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Synthesis of Tricyclic and Tetracyclic Lactone Derivatives of Thieno[2,3-b]pyrazine or Thieno[2,3-b]quinoline: Preliminary Antitumor and Antiparasitic Activity Evaluation Thieno[2,3-b]pyrazine或Thieno[2,3-b]quinoline类三环和四环内酯衍生物的合成:初步抗肿瘤和抗寄生虫活性评价 Martins, Maria F.; Ribeiro, Francisco; Borges, Ana; Calhelha, Ricardo C.; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Queiroz, Maria-Joao R. P. 分享 收藏
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SAR Study of 4,8-Disubstituted Pyrimido[5,4-d]pyrimidines Exhibiting Antitrypanosomal and Antileishmanial Activity 具有抗锥虫和抗利什曼活性的4,8-二取代嘧啶并 [5,4-d] 嘧啶的SAR研究 Lopes, Andre; Teixeira, Sofia; Santarem, Nuno; Greco, Alessandro; Pagliaro, Angela; Keminer, Oliver; Gul, Sheraz; Cordeiro-da-Silva, Anabela; Carvalho, Maria Alice 分享 收藏
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Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents 鉴定利用环胍的氨基二氢三嗪基序作为抗布氏锥虫剂的创新叶酸抑制剂 Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Simo, Claude U. Konchie; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarem, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele 分享 收藏
Discovery of 1,3,4-Oxadiazole Derivatives as Broad-Spectrum Antiparasitic Agents 1,3,4-恶二唑衍生物作为广谱抗寄生虫药的发现 Corfu, Alexandra Ioana; Santarem, Nuno; Luelmo, Sara; Mazza, Gaia; Greco, Alessandro; Altomare, Alessandra; Ferrario, Giulio; Nasta, Giulia; Keminer, Oliver; Aldini, Giancarlo; Tamborini, Lucia; Basilico, Nicoletta; Parapini, Silvia; Gul, Sheraz; Cordeiro-da-Silva, Anabela; Conti, Paola; Borsari, Chiara 分享 收藏
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The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents aryl-2-nitroethyl三氨基嘧啶作为抗布氏锥虫剂的发现 Linciano, Pasquale; Pozzi, Cecilia; Tassone, Giusy; Landi, Giacomo; Mangani, Stefano; Santucci, Matteo; Luciani, Rosaria; Ferrari, Stefania; Santarem, Nuno; Tagliazucchi, Lorenzo; Cordeiro-da-Silva, Anabela; Tonelli, Michele; Tondi, Donatella; Bertarini, Laura; Gul, Sheraz; Witt, Gesa; Moraes, Carolina B.; Costantino, Luca; Costi, Maria Paola 分享 收藏
High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents Linciano, Pasquale; Quotadamo, Antonio; Luciani, Rosaria; Santucci, Matteo; Zorn, Kimberley M.; Foil, Daniel H.; Lane, Thomas R.; da Silva, Anabela Cordeiro; Santarem, Nuno; Moraes, Carolina B.; Freitas-Junior, Lucio; Wittig, Ulrike; Mueller, Wolfgang; Tonelli, Michele; Ferrari, Stefania; Venturelli, Alberto; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Ekins, Sean; Costi, Maria Paola 分享 收藏
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