arrow
Back
O

Olivier Boutaud

vanderbilt university

38H-index
168Paper Count
4.2KCitation Count
Published Papers 81
Publication Date
Drug Repurposing: Conversion of the Peripherally Restricted HIV Protease Inhibitor Amprenavir to Potent; Selective; and CNS-Penetrant Agonists for the Cannabinoid Receptor 2
err2026-02-05
err0
errOAAI
errDaniel H. Haymer; Renn A. Duncan; Alice L. Rodriguez; Allie Han; Richard J. Lindsay; N. Kithmini Wijesiri; Analisa Thompson Gray; Srinivasan Krishnan; Aidong Qi; Benjamin P. Brown; Olivier Boutaud; Darren W. Engers; Carrie K. Jones; Colleen M. Niswender; Craig W. Lindsley; Aaron M. Bender
errShare
errSave
Discovery of VU6025733 (AG06827): A Highly Selective; Orally Bioavailable; and Structurally Distinct M4 Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM) with Robust In Vivo Efficacy
err2026-01-25
err0
errOAAI
errAlison R. Gregro; Charlotte Park; Madeline F. Long; Logan A. Baker; Katrina A. Bollinger; Anna E. Ringuette; Li Peng; Vincent B. Luscombe; Natasha B. Billard; Alice L. Rodriguez; Colleen M. Niswender; Weimin Peng; Jonathan W. Dickerson; Jerri M. Rook; Jordan O’Neill; Sichen Chang; Harrie C. M. Boonen; Thomas Jensen; Morten S. Thomsen; Thomas M. Bridges; Olivier Boutaud; P. Jeffrey Conn; Darren W. Engers; Craig W. Lindsley; Kayla J. Temple
errShare
errSave
Discovery of 7-(Pyridin-3-yl)thieno[3; 2-b]pyridine-5-carboxamides as Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5
err2026-01-25
err0
errOAAI
errScott H. Henderson; Anna E. Ringuette; David L. Whomble; Rory A. Capstick; Alexa E. Richardson; Mallory A. Maurer; Natasha B. Billard; Xia Lei; Joshua C. Wilkinson; Sri H. Kethanapalli; Hyekyung P. Cho; Alice L. Rodriguez; Colleen M. Niswender; Weimin Peng; Jerri M. Rook; Sichen Chang; Anna L. Blobaum; Olivier Boutaud; Andrew S. Felts; P. Jeffrey Conn; Craig W. Lindsley; Kayla J. Temple
errShare
errSave
Discovery of VU6083859, a TAOK1 Selective Inhibitor, and VU6080195, a pan-TAOK Activator
err2026-01-01
err0
errOAAI
errSchultz, Daniel C.; Parr, Lauren C.; Sweet, Hunter; Lamb, Sean; Engers, Julie L.; Napier, Nathaniel C.; McKinnie, Hallie G.; Whomble, David; Kramlinger, Valerie; Boutaud, Olivier; Lindsley, Craig W.
errShare
errSave
Discovery of VU6052254: A Novel; Potent M1 Positive Allosteric Modulator
err2025-11-26
err0
errOAAI
errJulie L. Engers; Joseph D. Bungard; Christopher C. Presley; Irene Zagol-Ikapitte; Katherine J. Watson; Sichen Chang; Colin O’Carroll; P. Markus Dey; Ethan S. Burstein; Jonathan W. Dickerson; Analisa Thompson Gray; Michael Bubser; Jerri M. Rook; Hyekyung P. Cho; Valerie M. Kramlinger; Olivier Boutaud; Carrie K. Jones; P. Jeffrey Conn; Darren W. Engers; Craig W. Lindsley
errShare
errSave
Optimization of Selective and CNS Penetrant Alkyne-Based TREK Inhibitors: The Discovery and Characterization of ONO-9517601 (VU6022856) and ONO-7927846 (VU6024391)
err2025-10-01
err0
PREAI
errTanaka, Motoyuki; Sekioka, Yoko; Hashimoto, Gakuji; Mori, Takahiro; Shono, Tomoyuki; Isaji, Yuuki; Hisaichi, Katsuya; Childress, Elizabeth S.; Bollinger, Sean; Schmitt, Joza A.; Chopko, Trevor C.; Garrison, Aaron T.; Perry, Charles K.; Chronister, Keagan; Kramer, Meghan; Chang, Sichen; Watson, Katherine J.; Dickerson, Jonathan W.; Bubser, Michael; Rook, Jerri M.; Jones, Carrie K.; Boutaud, Olivier; Bridges, Thomas M.; Denton, Jerod S.; Engers, Darren W.; Kurata, Haruto; Lindsley, Craig W.
