EGFR complexes (vol 158, pg 232, 2018) O'Brien, Shannon L.; Johnstone, Elizabeth K. M.; Devost, Dominic; Conroy, Jacinta; Reichelt, Melissa E.; Purdue, Brooke W.; Ayoub, Mohammed A.; Kawai, Tatsuo; Inoue, Asuka; Eguchi, Satoru; Hebert, Terence E.; Pfleger, Kevin D. G.; Thomas, Walter G. 分享 收藏
Therapeutic Inhibition of Acid-Sensing Ion Channel 1a Recovers Heart Function After Ischemia-Reperfusion Injury Redd, Meredith A.; Scheuer, Sarah E.; Saez, Natalie J.; Yoshikawa, Yusuke; Chiu, Han Sheng; Gao, Ling; Hicks, Mark; Villanueva, Jeanette E.; Joshi, Yashutosh; Chow, Chun Yuen; Cuellar-Partida, Gabriel; Peart, Jason N.; Hoe, Louise E. See; Chen, Xiaoli; Sun, Yuliangzi; Suen, Jacky Y.; Hatch, Robert J.; Rollo, Ben; Xia, Di; Alzubaidi, Mubarak A. H.; Maljevic, Snezana; Quaife-Ryan, Gregory A.; Hudson, James E.; Porrello, Enzo R.; White, Melanie Y.; Cordwell, Stuart J.; Fraser, John F.; Petrou, Steven; Reichelt, Melissa E.; Thomas, Walter G.; King, Glenn F.; Macdonald, Peter S.; Palpant, Nathan J. 分享 收藏
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Modular transient nanoclustering of activated β2-adrenergic receptors revealed by single-molecule tracking of conformation-specific nanobodies Gormal, Rachel S.; Padmanabhan, Pranesh; Kasula, Ravikiran; Bademosi, Adekunle T.; Coakley, Sean; Giacomotto, Jean; Blum, Ailisa; Joensuu, Merja; Wallis, Tristan P.; Lo, Harriet P.; Budnar, Srikanth; Rae, James; Ferguson, Charles; Bastiani, Michele; Thomas, Walter G.; Pardon, Els; Steyaert, Jan; Yap, Alpha S.; Goodhill, Geoffrey J.; Hilliard, Massimo A.; Parton, Robert G.; Meunier, Frederic A. 分享 收藏
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A High-Fat Diet Increases Influenza A Virus-Associated Cardiovascular Damage Siegers, Jurre Y.; Novakovic, Boris; Hulme, Katina D.; Marshall, Rebecca J.; Bloxham, Conor J.; Thomas, Walter G.; Reichelt, Mellissa E.; Leijten, Lonneke; van Run, Peter; Knox, Karen; Sokolowski, Kamil A.; Tse, Brian W. C.; Chew, Keng Yih; Christ, Angelika N.; Howe, Greg; Bruxner, Timothy J. C.; Karolyi, Mario; Pawelka, Erich; Koch, Rebecca M.; Bellmann-Weiler, Rosa; Burkert, Francesco; Weiss, Gunter; Samanta, Romit J.; Openshaw, Peter J. M.; Bielefeldt-Ohmann, Helle; van Riel, Debby; Short, Kirsty R. 分享 收藏
THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein-coupled receptors 药理学2019/20简明指南: g蛋白偶联受体 Alexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Sharman, Joanna L.; Southan, Christopher; Davies, Jamie A.; Arumugam, Thiruma V.; Bennett, Andrew; Sjogren, Benita; Sobey, Christopher; Wong, Szu Shen; Abbracchio, Maria P.; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Beaulieu, Jean-Martin; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chun, Jerold; Cianciulli, Antonia; Clapp, Lucie H.; Couture, Rejean; Csaba, Zsolt; Dent, Gordon; Singh, Khuraijam Dhanachandra; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward; Fong, Tung M.; Fumagalli, Marta; Gainetdinov, Raul R.; de Gasparo, Marc; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie; Heinemann, Akos; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence; Mitolo, Vincenzo; Mouillac, Bernard; Murphy, Philip M.; Nahon, Jean-Louis; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria