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Stefan Knapp

dkfz and uct frankfurt-marburg

111H-index
1.3KPaper Count
4.8WCitation Count
Published Papers 408
Publication Date
USP22 is a novel vulnerability regulating MEIS1 protein abundance and gene transcription in KMT2Ar acute leukemia
errBlood
IF23.1
err2026-07-09
err0
PREAI
errSarah Bröchtel; Constanze Schneider; Marius Müller; Christina Villinger; Thomas Plenge; Manoj K. Gupta; Luca Immanuel Kesel; Sebastian Scheich; Sebastian Wolf; Ali Yavuz Cakir; Björn Häupl; Florian Büttner; Stefan Knapp; Hubert Serve; Kimberly Stegmaier; Florian Perner; Thomas Oellerich; Anjali Cremer
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First Structure–Activity-Relationship Study of Potent G2A Antagonists
err2026-06-11
err0
errOAAI
errVictor Hernandez-Olmos; Jan Heering; Felix F. Lillich; Beatrice Marinescu; Sheila Nevermann; Johanna H. M. Ehrler; Dmytro S. Radchenko; Yurii S. Moroz; Astrid Kaiser; Andreas Krämer; Stefan Knapp; Manfred Schubert-Zsilavecz; Mohamad Wessam Alnouri; Stefan Offermanns; Dieter Steinhilber; Marco Sisignano; Ewgenij Proschak
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Identification and Validation of 3-Cyano-Quinoline Ligands Targeting Integrin-Linked Kinase (ILK)
err2026-05-25
err0
errOAAI
errFrancesco Aleksy Greco; Kamal Rayees Abdul Azeez; Marko Mitrović; Saran Aswathaman Sivashanmugam; Martin Peter Schwalm; Franziska Preuss; Deep Chatterjee; Viktoria Morasch; Sebastian Mathea; Thomas Hanke; Susanne Müller; Stefan Knapp
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Targeted degradation of USP7 in solid cancer cells reveals distinct effects of deubiquitinase degraders and inhibitors
err2026-05-13
err0
errOAAI
errNikolas Klink; Sebastian Urban; Johanna A. Seier; Bikash Adhikari; Martin P. Schwalm; Juliane Müller; Madeleine Dorsch; Philine Steinbach; Jennifer Jung; Markus Vogt; Farnusch Kaschani; Johannes Koch; Siska Führer; Markus Kaiser; Nina Schulze; Stefan Knapp; Elmar Wolf; Annette Paschen; Barbara M. Grüner; Malte Gersch
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Discovery and Development of a Potent LIMK2 Isoform-Specific Degrader
err2026-05-01
err0
errOAAI
errKamal Rayees Abdul Azeez; Hayuningbudi Saraswati; Thorsten Mosler; Thomas Hanke; Hung Ho-Xuan; Noah Neder; Saran Aswathaman Sivashanmugam; Marcel Heinz; Martin-Peter Schwalm; Giulio Giuliani; Rajeshwari Rathore; Rubina Kazi; Rahul Kumar; Marko Mitrovic; Cristian Prieto-Garcia; Henry J. Bailey; Sebastian Mathea; Gerhard Hummer; Ivan Đikić; Susanne Müller; Alexandra Stolz; Daniela S Krause; Stefan Knapp
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Structure Merging Approach Leads to New Dual Potent and Selective USP25/USP28 Inhibitors
err2026-04-22
err0
errOAAI
errVictor Hernandez-Olmos; Jonathan Vincent Patzke; Caroline E. Stone; Radhika Karal Nair; Kathrin Weller; Florian Sauer; Erik Endres; Oumaima Jamai; Lea Rachor; Cornelia H. Warmutz; Martin P. Schwalm; Marko Mitrovic; Vincent Grenier; Johanna H. M. Ehrler; Anna Proschak; Jan Heering; Christoph Sotriffer; Monique P. C. Mulder; Stefan Knapp; Caroline Kisker; Ewgenij Proschak
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Discovery of APO-50815, a Potent WEE1 Kinase Inhibitor with Exceptional Efficacy against Patient-Derived Colorectal Cancer Organoids
err2026-04-05
err0
PREAI
