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Identification and Optimization of a Novel HIV-1 Integrase Inhibitor Adu-Ampratwum, Daniel; Pan, Yuhan; Koneru, Pratibha C.; Antwi, Janet; Hoyte, Ashley C.; Kessl, Jacques; Griffin, Patrick R.; Kvaratskhelia, Mamuka; Fuchs, James R.; Larue, Ross C. Share Save
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HIV-1 Integrase-Targeted Short Peptides Derived from a Viral Protein R Sequence Zhao, Xue Zhi; Metifiot, Mathieu; Kiselev, Evgeny; Kessl, Jacques J.; Maddali, Kasthuraiah; Marchand, Christophe; Kvaratskhelia, Mamuka; Pommier, Yves; Burke, Terrence R., Jr. Share Save
A New Class of Allosteric HIV-1 Integrase Inhibitors Identified by Crystallographic Fragment Screening of the Catalytic Core Domain Patel, Disha; Antwi, Janet; Koneru, Pratibha C.; Serrao, Erik; Forli, Stefano; Kessl, Jacques J.; Feng, Lei; Deng, Nanjie; Levy, Ronald M.; Fuchs, James R.; Olson, Arthur J.; Engelman, Alan N.; Bauman, Joseph D.; Kvaratskhelia, Mamuka; Arnold, Eddy Share Save
The Competitive Interplay between Allosteric HIV-1 Integrase Inhibitor BI/D and LEDGF/p75 during the Early Stage of HIV-1 Replication Adversely Affects Inhibitor Potency Feng, Lei; Dharmarajan, Venkatasubramanian; Serrao, Erik; Hoyte, Ashley; Larue, Ross C.; Slaughter, Alison; Sharma, Amit; Plumb, Matthew R.; Kessl, Jacques J.; Fuchs, James R.; Bushman, Frederic D.; Engelman, Alan N.; Griffin, Patrick R.; Kvaratskhelia, Mamuka Share Save
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A New Class of Multimerization Selective Inhibitors of HIV-1 Integrase Sharma, Amit; Slaughter, Alison; Jena, Nivedita; Feng, Lei; Kessl, Jacques J.; Fadel, Hind J.; Malani, Nirav; Male, Frances; Wu, Li; Poeschla, Eric; Bushman, Frederic D.; Fuchs, James R.; Kvaratskhelia, Mamuka Share Save
BET proteins promote efficient murine leukemia virus integration at transcription start sites Sharma, Amit; Larue, Ross C.; Plumb, Matthew R.; Malani, Nirav; Male, Frances; Slaughter, Alison; Kessl, Jacques J.; Shkriabai, Nikolozi; Coward, Elizabeth; Aiyer, Sriram S.; Green, Patrick L.; Wu, Li; Roth, Monica J.; Bushman, Frederic D.; Kvaratskhelia, Mamuka Share Save
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The A128T Resistance Mutation Reveals Aberrant Protein Multimerization as the Primary Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors Feng, Lei; Sharma, Amit; Slaughter, Alison; Jena, Nivedita; Koh, Yasuhiro; Shkriabai, Nikolozi; Larue, Ross C.; Patel, Pratiq A.; Mitsuya, Hiroaki; Kessl, Jacques J.; Engelman, Alan; Fuchs, James R.; Kvaratskhelia, Mamuka Share Save
Allosteric integrase inhibitor potency is determined through the inhibition of HIV-1 particle maturation Jurado, Kellie A.; Wang, Hao; Slaughter, Alison; Feng, Lei; Kessl, Jacques J.; Koh, Yasuhiro; Wang, Weifeng; Ballandras-Colas, Allison; Patel, Pratiq A.; Fuchs, James R.; Kvaratskhelia, Mamuka; Engelman, Alan Share Save
Interaction of the HIV-1 Intasome with Transportin 3 Protein (TNPO3 or TRN-SR2) Larue, Ross; Gupta, Kushol; Wuensch, Christiane; Shkriabai, Nikolozi; Kessl, Jacques J.; Danhart, Eric; Feng, Lei; Taltynov, Oliver; Christ, Frauke; Van Duyne, Gregory D.; Debyser, Zeger; Foster, Mark P.; Kvaratskhelia, Mamuka Share Save
Multimode, Cooperative Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors Kessl, Jacques J.; Jena, Nivedita; Koh, Yasuhiro; Taskent-Sezgin, Humeyra; Slaughter, Alison; Feng, Lei; de Silva, Suresh; Wu, Li; Le Grice, Stuart F. J.; Engelman, Alan; Fuchs, James R.; Kvaratskhelia, Mamuka Share Save
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