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陆涛 (Tao Lu)

capital medical university

35H-index
226Paper Count
3.9KCitation Count
Published Papers 98
Publication Date
E3 Ligase SMURF2 Promotes Adipogenesis and Improves Obesity Complications by Suppressing TGF-β Signaling
err2026-05-18
err0
errOAAI
errXueqin Wu; Muchen Wu; Shiyu Du; Jiaxin Liu; Ruiping Wang; Yuhan Sun; Zhi Zheng; Junru Yang; Xiaowei Jia; Lulu Wang; Tao Lu; Chun Yang; Yan Gao; Dongliang Fang
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Design and Synthesis of Novel N-(1H-pyrazol-3-yl)pyrimidin-4-amine Aurora/HDAC Dual Inhibitors for Colorectal Cancer Treatment
err2025-11-10
err0
PREAI
errHao Cui; Xu Huang; Rui Li; Meng Zong; Shilong Sun; Hongmei Li; Yadong Chen; Tao Lu; Yong Zhu
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Decoding Secondary Motor Cortex Neuronal Activity During Cocaine Self-Administration: Insights From Longitudinal In Vivo Calcium Imaging
err2025-05-09
err0
errOAAI
errYingying Chen; Haoying Fu; Amith Korada; Michal A. Lange; Chandrashekar Rayanki; Tao Lu; Dongbing Lai; Shiaofen Fang; Changyong Guo; Yao-Ying Ma
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Design and synthesis of 1H-benzo[d]imidazole selective HDAC6 inhibitors with potential therapy for multiple myeloma
err2023-12-01
err3
PREAI
errLiu, Linfu; Zhang, Liyuan; Chen, Xuxi; Yang, Kang; Cui, Hao; Qian, Rui; Zhao, Shanshan; Wang, Liqun; Su, Xiaolan; Zhao, Manyu; Wang, Mengzhu; Hu, Zan; Lu, Tao; Zhu, Yong; Zhou, Qing-Qing; Yao, Yuqin
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Hydrophobic tag-based protein degradation: Development, opportunity and challenge
err2023-11-01
err23
PREAI
errHe, Qindi; Zhao, Xiaofei; Wu, Donglin; Jia, Siming; Liu, Canlin; Cheng, Zitian; Huang, Fei; Chen, Yadong; Lu, Tao; Lu, Shuai
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Rational discovery of dual FLT3/HDAC inhibitors as a potential AML therapy
err2023-11-01
err10
PREAI
errWang, Zhijie; Wu, Donglin; Zhao, Xiaofei; Liu, Canlin; Jia, Siming; He, Qindi; Huang, Fei; Cheng, Zitian; Lu, Tao; Chen, Yadong; Chen, Yun; Yang, Pei; Lu, Shuai
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Rational design of 4-((6-phenoxypyrimidin-4-yl) amino)-N-(4-(piperazin-1-yl)phenyl)-1H-pyrazole-3-carboxamide (LT-540-717) as orally bioavailable FLT3 inhibitor
err2023-08-01
err2
PREAI
errZhi, Yanle; Li, Hongmei; Yang, Pei; Jin, Qiaomei; Yao, Chao; Li, Baoquan; Ling, Jun; Guo, Hao; Li, Tonghui; Jin, Jianlin; Wang, Yue; Chen, Yadong; Lu, Tao; Lu, Shuai
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Carboxymethylated Alginate-Resiquimod Micelles Reverse the Immunosuppressive Tumor Microenvironment and Synergistically Enhance the Chemotherapy and Immunotherapy for Gastric Cancer
err2023-07-21
err9
PREAI
errChen, Jiamin; Liu, Xingxing; Zhao, Shujing; Chen, Hongyican; Lu, Tao; Wang, Jinfeng; Han, Jiahui; Wu, Wangran; Shen, Xian; Li, Chao
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Discovery of Thieno[3,2-d]pyrimidine derivatives as potent and selective inhibitors of ataxia telangiectasia mutated and Rad3 related (ATR) kinase
err2023-07-01
err6
PREAI
errDuan, Yunxin; Cheng, Haodong; Zhuang, Lili; Xia, Jiawei; Xu, Yerong; Zhang, Ruyue; Sun, Rui; Lu, Tao; Chen, Yadong
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Burden of vitiligo on Chinese patients: An online survey
err2023-02-21
err0
errOAAI
errAmer, Abdulrahman; Wu, Yan; Li, Chunying; Du, Juan; Jia, Hong; Li, Shanshan; Tu, Caixia; Li, Qiang; Liu, Hongxia; Zhang, Junling; Lu, Tao; Liu, Jinsong; Mei, Aihua; Liu, Han; Tian, Fei; Lu, Chong; Li, Zihan; Cao, Lixin; Gao, Xinghua
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Recent advances in targeted protein degraders as potential therapeutic agents
err2023-02-15
err18
errOAAI
errYang, Na; Kong, Bo; Zhu, Zhaohong; Huang, Fei; Zhang, Liliang; Lu, Tao; Chen, Yadong; Zhang, Yanmin; Jiang, Yulei
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Atroposelective Amination of Indoles via Chiral Center Induced Chiral Axis Formation
err2022-12-17
err3
errOAAI
errWang, Yong; Yan, Jingxue; Jiang, Yiqing; Wei, Zexuan; Tu, Zhenlin; Dong, Chao; Lu, Tao; Chen, Yadong; Feng, Jie
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Multimodal multi-task deep neural network framework for kinase-target prediction
err2022-11-11
err2
PREAI
errHua, Yi; Luo, Lin; Qiu, Haodi; Huang, Dingfang; Zhao, Yang; Liu, Haichun; Lu, Tao; Chen, Yadong; Zhang, Yanmin; Jiang, Yulei
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Identification and structural analysis of a selective tropomyosin receptor kinase C (TRKC) inhibitor
err2022-11-01
err4
PREAI
errWang, Zhijie; Ren, Jiwei; Jia, Kun; Zhao, Yuming; Liang, Li; Cheng, Zitian; Huang, Fei; Zhao, Xiaofei; Cheng, Jie; Song, Shiyu; Sheng, Tiancheng; Wan, Weiqi; Shu, Qingqing; Wu, Donglin; Zhang, Junhao; Lu, Tao; Chen, Yadong; Ran, Ting; Lu, Shuai
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Design and synthesis of highly TRAIL expression HDAC inhibitors based on ONC201 to promote apoptosis of colorectal cancer (vol 238, 114484, 2022)
err2022-10-01
err0
PREAI
errCui, Hao; Hu, Zan; Yang, Kang; Huang, Jingkun; Wu, Yichao; Chen, Quanwei; Wei, Ran; Wang, Penfeng; Wang, Hui; Li, Hongmei; Chen, Yadong; Lu, Tao; Yao, Yuqin; Zhu, Yong
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Design and synthesis of highly TRAIL expression HDAC inhibitors based on ONC201 to promote apoptosis of colorectal cancer
err2022-08-01
err9
PREAI
errCui, Hao; Hu, Zan; Yang, Kang; Huang, Jingkun; Wu, Yichao; Chen, Quanwei; Wei, Ran; Wang, Penfeng; Wang, Hui; Li, Hongmei; Chen, Yadong; Lu, Tao; Yao, Yuqin; Zhu, Yong
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Novel GSK-3 kinase inhibitor Pym-5 induces GSK-3β rather than GSK-3α-dependent melanogenesis in murine melanoma cells
err2022-06-01
err2
PREAI
errJia, Qi; Tao, Li; Zhou, Yinyin; Song, Li; Wei, Zhonghong; Lu, Tao; Woodgett, James R.; Lu, Yin
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Research Directions

新药分子设计与合成研究计算机辅助药物设计有机合成化学药物生物统计与计算药学