errJoel L. Syphers; Josephine A. Wright; Rebekah de Nys; Tharindie N. Silva; Laura Vrbanac; Katherine Barratt; Julia Leeflang; Sadia Hasan; Sophie F. Thomson; Adarsh Kumar; Andreas Krämer; Christopher Lenz; Yi Sing Gee; Aeson Chang; Savannah Young; Erica K. Sloan; Stefan Knapp; Daniel L. Worthley; Siddhartha Mukherjee; Kieran Stockton
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Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery
err2026-01-23
err0
errOAAI
errMarko Mitrović; Francesco Aleksy Greco; Yiliam Cruz García; Aleksandar Lučić; Lasse Hoffmann; Rohit Chander; Julia Schönfeld; Nick Liebisch; Saran Aswathaman Sivashanmugam; Martin Peter Schwalm; Markus Egner; Max Lewandowski; Daniel Merk; Viktoria Morasch; Elmar Wolf; Susanne Müller; Thomas Hanke; Ewgenij Proschak; Kerstin Hiesinger; Stefan Knapp
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Enantioselective protein affinity selection mass spectrometry (E-ASMS)
err2025-12-17
err0
errOAAI
errXiaoyun Wang; Jianxian Sun; Shabbir Ahmad; Diwen Yang; Fengling Li; U. Hang Chan; Hong Zeng; Conrad V. Simoben; Stuart R. Green; Madhushika Silva; Scott Houliston; Aiping Dong; Albina Bolotokova; Elisa Gibson; Maria Kutera; Pegah Ghiabi; Ivan Kondratov; Tetiana Matviyuk; Alexander Chuprina; Danai Mavridi; Christopher Lenz; Andreas C. Joerger; Benjamin D. Brown; Richard B. Heath; Wyatt W. Yue; Lucy K. Robbie; Tyler S. Beyett; Susanne Müller; Stefan Knapp; Dafydd R. Owen; Rachel Harding; Matthieu Schapira; Peter J. Brown; Vijayaratnam Santhakumar; Suzanne Ackloo; Cheryl H. Arrowsmith; Aled M. Edwards; Hui Peng; Levon Halabelian
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Targeting bacterial kinases as a strategy to counteract antibiotic resistance
err2025-12-04
err0
errOAAI
errVanessa Buffa; Julien Kowalewski; Guoman Qi; Robin Deutscher; Matijas Cica; Marion Richardoz; Mathilde Tomaszczyk; Andreas Krämer; Stefan Knapp; Catherine Dunyach-Remy; Katharina Rox; Jean-Francois Guichou; Corinne Lionne; Felix Hausch
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Overcoming Ligand Discovery Challenges: Developing Peptide-Based Tracers for SPSB2
err2025-12-01
err0
PREAI
errLenz, Christopher; Elson, Lewis; Dopfer, Johannes; Farges, Frederic; Kramer, Andreas; Lohr, Frank; Muller, Susanne; Gueret, Stephanie M.; Waldmann, Herbert; Dotsch, Volker; Saxena, Krishna; Knapp, Stefan
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Inhibitors supercharge kinase turnover through native proteolytic circuits
errNature
IF48.5
err2025-11-26
err0
errOAAI
errNatalie S. Scholes; Martino Bertoni; Arnau Comajuncosa-Creus; Katharina Kladnik; Xuefei Guo; Fabian Frommelt; Matthias Hinterndorfer; Hlib Razumkov; Polina Prokofeva; Martin P. Schwalm; Florian Born; Sandra Roehm; Hana Imrichova; Brianda L. Santini; Eleonora Barone; Caroline Schätz; Miquel Muñoz i Ordoño; Severin Lechner; Andrea Rukavina; Iciar Serrano; Miriam Abele; Anna Koren; Stefan Kubicek; Stefan Knapp; Nathanael S. Gray; Giulio Superti-Furga; Bernhard Kuster; Yigong Shi; Patrick Aloy; Georg E. Winter
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Nucleobase catalysts for the enzymatic activation of 8-oxoguanine DNA glycosylase 1
err2025-10-29
err0
errOAAI
errEmily C. Hank; Nicholas D'Arcy-Evans; Emma Rose Scaletti; Carlos Benítez-Buelga; Olov Wallner; Florian Ortis; Kaixin Zhou; Liuzhen Meng; Alicia del Prado; Patricia Calvo; Ingrid Almlöf; Elisee Wiita; Karen Nierlin; Sara Kosenina; Andreas Krämer; Alice Eddershaw; Mario Kehler; Maeve Long; AnnSofie Jemth; Holly Dawson; Josephine Stewart; Adam Dickey; Mikhael Elijah Astorga; Marek Varga; Evert Homan; Martin Scobie; Stefan Knapp; Leandro Sastre; Pål Stenmark; Miguel de Vega; Thomas Helleday; Maurice Michel
