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Lead optimization and mode-of-action elucidation for novel antifibrotics Merchant, Kevin; Porras-Gonzalez, Diana; Wei, Xin; Kratochvi, Michal; Shitov, Vladimir; Ma, Huilong; Lang, Niklas; Agami, Ahmed; Woegrath, Melanie; Kneidinger, Nikolaus; Yildrim, Ali Oender; Schiller, Herbert B.; Plettenburg, Oliver; Gerckens, Michael; Burgstaller, Gerald Share Save
Patterned thin film enzyme electrodes via spincoating and glutaraldehyde vapor crosslinking: towards scalable fabrication of integrated sensor-on-CMOS devices Adalian, Dvin; Madero, Xiomi; Chen, Samson; Jilani, Musab; Smith, Richard D.; Li, Songtai; Ahlbrecht, Christin; Cardenas, Juan; Agarwal, Abhinav; Emami, Azita; Plettenburg, Oliver; Petillo, Peter A.; Scherer, Axel Share Save
Development of novel PEX5-PEX14 protein-protein interaction (PPI) inhibitors based on an oxopiperazine template Marciniak, Monika; Mroz, Piotr; Napolitano, Valeria; Kalel, Vishal C.; Fino, Roberto; Pykacz, Emilia; Schliebs, Wolfgang; Plettenburg, Oliver; Erdmann, Ralf; Sattler, Michael; Popowicz, Grzegorz M.; Dawidowski, Maciej Share Save
Development of a peptide drug restoring AMPK and adipose tissue functionality in cancer cachexia Ji, Honglei; Englmaier, Felix; Morigny, Pauline; Giroud, Maude; Graesle, Pamina; Brings, Sebastian; Szendroedi, Julia; Diaz, Mauricio Berriel; Plettenburg, Oliver; Herzig, Stephan; Rohm, Maria Share Save
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Silmitasertib (CX-4945), a Clinically Used CK2-Kinase Inhibitor with Additional Effects on GSK3β and DYRK1A Kinases: A Structural Perspective Grygier, Przemyslaw; Pustelny, Katarzyna; Nowak, Jakub; Golik, Przemyslaw; Popowicz, Grzegorz M.; Plettenburg, Oliver; Dubin, Grzegorz; Menezes, Filipe; Czarna, Anna Share Save
The Myxobacterial Antibiotic Myxovalargin: Biosynthesis, Structural Revision, Total Synthesis, and Molecular Characterization of Ribosomal Inhibition Koller, Timm O.; Scheid, Ullrich; Koesel, Teresa; Herrmann, Jennifer; Krug, Daniel; Boshoff, Helena I. M.; Beckert, Bertrand; Evans, Joanna C.; Schlemmer, Jan; Sloan, Becky; Weiner, