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SaveDesign and synthesis of 1H-benzo[d]imidazole selective HDAC6 inhibitors with potential therapy for multiple myeloma
Liu, Linfu; Zhang, Liyuan; Chen, Xuxi; Yang, Kang; Cui, Hao; Qian, Rui; Zhao, Shanshan; Wang, Liqun; Su, Xiaolan; Zhao, Manyu; Wang, Mengzhu; Hu, Zan; Lu, Tao; Zhu, Yong; Zhou, Qing-Qing; Yao, Yuqin
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SaveHydrophobic tag-based protein degradation: Development, opportunity and challenge
He, Qindi; Zhao, Xiaofei; Wu, Donglin; Jia, Siming; Liu, Canlin; Cheng, Zitian; Huang, Fei; Chen, Yadong; Lu, Tao; Lu, Shuai
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SaveRational discovery of dual FLT3/HDAC inhibitors as a potential AML therapy
Wang, Zhijie; Wu, Donglin; Zhao, Xiaofei; Liu, Canlin; Jia, Siming; He, Qindi; Huang, Fei; Cheng, Zitian; Lu, Tao; Chen, Yadong; Chen, Yun; Yang, Pei; Lu, Shuai
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SaveRational design of 4-((6-phenoxypyrimidin-4-yl) amino)-N-(4-(piperazin-1-yl)phenyl)-1H-pyrazole-3-carboxamide (LT-540-717) as orally bioavailable FLT3 inhibitor
Zhi, Yanle; Li, Hongmei; Yang, Pei; Jin, Qiaomei; Yao, Chao; Li, Baoquan; Ling, Jun; Guo, Hao; Li, Tonghui; Jin, Jianlin; Wang, Yue; Chen, Yadong; Lu, Tao; Lu, Shuai
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SaveCarboxymethylated Alginate-Resiquimod Micelles Reverse the Immunosuppressive Tumor Microenvironment and Synergistically Enhance the Chemotherapy and Immunotherapy for Gastric Cancer
Chen, Jiamin; Liu, Xingxing; Zhao, Shujing; Chen, Hongyican; Lu, Tao; Wang, Jinfeng; Han, Jiahui; Wu, Wangran; Shen, Xian; Li, Chao
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SaveDiscovery of Thieno[3,2-d]pyrimidine derivatives as potent and selective inhibitors of ataxia telangiectasia mutated and Rad3 related (ATR) kinase
Duan, Yunxin; Cheng, Haodong; Zhuang, Lili; Xia, Jiawei; Xu, Yerong; Zhang, Ruyue; Sun, Rui; Lu, Tao; Chen, Yadong
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SaveBurden of vitiligo on Chinese patients: An online survey
Amer, Abdulrahman; Wu, Yan; Li, Chunying; Du, Juan; Jia, Hong; Li, Shanshan; Tu, Caixia; Li, Qiang; Liu, Hongxia; Zhang, Junling; Lu, Tao; Liu, Jinsong; Mei, Aihua; Liu, Han; Tian, Fei; Lu, Chong; Li, Zihan; Cao, Lixin; Gao, Xinghua
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SaveMultimodal multi-task deep neural network framework for kinase-target prediction
Hua, Yi; Luo, Lin; Qiu, Haodi; Huang, Dingfang; Zhao, Yang; Liu, Haichun; Lu, Tao; Chen, Yadong; Zhang, Yanmin; Jiang, Yulei
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SaveIdentification and structural analysis of a selective tropomyosin receptor kinase C (TRKC) inhibitor
Wang, Zhijie; Ren, Jiwei; Jia, Kun; Zhao, Yuming; Liang, Li; Cheng, Zitian; Huang, Fei; Zhao, Xiaofei; Cheng, Jie; Song, Shiyu; Sheng, Tiancheng; Wan, Weiqi; Shu, Qingqing; Wu, Donglin; Zhang, Junhao; Lu, Tao; Chen, Yadong; Ran, Ting; Lu, Shuai
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SaveDesign and synthesis of highly TRAIL expression HDAC inhibitors based on ONC201 to promote apoptosis of colorectal cancer (vol 238, 114484, 2022)
Cui, Hao; Hu, Zan; Yang, Kang; Huang, Jingkun; Wu, Yichao; Chen, Quanwei; Wei, Ran; Wang, Penfeng; Wang, Hui; Li, Hongmei; Chen, Yadong; Lu, Tao; Yao, Yuqin; Zhu, Yong
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SaveDesign and synthesis of highly TRAIL expression HDAC inhibitors based on ONC201 to promote apoptosis of colorectal cancer
Cui, Hao; Hu, Zan; Yang, Kang; Huang, Jingkun; Wu, Yichao; Chen, Quanwei; Wei, Ran; Wang, Penfeng; Wang, Hui; Li, Hongmei; Chen, Yadong; Lu, Tao; Yao, Yuqin; Zhu, Yong
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