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Un-LOK-ing a New Approach for Conformational Selective Targeting of STK10 (LOK)
err2025-10-13
err0
errOAAI
errMartina Dettenhöfer; Laura Nadine Tandara; Jennifer Alisa Amrhein; Christian Georg Kurz; Martin Peter Schwalm; Theresa Elisabeth Mensing; Laurenz Maximilian Wahl; Andreas Krämer; Joshua Gerninghaus; Christopher Lenz; Lewis Elson; Benedict-Tilman Berger; Martin Schröder; Krishna Saxena; Susanne Müller; Stefan Knapp; Francesco Aleksy Greco; Thomas Hanke
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Click Chemistry Enables Rapid Development of Potent sEH PROTACs Using a Direct-to-Biology Approach
err2025-10-06
err0
errOAAI
errJulia Schoenfeld; Nick Liebisch; Steffen Brunst; Lilia Weizel; Stefan Knapp; Aimo Kannt; Ewgenij Proschak; Kerstin Hiesinger
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Inhibition of Nonsense-Mediated Decay in Small Cell Lung Cancer Promotes Tumor Cell Death and T Cell Cytotoxicity
err2025-08-29
err0
PREAI
errLucia A. Torres Fernández; Volker Boehm; Joel Kaufmann; Agnieszka Rumińska; Christian Müller; Nazanin Alavinejad; Beaunelle de Bruijn; Laura Lovric; Kian R. Weihrauch; Laura Kaiser; Marcel Schmiel; Lukas Maas; Filippo Beleggia; Graziella Bosco; Ariadne Androulidaki; Liu Fanyu; Silvia von Karstedt; Maria Cartolano; Johannes Brägelmann; Justinas Valiulis; Joshua D’Rozario; Nina Wobst; Katja Höpker; Felix John; Jürgen Wolf; Alexander Quaas; Stefan Knapp; Anna Schöllhorn; Jonas P. Becker; Angelika B. Riemer; Cecile Gouttefangeas; Hans-Georg Rammensee; Niels Gehring; Martin Peifer; Roman K. Thomas; Julie George
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Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.
err2025-08-22
err0
PREAI
errTheresa E. Mensing; Christian G. Kurz; Jennifer A. Amrhein; Theresa A.L. Ehret; Franziska Preuss; Sebastian Mathea; Marwah Karim; Do Hoang Nhu Tran; Zuzana Kadlecova; Tuomas A. Tolvanen; Daniel Martinez-Molina; Susanne Müller; Shirit Einav; Stefan Knapp; Thomas Hanke
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A twist in the tale: shifting from covalent targeting of a tyrosine in JAK3 to a lysine in MK2
err2025-08-22
err0
errOAAI
errLaura Hillebrand ‡; Guiqun Wang ‡; Alexander Rasch; Benedikt Masberg; Apirat Chaikuad; Thales Kronenberger; Ellen Günther; Michael Forster; Antti Poso; Michael Lämmerhofer; Stefan A. Laufer; Stefan Knapp; Matthias Gehringer
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Discovery of an Exquisitely Selective WDR5 Chemical Probe Accelerated by a High-Quality DEL-ML Hit
err2025-08-06
err0
errOAAI
errLasse Hoffmann; Christopher Lenz; Frederic Farges; Serah W. Kimani; Johannes Dopfer; Sabrina Keller; Martin P. Schwalm; Hanna Holzmann; Andreas Krämer; Aiping Dong; Fengling Lu; Irene Chau; Levon Halebelian; Matthias Gstaiger; Susanne Müller; Stefan Knapp; Vaclav Nemec
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Structural analysis of TRIM family PRYSPRY domains and its implications for E3-ligand design
err2025-07-30
err0
errOAAI
errRezart Zhubi; Apirat Chaikuad; Christian J. Muñoz Sosa; Andreas C. Joerger; Stefan Knapp
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