Not logged in
Share
Save
Share
SaveDiscovery of a novel, selective CK2 inhibitor class with an unusual basic scaffold
Khalifa, Hend; ElHady, Ahmed K.; Liu, Ting; Elgaher, Walid A. M.; Filhol-Cochet, Odile; Cochet, Claude; Abadi, Ashraf H.; Hamed, Mostafa M.; Abdel-Halim, Mohammad; Engel, Matthias
Share
Save
Share
SaveGIMAP5 deficiency reveals a mammalian ceramide-driven longevity assurance pathway (vol 25, pg 282, 2024)
Park, Ann Y.; Leney-Greene, Michael; Lynberg, Matthew; Gabrielski, Justin Q.; Xu, Xijin; Schwarz, Benjamin; Zheng, Lixin; Balasubramaniyam, Arasu; Ham, Hyoungjun; Chao, Brittany; Zhang, Yu; Matthews, Helen F.; Cui, Jing; Yao, Yikun; Kubo, Satoshi; Chanchu, Jean Michel; Morawski, Aaron R.; Cook, Sarah A.; Jiang, Ping; Ravell, Juan C.; Cheng, Yan H.; George, Alex; Faruqi, Aiman; Pagalilauan, Alison M.; Bergerson, Jenna R. E.; Ganesan, Sundar; Chauvin, Samuel D.; Aluri, Jahnavi; Edwards-Hicks, Joy; Bohrnsen, Eric; Tippett, Caroline; Omar, Habib; Xu, Leilei; Butcher, Geoffrey W.; Pascall, John; Karakoc-Aydiner, Elif; Kiykim, Ayca; Maecker, Holden; Tezcan, Ilhan; Esenboga, Saliha; Heredia, Raul Jimenez; Akata, Deniz; Tekin, Saban; Kara, Altan; Kuloglu, Zarife; Unal, Emel; Kendirli, Tanil; Dogu, Figen; Karabiber, Esra; Atkinson, T. Prescott; Cochet, Claude; Filhol, Odile; Bosio, Catherine M.; Davis, Mark M.; Lifton, Richard P.; Pearce, Erika L.; Daumke, Oliver; Aytekin, Caner; Sahin, Gulseren Evirgen; Aksu, Aysel Unlusoy; Uzel, Gulbu; Rao, V. Koneti; Sari, Sinan; Dalgic, Buket; Boztug, Kaan; Cagdas, Deniz; Haskologlu, Sule; Ikinciogullari, Aydan; Schwefel, David; Vilarinho, Silvia; Baris, Safa; Ozen, Ahmet; Su, Helen C.; Lenardo, Michael J.
Share
SaveGIMAP5 deficiency reveals a mammalian ceramide-driven longevity assurance pathway
Park, Ann Y.; Leney-Greene, Michael; Lynberg, Matthew; Gabrielski, Justin Q.; Xu, Xijin; Schwarz, Benjamin; Zheng, Lixin; Balasubramaniyam, Arasu; Ham, Hyoungjun; Chao, Brittany; Zhang, Yu; Matthews, Helen F.; Cui, Jing; Yao, Yikun; Kubo, Satoshi; Chanchu, Jean Michel; Morawski, Aaron R.; Cook, Sarah A.; Jiang, Ping; Ravell, Juan C.; Cheng, Yan H.; George, Alex; Faruqi, Aiman; Pagalilauan, Alison M.; Bergerson, Jenna R. E.; Ganesan, Sundar; Chauvin, Samuel D.; Aluri, Jahnavi; Edwards-Hicks, Joy; Bohrnsen, Eric; Tippett, Caroline; Omar, Habib; Xu, Leilei; Butcher, Geoffrey W.; Pascall, John; Karakoc-Aydiner, Elif; Kiykim, Ayca; Maecker, Holden; Tezcan, Ilhan; Esenboga, Saliha; Heredia, Raul Jimenez; Akata, Deniz; Tekin, Saban; Kara, Altan; Kuloglu, Zarife; Unal, Emel; Kendirli, Tanil; Dogu, Figen; Karabiber, Esra; Atkinson, T. Prescott; Cochet, Claude; Filhol, Odile; Bosio, Catherine M.; Davis, Mark M.; Lifton, Richard P.; Pearce, Erika L.; Daumke, Oliver; Aytekin, Caner; Sahin, Guelseren Evirgen; Aksu, Aysel uenluesoy; Uzel, Gulbu; Koneti Rao, V.; Sari, Sinan; Boztug, Kaan; Cagdas, Deniz; Haskologlu, Sule; Ikinciogullari, Aydan; Schwefel, David; Vilarinho, Silvia; Baris, Safa; Ozen, Ahmet; Su, Helen C.; Lenardo, Michael J.