errShare
errSave
Protective role of epithelial deoxyhypusine synthase in colorectal carcinogenesis caused by deletion of the adenomatous polyposis coli gene
err2025-08-24
err0
errOAAI
errAlain P. Gobert; Caroline V. Hawkins; Lydia A. Snyder; Kamery J. Williams; Daniel P. Barry; Margaret M. Allaman; Mohammad Asim; Kara M. McNamara; Shane M. Carey; Alberto G. Delgado; Regina N. Tyree; Kristie L. Rose; Yu Wang; Shilin Zhao; Olivier Boutaud; Irène Zagol-Ikapitte; M. Blanca Piazuelo; M. Kay Washington; Lori A. Coburn; Keith T. Wilson
errShare
errSave
Total Synthesis and Pharmacological Evaluation of Phochrodines A-C
err2025-04-01
err0
errOAAI
errBouchard, Jacob L.; Chang, Sichen; Krishnan, Srinivasan; Presley, Christopher C.; Boutaud, Olivier; Schley, Nathan D.; Engers, Darren W.; Engers, Julie L.; Lindsley, Craig W.; Bender, Aaron M.
errShare
errSave
Discovery of Thieno[3,2-b]pyridine-5-carboxamide and 2,3-Difluorobenzamide Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5
err2025-04-01
err0
errOAAI
errCrocker, Katherine E.; Henderson, Scott H.; Capstick, Rory A.; Whomble, David L.; Bender, Aaron M.; Felts, Andrew S.; Han, Changho; Engers, Julie L.; Billard, Natasha B.; Maurer, Mallory A.; Cho, Hyekyung P.; Rodriguez, Alice L.; Niswender, Colleen M.; O'Neill, Jordan; Watson, Katherine J.; Chang, Sichen; Blobaum, Anna L.; Boutaud, Olivier; Peng, Weimin; Rook, Jerri M.; Conn, P. Jeffrey; Lindsley, Craig W.; Temple, Kayla J.
errShare
errSave
Application of Deuterium in an M1 Positive Allosteric Modulator Back-Up Program: The Discovery of VU6045422
err2025-03-25
err0
errOAAI
errEngers, JL; Li, JM; Han, CH; Long, MF; Gregro, AR; Presley, CC; Dickerson, JW; Peng, WM; Cho, HP; Rodriguez, AL; Xiang, ZX; Boutaud, O; O'Carroll, C; Dey, PM; Burstein, ES; Niswender, CM; Rook, JM; Conn, PJ; Engers, DW; Lindsley, CW
errShare
errSave
Discovery of ONO-2920632 (VU6011887): A Highly Selective and CNS Penetrant TREK-2 (TWIK-Related K+ Channel 2) Preferring Activator In Vivo Tool Compound
err2025-02-21
err1
errOAAI
errYashiro, K; Iwaki, Y; Urata, H; Kokubo, M; Mori, T; Sekioka, Y; Isami, K; Kato, J; Wieting, J; Mcgowan, KM; Bridges, TM; Boutaud, O; Engers, DW; Denton, JS; Kurata, H; Lindsley, CW
errShare
errSave
Further Optimization of the mGlu1 PAM VU6024578/BI02982816: Discovery and Characterization of VU6033685
err2025-02-05
err0
errOAAI
errReed, Carson W.; Kalbfleisch, Jacob F.; Turkett, Jeremy A.; Trombley, Trevor A.; Spearing, Paul K.; Haymer, Daniel H.; Quitalig, Marc; Dickerson, Jonathan W.; Foster, Daniel J.; Blobaum, Annie L.; Boutaud, Olivier; Cho, Hyekyung P.; Niswender, Colleen M.; Rook, Jerri M.; Priepke, Henning; Sommer, Heiko; Scheuerer, Stefan; Ursu, Daniel; Conn, P. Jeffrey; Melancon, Bruce J.; Lindsley, Craig W.
errShare
errSave
Chronic Gastroesophageal Reflux Dysregulates Proteostasis in Esophageal Epithelial Cells
err2025-01-01
err1
PREAI
errPaulrasu, Kodisundaram; Gokulan, Ravindran Caspa; El-Rifai, Wael; Chen, Zhibin; Que, Jianwen; Wang, Timothy C.; Boutaud, Olivier G.; Briegel, Karoline; Dikalov, Sergey I.; Garcia-Buitrago, Monica T.; Zaika, Alexander I.
