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Regioselective synthesis of aza-saccharins via anionic [1; 4] Fries-type rearrangement of aryl sulfonimidoyl fluorides
err2026-04-29
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errOAAI
errMario Leypold; Lorenzo Poli; Max Earl; Okky D. Putra; Karolina Kwapien; Richard J. Lewis; John J. Murphy; Marta Passamonti; Lena M. von Sydow; Victor Spelling; Ioannis Asproudis; Malvika Sardana; Claudia Gatti; Hikaru Seki; Thomas Lemaitre; Radvile Juskaite; Ranganath Gopalakrishnan; Stuart J. Francis; Cristina Gardelli; Per-Ola Norrby; Werngard Czechtizky
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DMPK Considerations for the Development of Covalent Drugs: Insights from an IQ Assessment
err2026-04-28
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PREAI
errJulian Dopstadt; Kamelia Behnia; Xiaoming Cui; Nicola Colclough; Martin Dowty; Julius Enoru; Robert S. Foti; Felix Huth; Frank Jacobs; Rohitash Jamwal; Benjamin M. Johnson; Shyam Kamble; Julie Lade; Sandhya Mandlekar; Hlaing Holly Maw; Kowser Miah; Mike Mohutsky; Holger Scheible; Hao Sun; Shuai Wang; Matthias Beat Wittwer; Sean Xiaochun Zhu; Stefanie Zimmermann; Rowan Stringer
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Purge Factor Analysis and Proposal for Non-conjugatable Impurity Clearance in Post-conjugation Purification of ADCs
err2026-04-28
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PREAI
errLara Fernandez-Cerezo; Osama Chahrour; Seb Caille; Andrew M. Poulton; Chloe Westley; Lan Yang; Melissa Holstein; Petr Jirasek; Pavlo Kos; Paul G. Bulger
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A plain language review of results from the LAURA study: osimertinib after chemoradiotherapy for patients with EGFR-mutated non-small cell lung cancer that cannot be removed by surgery
err2026-04-27
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errShun Lu; Terufumi Kato; Xiaorong Dong; Myung-Ju Ahn; Le-Van Quang; Nopadol Soparattanapaisarn; Takako Inoue; Chih-Liang Wang; Meijuan Huang; James Chih-Hsin Yang; Manuel Cobo; Mustafa Özgüroğlu; Ignacio Casarini; Virote Sriuranpong; Eduardo Cronemberger; Toshiaki Takahashi; Yotsawaj Runglodvatana; Ming Chen; Xiangning Huang; Ellie Grainger; Dana Ghiorghiu; Toon van der Gronde; Suresh S Ramalingam
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Effects of Dapagliflozin on Cardiovascular Outcomes in Patients With Type 2 Diabetes at Risk of Liver Fibrosis
err2026-04-27
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errJan Oscarsson; Monika Huhn; Yunyun Jiang; Ingrid Gause-Nilsson; Stephen D. Wiviott; Filipe A. Moura; John P. H. Wilding; Simona Cernea; Luc Van Gaal; Avivit Cahn; Deepak L. Bhatt; Peter A. Johansson; C. David Sjöström
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Enhancement of a nuclear factor of activated T cells (NFAT) reporter for the study of G protein-coupled receptors
err2026-04-26
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errEdward Wills; Anjana Saji; Jonathan Sumner; Aman Khan; Claudia M. Sisk; Mona Shehata; Benjamin Taylor; Graham Ladds
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Intestinal Organoid-Based Mathematical Modeling Predicts Clinical Gastrointestinal Toxicity of Oral Oncology Drugs
err2026-04-25
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errCarmen Pin; Deepa Maheshvare M.; Louis Gall; Andrew Hall; Muireann Coen; Ambra Bianco; Shimeng Liu; Kenneth Pryde
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Switchable N–H vs. C3–H carboxylation of indoles using dual-function reagents
err2026-04-17
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errKatherine E. Marris; Jazmine T. Thorne; Daniel J. Ryder-Mahoney; Ryan A. Bragg; Charles S. Elmore; Gregory J. P. Perry
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Preclinical characterization of AZD1163, a first-in-class anti-PAD2/4 bispecific antibody for the treatment of rheumatoid arthritis
errmAbs
IF7.3
err2026-04-15
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errOAAI
errGary P. Sims; Lacie Scaletta; John Andrews; Dorothy A. Sims; Martin Strain; Anna Sigurdardottir; Teneema Kuriakose; Elizabeth England; Lichchavi Rajasinghe; Fanyi Jiang; Ximing Xiong; Frances Neal; Lisa Vinall; Philip Newton; Elin Boger; Chong Kim; Helena Dahlbäck; Susanne Prothon; Jacob Leander; Erika Darrah; Mia Collins; Garry Douglas; Nicholas White; Katie Day; Katherine A. Vousden; Catherine E. Huntington; David Close
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Biophysical Modeling Elucidates Mechanistic Principles for Rational Molecular Glue Design
err2026-04-13
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errOAAI
errSeok Joo Chae; Jonathon DeBonis; Joseph Quinlan; Ryan Richards; Junmin Wang; Gustavo Gutierrez; Jonathan Tart; Maxime Couturier; Sergio Martinez Cuesta; Meizhong Jin; Oleg A. Igoshin
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A first-in-human Phase 1/1b randomized trial evaluating the safety and immunogenicity of a respiratory syncytial virus (RSV) virus-like particle subunit vaccine (IVX-121) in healthy young and older adults
err2026-03-03
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errIlse De Coster; Isabel Leroux-Roels; Kanchanamala Withanage; Leen Suykens; Valentino D’Onofrio; Geert Leroux-Roels; Pierre van Damme; Max Ciarlet; Elizabeth M. Adams; Wasima Rida; Judy Wen; Margaret MacDonald; Jennifer Price; Niranjan Kanesa-thasan
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Osimertinib after definitive chemoradiotherapy in patients with unresectable stage III EGFR-mutated NSCLC: LAURA China cohort
err2026-02-23
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errOAAI
errXiaorong Dong; Hong Jian; Meijuan Huang; Shuanghu Yuan; Zhengfei Zhu; Lin Wu; Ming Chen; Nan Bi; Yi Pan; Yingyi Wang; Dongqing Lv; Elena Armenteros Monterroso; Xiangning Huang; Rui Mao; Wei Fu; Yi Zhao; Shun Lu
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Automated DFT-Machine Learning Integration Enables Data-Efficient and Generalizable Feasibility Predictions in Metallaphotoredox sp2–sp3 Cross-Coupling Reactions
err2026-02-10
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PREAI
errMichele Assante; Sara Pahlen; Brenda Pijper; Lili Cao; Ole Specht; Nadja Simeth; Alexei Lapkin; Clive Green; Ola Engkvist; Giulia Bergonzini; Mikhail Kabeshov
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Camizestrant in combination with capivasertib for women with ER-positive, HER2-negative advanced breast cancer: results from SERENA-1☆
err2026-01-21
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errC. Vaklavas; M. Oliveira; A.C. Armstrong; I. Moreno; C. Twelves; I. Victoria Ruiz; B. Bermejo de las Heras; T. Brier; C. Ciardullo; L. Gibbons; T. Jack; T. Klinowska; J.P.O. Lindemann; A.M. Mathewson; R. Maudsley; C.J. Morrow; A. Sykes; R.D. Baird
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