Share
SaveA new scaffold-free tumoroid model provides a robust preclinical tool to investigate invasion and drug response in Renal Cell Carcinoma
Seraudie, Irinka; Pillet, Catherine; Cesana, Beatrice; Bazelle, Pauline; Jeanneret, Florian; Evrard, Bertrand; Chalmel, Frederic; Bouzit, Assilah; Battail, Christophe; Long, Jean-Alexandre; Descotes, Jean Luc; Cochet, Claude; Filhol, Odile
Share
Save
Share
Save
Share
Save
Share
Save
Share
SaveCIGB-300 anticancer peptide regulates the protein kinase CK2-dependent phosphoproteome
Perera, Yasser; Ramos, Yassel; Padron, Gabriel; Caballero, Evelin; Guirola, Osmany; Caligiuri, Lorena G.; Lorenzo, Norailys; Gottardo, Florencia; Farina, Hernan G.; Filhol, Odile; Cochet, Claude; Perea, Silvio E.
Share
SaveDiscovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors
Kufareva, Irina; Bestgen, Benoit; Brear, Paul; Prudent, Renaud; Laudet, Beatrice; Moucadel, Virginie; Ettaoussi, Mohamed; Sautel, Celine F.; Krimm, Isabelle; Engel, Matthias; Filhol, Odile; Le Borgne, Marc; Lomberget, Thierry; Cochet, Claude; Abagyan, Ruben
Share
Save2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action
Bestgen, Benoit; Kufareva, Irina; Seetoh, Weiguan; Abell, Chris; Hartmann, Rolf W.; Abagyan, Ruben; Le Borgne, Marc; Filhol, Odile; Cochet, Claude; Lomberget, Thierry; Engel, Matthias
Share
Save2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 1. Identification of an Allosteric Binding Site
Bestgen, Benoit; Krimm, Isabelle; Kufareva, Irina; Kamal, Ahmed Ashraf Moustafa; Seetoh, Wei-Guang; Abell, Chris; Hartmann, Rolf W.; Abagyan, Ruben; Cochet, Claude; Le Borgne, Marc; Engel, Matthias; Lomberget, Thierry
Share
SaveTRIM17 and TRIM28 antagonistically regulate the ubiquitination and anti-apoptotic activity of BCL2A1
Lionnard, Loic; Duc, Pauline; Brennan, Margs S.; Kueh, Andrew J.; Pal, Martin; Guardia, Francesca; Mojsa, Barbara; Damiano, Maria-Alessandra; Mora, Stephan; Lassot, Irena; Ravichandran, Ramya; Cochet, Claude; Aouacheria, Abdel; Potts, Patrick Ryan; Herold, Marco J.; Desagher, Solange; Kucharczak, Jerome
Share
SaveThe tyrosine-kinase inhibitor sunitinib targets vascular endothelial (VE)-cadherin: a marker of response to antitumoural treatment in metastatic renal cell carcinoma
Polena, Helena; Creuzet, Julie; Dufies, Maeva; Sidibe, Adama; Khalil-Mgharbel, Abir; Salomon, Aude; Deroux, Alban; Quesada, Jean-Louis; Roelants, Caroline; Filhol, Odile; Cochet, Claude; Blanc, Ellen; Ferlay-Segura, Celine; Borchiellini, Delphine; Ferrero, Jean-Marc; Escudier, Bernard; Negrier, Sylvie; Pages, Gilles; Vilgrain, Isabelle
Share
Save
Share
SaveProtein kinase CK2 controls T-cell polarization through dendritic cell activation in response to contact sensitizers
de Bourayne, Marie; Gallais, Yann; El Ali, Zeina; Rousseau, Philippe; Damiens, Marie-Helene; Cochet, Claude; Filhol, Odile; Chollet-Martin, Sylvie; Pallardy, Marc; Kerdine-Romer, Saadia
Share
Save
Share
Save