A.; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric; Ramachandran, Rithwik; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie; Thomas, Walter; Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Aldrich, Richard W.; Becirovic, Elvir; Biel, Martin; Catterall, William A.; Conner, Alex C.; Davies, Paul; Delling, Markus; Di Virgilio, Francesco; Falzoni, Simonetta; George, Chandy; Goldstein, Steve A. N.; Grissmer, Stephan; Ha, Kotdaji; Hammelmann, Verena; Hanukoglu, Israel; Jarvis, Mike; Jensen, Anders A.; Kaczmarek, Leonard K.; Kellenberger, Stephan; Kennedy, Charles; King, Brian; Lynch, Joseph W.; Perez-Reyes, Edward; Plant, Leigh D.; Rash, Lachlan D.; Ren, Dejian; Sivilotti, Lucia G.; Smart, Trevor G.; Snutch, Terrance P.; Tian, Jinbin; Van den Eynde, Charlotte; Vriens, Joris; Wei, Aguan D.; Winn, Brenda T.; Wulff, Heike; Xu, Haoxing; Yue, Lixia; Zhang, Xiaoli; Zhu, Michael; Coons, Laurel; Fuller, Peter; Korach, Kenneth S.; Young, Morag; Bryant, Clare; Farndale, Richard W.; Hobbs, Adrian; Jarvis, Gavin E.; MacEwan, David; Monie, Tom P.; Waldman, Scott; Beuve, Annie; Boison, Detlev; Brouckaert, Peter; Burnett, John C.; Burns, Kathryn; Dessauer, Carmen; Friebe, Andreas; Garthwaite, John; Gertsch, Jurg; Helsby, Nuala; Izzo, Angelo A.; Koesling, Doris; Kuhn, Michaela; Ostrom, Rennolds; Papapetropoulos, Andreas; Potter, Lincoln R.; Pyne, Nigel J.; Pyne, Susan; Russwurm, Michael; Schmidt, Harald H. H. W.; Seifert, Roland; Stasch, Johannes-Peter; Szabo, Csaba; van der Stelt, Mario; van der Vliet, Albert; Watts, Val; Anderson, Catriona M. H.; Broer, Stefan; Dawson, Paul; Hagenbuch, Bruno; Hammond, James R.; Hancox, Jules; Inui, Ken-ichi; Kanai, Yoshikatsu; Kemp, Stephan; Thwaites, David T.; Verri, Tiziano 分享 收藏
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BRET-based assay to monitor EGFR transactivation by the AT1R reveals Gq/11 protein-independent activation and AT1R-EGFR complexes O'Brien, Shannon L.; Johnstone, Elizabeth K. M.; Devost, Dominic; Conroy, Jacinta; Reichelt, Melissa E.; Purdue, Brooke W.; Ayoub, Mohammed A.; Kawai, Tatsuo; Inoue, Asuka; Eguchi, Satoru; Hebert, Terence E.; Pfleger, Kevin D. G.; Thomas, Walter G. 分享 收藏
Functional screening in human cardiac organoids reveals a metabolic mechanism for cardiomyocyte cell cycle arrest Mills, Richard J.; Titmarsh, Drew M.; Koenig, Xaver; Parker, Benjamin L.; Ryall, James G.; Quaife-Ryan, Gregory A.; Voges, Holly K.; Hodson, Mark P.; Ferguson, Charles; Drowley, Lauren; Plowright, Alleyn T.; Needham, Elise J.; Wang, Qing-Dong; Gregorevic, Paul; Xin, Mei; Thomas, Walter G.; Parton, Robert G.; Nielsen, Lars K.; Launikonis, Bradley S.; James, David E.; Elliott, David A.; Porrello, Enzo R.; Hudson, James E. 分享 收藏
Cavin-1 deficiency modifies myocardial and coronary function, stretch responses and ischaemic tolerance: roles of NOS over-activity Kaakinen, Mika; Reichelt, Melissa E.; Ma, Zhibin; Ferguson, Charles; Martel, Nick; Porrello, Enzo R.; Hudson, James E.; Thomas, Walter G.; Parton, Robert G.; Headrick, John P. 分享 收藏
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Gaq proteins: molecular pharmacology and therapeutic potential Kamato, Danielle; Mitra, Partha; Davis, Felicity; Osman, Narin; Chaplin, Rebecca; Cabot, Peter J.; Afroz, Rizwana; Thomas, Walter; Zheng, Wenhua; Kaur, Harveen; Brimble, Margaret; Little, Peter J. 分享 收藏