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Herman S. Overkleeft

leiden university

83H-index
925Paper Count
2.9WCitation Count
Published Papers 382
Publication Date
Fully protected pyrophosphates via phosphorobromidates for the synthesis of biopolymers
err2026-04-16
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errSven Wijngaarden; Femke L. A. M. van der Heijden; Koen J. Rijpkema; Bob van Puffelen; Nico J. Meeuwenoord; Danicia Ramcharan; Gijsbert A. van der Marel; Jeroen D. C. Codée; Herman S. Overkleeft; Dmitri V. Filippov
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A Practical and Flexible De Novo Synthesis of Deoxygenated Carbasugars and Their Cyclitol Epoxides
err2026-04-13
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errYevhenii Radchenko; Nick D. F. Puijmbroeck; Sanne M. Verduin; Jeroen D. C. Codée; Herman S. Overkleeft
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Carfilzomib-specific proteasome β5/β2 inhibition drives cardiotoxicity via remodeling of protein homeostasis and the renin-angiotensin-system
err2025-07-29
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errMax Mendez-Lopez; Andrej Besse; Christian Zuppinger; Christian Perez-Shibayama; Cristina Gil-Cruz; Bogdan I. Florea; Angelina De Martin; Mechthild Lütge; Deborah Beckerova; Simon Klimovic; Xiang Zhou; Leo Rasche; Jan Pribyl; Vladimir Rotrekl; Burkhard Ludewig; Herman S. Overkleeft; Lenka Besse; Christoph Driessen
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LIMP-2 deficiency-associated glycolipid abnormalities in mice
err2025-07-08
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errPaulo Gaspar; André R.A. Marques; Maria J. Ferraz; Markus Damme; Gertjan Kramer; Mina Mirzaian; Marion Gijbels; Roelof Ottenhoff; Cindy van Roomen; Herman S. Overkleeft; Michael Schwake; Saskia Heybrock; Maria Carmo Macário; Paul Saftig; Johannes M. Aerts
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Synthesis of a Set of Staphylococcus Aureus Capsular Polysaccharide Type 1 Oligosaccharides Carrying Taurine Esters
err2025-03-01
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PREAI
errOsterlid, Kitt Emilie; Cergano, Renata; Overkleeft, Herman S.; van der Marel, Gijsbert A.; Codee, Jeroen D. C.
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Activity-Based Protein Profiling Identifies an α-Amylase Family Protein Contributing to the Virulence of Methicillin-Resistant Staphylococcus aureus
err2025-02-06
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PREAI
errUddin, Md Jalal; Julin, Kjersti; Overkleeft, Herman S.; Johannessen, Mona; Lentz, Christian S.
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Precision Activity-Based α-Amylase Probes for Dissection and Annotation of Linear and Branched-Chain Starch-Degrading Enzymes
err2024-12-27
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PREAI
errPickles, Isabelle B.; Chen, Yurong; Moroz, Olga; Brown, Haley A.; de Boer, Casper; Armstrong, Zachary; Mcgregor, Nicholas G. S.; Artola, Marta; Codee, Jeroen D. C.; Koropatkin, Nicole M.; Overkleeft, Herman S.; Davies, Gideon J.
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Synthesis and Biological Evaluation of Deoxycyclophellitols as Human Retaining β-Glucosidase Inhibitors
err2024-11-03
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errRadchenko, Yevhenii; Su, Qin; Schroder, Sybrin S.; van Gijlswijk, Luke; Artola, Marta; Aerts, Johannes M. F. G.; Codee, Jeroen D. C.; Overkleeft, Herman S.
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substrates for GBA1 in the discovery of glycosylated sterols
err2024-11-01
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PREAI
errBannink, Stef; Bila, Kateryna O.; van Weperen, Joosje; Ligthart, Nina A. M.; Ferraz, Maria J.; Boot, Rolf G.; van der Vliet, Daan; Boer, Daphne. E. C.; Overkleeft, Herman S.; Artola, Marta; Aerts, Johannes M. F. G.
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From Mechanism-Based Retaining Glycosidase Inhibitors to Activity-Based Glycosidase Profiling
err2024-08-30
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errArtola, Marta; Aerts, Johannes M. F. G.; van der Marel, Gijsbert A.; Rovira, Carme; Codee, Jeroen D. C.; Davies, Gideon J.; Overkleeft, Herman S.
