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D

David W. Gray

University of Dundee

H指数:34

被引数:4,989

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Small-molecule inhibitors block NorA efflux by conformational trapping

小分子抑制剂通过构象捕获阻断NorA外排

Nature Chemical Biology

IF13.7

2026-09-160

OAAI

Experience from an HTS campaign: Investigation of susceptibility and rescue of SARS-CoV-2 nsp3 protease assay from metal contamination

高通量筛选（HTS）实验的经验：SARS-CoV-2 nsp3蛋白酶检测试剂盒对金属污染的敏感性与修复研究

SLAS Technology

IF3.7

2026-03-130

OAAI

Characterisation of RNA guanine-7 methyltransferase (RNMT) using a small molecule approach

BIOCHEMICAL JOURNAL

IF4.3

2025-02-170

OAAI

Pharmacological and structural understanding of the Trypanosoma cruzi proteasome provides key insights for developing site-specific inhibitors

JOURNAL OF BIOLOGICAL CHEMISTRY

IF3.9

2025-01-011

PRE

Identification and Validation of Compounds Targeting Leishmania major Leucyl-Aminopeptidase M17

ACS INFECTIOUS DISEASES

IF3.8

2024-05-161

OAAI

Application of an NMR/Crystallography Fragment Screening Platform for the Assessment and Rapid Discovery of New HIV-CA Binding Fragments

IF3.4

2024-05-061

OAAI

Identification of a potent and selective LAPTc inhibitor by RapidFire-Mass Spectrometry, with antichagasic activity

PLOS NEGLECTED TROPICAL DISEASES

IF3.4

2024-02-151

OAAI

Design of the Global Health chemical diversity library v2 for screening against infectious diseases

PLOS NEGLECTED TROPICAL DISEASES

IF3.4

2023-12-274

OAAI

Design and Synthesis of Covalent Inhibitors of FabA

IF4.3

2023-03-270

OAAI

Assessment of the drugability of initial malaria infection through miniaturized sporozoite assays and high-throughput screening

COMMUNICATIONS BIOLOGY

IF5.1

2023-02-237

OAAI

Live-imaging rate-of-kill compound profiling for Chagas disease drug discovery with a new automated high-content assay

PLOS NEGLECTED TROPICAL DISEASES

IF3.4

2021-10-116

OAAI

Structure-Activity Relationships of Pyrazolo[1,5-a]pyrimidin-7(4H)-ones as Antitubercular Agents

ACS INFECTIOUS DISEASES

IF3.8

2021-01-0614

OAAI

Targeting N-myristoylation for therapy of B-cell lymphomas

NATURE COMMUNICATIONS

IF15.7

2020-10-2243

OAAI

Targeting N-myristoylation in B-cell lymphomas as a therapeutic strategy

CANCER RESEARCH

IF16.6

2020-08-150

PRE

Discovery of an Allosteric Binding Site in Kinetoplastid Methionyl-tRNA Synthetase

ACS INFECTIOUS DISEASES

IF3.8

2020-04-1013

OAAI

Novel pharmacological actions of trequinsin hydrochloride improve human sperm cell motility and function

BRITISH JOURNAL OF PHARMACOLOGY

IF7.7

2019-12-1123

OAAI

Trypanosoma cruzi Phosphomannomutase and Guanosine Diphosphate-Mannose Pyrophosphorylase Ligandability Assessment

克氏锥虫磷酸变位酶和二磷酸鸟苷-甘露糖焦磷酸化酶可连接性评估

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2019-10-016

OAAI

Identification of Novel Trypanosoma cruzi Proteasome Inhibitors Using a Luminescence-Based High-Throughput Screening Assay

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2019-09-0116

OAAI

Burkholderia pseudomallei d-alanine-d-alanine ligase; detailed characterisation and assessment of a potential antibiotic drug target

IF4.2

2019-07-165

OAAI

Substituted Aminoacetamides as Novel Leads for Malaria Treatment

IF3.4

2019-07-036

OAAI

Norcross, Neil R.; Wilson, Caroline; Baragana, Beatriz; Hallyburton, Irene; Osuna-Cabello, Maria; Norval, Suzanne; Riley, Jennifer; Fletcher, Daniel; Sinden, Robert; Delves, Michael; Ruecker, Andrea; Duffy, Sandra; Meister, Stephan; Antonova-Koch, Yevgeniya; Crespo, Benigno; de Cozar, Cristina; Sanz, Laura M.; Javier Gamo, Francisco; Avery, Vicky M.; Frearson, Julie A.; Gray, David W.; Fairlamb, Alan H.; Winzeler, Elizabeth A.; Waterson, David; Campbell, Simon F.; Willis, Paul A.; Read, Kevin D.; Gilbert, Ian H.