errShare
errSave
Discovery of VU6024578/BI02982816: An mGlu1 Positive Allosteric Modulator with Efficacy in Preclinical Antipsychotic and Cognition Models
err2024-12-12
err0
errOAAI
errReed, Carson W.; Kalbfleisch, Jacob F.; Turkett, Jeremy A.; Trombley, Trevor A.; Nastase, Anthony F.; Spearing, Paul K.; Haymer, Daniel H.; Sarwar, Mohammad Moshin; Quitalig, Marc; Dickerson, Jonathan W.; Blobaum, Annie L.; Boutaud, Olivier; Voehringer, Patrizia; Schuelert, Niklas; Cho, Hyekyung P.; Niswender, Colleen M.; Rook, Jerri M.; Priepke, Henning; Ursu, Daniel; Conn, P. Jeffrey; Melancon, Bruce J.; Lindsley, Craig W.
errShare
errSave
Discovery of VU0467319: an M1 Positive Allosteric Modulator Candidate That Advanced into Clinical Trials
err2024-12-11
err0
errOAAI
errPoslunsey, Michael S.; Wood, Michael R.; Han, Changho; Stauffer, Shaun R.; Panarese, Joseph D.; Melancon, Bruce J.; Engers, Julie L.; Dickerson, Jonathan W.; Peng, Weimin; Noetzel, Meredith J.; Cho, Hyekyung P.; Rodriguez, Alice L.; Hopkins, Corey R.; Morrison, Ryan; Crouch, Rachel D.; Bridges, Thomas M.; Blobaum, Anna L.; Boutaud, Olivier; Daniels, J. Scott; Kates, Michael J.; Castelhano, Arlindo; Rook, Jerri M.; Niswender, Colleen M.; Jones, Carrie K.; Conn, P. Jeffrey; Lindsley, Craig W.
errShare
errSave
Discovery of 4-(5-Membered)Heteroarylether-6-methylpicolinamide Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5
err2024-11-18
err0
errOAAI
errChildress, Elizabeth S.; Capstick, Rory A.; Crocker, Katherine E.; Ledyard, Miranda L.; Bender, Aaron M.; Maurer, Mallory A.; Billard, Natasha B.; Cho, Hyekyung P.; Rodriguez, Alice L.; Niswender, Colleen M.; Peng, Weimin; Rook, Jerri M.; Chang, Sichen; Blobaum, Anna L.; Boutaud, Olivier; Thompson Gray, Analisa; Jones, Carrie K.; Conn, P. Jeffrey; Felts, Andrew S.; Lindsley, Craig W.; Temple, Kayla J.
errShare
errSave
Platelet Activation in Patients with Peripheral Artery Disease From 43 Sites: Assessment of Samples Transported by Overnight Mail
err2024-11-12
err0
PREAI
errStubblefield, William; Sullivan, Alexander; Amin, Taneem; Boutaud, Olivier; Cahill, Katherine; Flaherty, David; Matlock, Brittany; Berger, Jeffrey; Beckman, Joshua
errShare
errSave
Discovery of VU6016235: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M4 Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)
err2024-09-24
err0
errOAAI
errEngers, Julie L.; Baker, Logan A.; Chang, Sichen; Luscombe, Vincent B.; Rodriguez, Alice L.; Niswender, Colleen M.; Cho, Hyekyung P.; Bubser, Michael; Gray, Analisa Thompson; Jones, Carrie K.; Peng, Weimin; Rook, Jerri M.; Bridges, Thomas M.; Boutaud, Olivier; Conn, P. Jeffrey; Engers, Darren W.; Lindsley, Craig W.; Temple, Kayla J.
errShare
errSave
Discovery of VU6007496: Challenges in the Development of an M1 Positive Allosteric Modulator Backup Candidate
err2024-08-28
err2
errOAAI
errEngers, Julie L.; Bollinger, Katrina A.; Capstick, Rory A.; Long, Madeline F.; Bender, Aaron M.; Dickerson, Jonathan W.; Peng, Weimin; Presley, Christopher C.; Cho, Hyekyung P.; Rodriguez, Alice L.; Niswender, Colleen M.; Moran, Sean P.; Xiang, Zixiu; Blobaum, Anna L.; Boutaud, Olivier; Rook, Jerri M.; Engers, Darren W.; Conn, P. Jeffrey; Lindsley, Craig W.
errShare
errSave
Development of VU6036864: A Triazolopyridine-Based High-Quality Antagonist Tool Compound of the M5 Muscarinic Acetylcholine Receptor
err2024-08-06
err0
errOAAI
errLi, Jinming; Orsi, Douglas L.; Engers, Julie L.; Long, Madeline F.; Capstick, Rory A.; Maurer, Mallory A.; Presley, Christopher C.; Vinson, Paige N.; Rodriguez, Alice L.; Han, Allie; Cho, Hyekyung P.; Chang, Sichen; Jackson, Megan; Bubser, Michael; Blobaum, Anna L.; Boutaud, Olivier; Nader, Michael A.; Niswender, Colleen M.; Conn, P. Jeffrey; Jones, Carrie K.; Lindsley, Craig W.; Han, Changho
errShare
errSave