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A PIKfyve modulator combined with an integrated stress response inhibitor to treat lysosomal storage diseases
err2024-08-16
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errWilliam C. Hou; Lynée A. Massey; Derek Rhoades; Yin Wu; Wen Ren; Chiara Frank; Herman S. Overkleeft; Jeffrey W. Kelly
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Novel N,N-Dimethyl-idarubicin Analogues Are Effective Cytotoxic Agents for ABCB1-Overexpressing, Doxorubicin-Resistant Cells
err2024-08-01
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errvan Gelder, Merle A.; Li, Yufeng; Wander, Dennis P. A.; Berlin, Ilana; Overkleeft, Hermen S.; van der Zanden, Sabina Y.; Neefjes, Jacques J. C.
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Epi-Cyclophellitol Cyclosulfate, a Mechanism-Based Endoplasmic Reticulum α-Glucosidase II Inhibitor, Blocks Replication of SARS-CoV-2 and Other Coronaviruses
err2024-07-25
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errThaler, Melissa; Ofman, Tim P.; Kok, Ken; Heming, Jurriaan J. A.; Moran, Elisha; Pickles, Isabelle; Leijs, Anouk A.; van den Nieuwendijk, Adrianus M. C. H.; van den Berg, Richard J. B. H. N.; Ruijgrok, Gijs; Armstrong, Zachary; Salgado-Benvindo, Clarisse; Ninaber, Dennis K.; Snijder, Eric J.; van Boeckel, Constant A. A.; Artola, Marta; Davies, Gideon J.; Overkleeft, Herman S.; van Hemert, Martijn J.
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Parascedosporium putredinis NO1 tailors its secretome for different lignocellulosic substrates
err2024-07-02
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errScott, Conor J. R.; Mcgregor, Nicholas G. S.; Leadbeater, Daniel R.; Oates, Nicola C.; Hossbach, Janina; Abood, Amira; Setchfield, Alexander; Dowle, Adam; Overkleeft, Herman S.; Davies, Gideon J.; Bruce, Neil C.
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Detection of Sulfoquinovosidase Activity in Cell Lysates Using Activity-Based Probes
err2024-05-21
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errLi, Zirui; Pickles, Isabelle B.; Sharma, Mahima; Melling, Benjamin; Pallasdies, Luise; Codee, Jeroen D. C.; Williams, Spencer J.; Overkleeft, Herman S.; Davies, Gideon J.
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Conformational and Electronic Variations in 1,2-and 1,5a-Cyclophellitols and their Impact on Retaining α-Glucosidase Inhibition
err2024-04-24
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errOfman, Tim P.; Heming, Jurriaan J. A.; Nin-Hill, Alba; Kuellmer, Florian; Moran, Elisha; Bennett, Megan; Steneker, Roy; Klein, Anne-Mei; Ruijgrok, Gijs; Kok, Ken; Armstrong, Zach W. B.; Aerts, Johannes M. F. G.; van Der Marel, Gijsbert A.; Rovira, Carme; Davies, Gideon J.; Artola, Marta; Codee, Jeroen D. C.; Overkleeft, Herman S.
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Synthesis and application of bacterial exopolysaccharides
err2024-02-01
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errRuijgrok, Gijs; Wu, Dung-Yeh; Overkleeft, Herman S.; Codee, Jeroen D. C.
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Selective labelling of GBA2 in cells with fluorescent β-d-arabinofuranosyl cyclitol aziridines
err2024-01-01
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errSu, Qin; Louwerse, Max; Lammers, Rob F.; Maurits, Elmer; Janssen, Max; Boot, Rolf G.; Borlandelli, Valentina; Offen, Wendy A.; Linzel, Daniel; Schroder, Sybrin P.; Davies, Gideon J.; Overkleeft, Herman S.; Artola, Marta; Aerts, Johannes M. F. G.
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Structure-guided design of C3-branched swainsonine as potent and selective human Golgi α-mannosidase (GMII) inhibitor
err2024-01-01
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PREAI
errKoemans, Tony; Bennett, Megan; Ferraz, Maria J.; Armstrong, Zachary; Artola, Marta; Aerts, Johannes M. F. G.; Codee, Jeroen D. C.; Overkleeft, Herman S.; Davies, Gideon J.
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Molecular Basis for Inhibition of Heparanases and β-Glucuronidases by Siastatin B
err2023-12-20
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errChen, Yurong; van den Nieuwendijk, Adrianus M. C. H.; Wu, Liang; Moran, Elisha; Skoulikopoulou, Foteini; van Riet, Vera; Overkleeft, Hermen S.; Davies, Gideon J.; Armstrong, Zachary
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