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Structural insights into the interaction of three Y- shaped ligands with PI3Kα Zhou, Qingtong; Liu, Xiao; Neri, Dario; Li, Wenxin; Favalli, Nicholas; Bassi, Gabriele; Yang, Su; Yang, Dehua; Vogt, Peter K.; Wang, Ming-Wei Share Save
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Nanobodies and chemical cross-links advance the structural and functional analysis of PI3Kα Hart, Jonathan R.; Liu, Xiao; Pan, Chen; Liang, Anyi; Ueno, Lynn; Xu, Yingna; Quezada, Alexandra; Zou, Xinyu; Yang, Su; Zhou, Qingtong; Schoonooghe, Steve; Hassanzadeh-Ghassabeh, Gholamreza; Xia, Tian; Shui, Wenqing; Yang, Dehua; Vogt, Peter K.; Wang, Ming-Wei Share Save
Cryo-EM structures of PI3Kα reveal conformational changes during inhibition and activation Liu, Xiao; Yang, Su; Hart, Jonathan R.; Xu, Yingna; Zou, Xinyu; Zhang, Huibing; Zhou, Qingtong; Xia, Tian; Zhang, Yan; Yang, Dehua; Wang, Ming-Wei; Vogt, Peter K. Share Save
Synthetic fluorescent MYC probe: Inhibitor binding site elucidation and development of a high-throughput screening assay Shirey, Ryan J.; Hart, Jonathan R.; Sridharan, BanuPriya; Novick, Scott J.; Turner, Lewis D.; Zhou, Bin; Nielsen, Alexander L.; Eubanks, Lisa M.; Ueno, Lynn; Hixon, Mark S.; Lairson, Luke L.; Spicer, Timothy P.; Scampavia, Louis D.; Griffin, Patrick R.; Vogt, Peter K.; Janda, Kim D. Share Save
A Single-Stranded DNA-Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks Bassi, Gabriele; Favalli, Nicholas; Vuk, Miriam; Catalano, Marco; Martinelli, Adriano; Trenner, Anika; Porro, Antonio; Yang, Su; Tham, Chuin Lean; Moroglu, Mustafa; Yue, Wyatt W.; Conway, Stuart J.; Vogt, Peter K.; Sartori, Alessandro A.; Scheuermann, Joerg; Neri, Dario Share Save
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Synthetic molecules for disruption of the MYC protein-protein interface Jacob, Nicholas T.; Miranda, Pedro O.; Shirey, Ryan J.; Gautam, Ritika; Zhou, Bin; Izquierdo, M. Elena de Orbe; Hixon, Mark S.; Hart, Jonathan R.; Ueno, Lynn; Vogt, Peter K.; Janda, Kim D. Share Save
tsRNA signatures in cancer Balatti, Veronica; Nigita, Giovanni; Veneziano, Dario; Drusco, Alessandra; Stein, Gary S.; Messier, Terri L.; Farina, Nicholas H.; Lian, Jane B.; Tomasello, Luisa; Liu, Chang-Gong; Palamarchuk, Alexey; Hart, Jonathan R.; Bell, Catherine; Carosi, Mariantonia; Pescarmona, Edoardo; Perracchio, Letizia; Diodoro, Maria; Russo, Andrea; Antenucci, Anna; Visca, Paolo; Ciardi, Antonio; Harris, Curtis C.; Vogt, Peter K.; Pekarsky, Yuri; Croce, Carlo M. Share Save
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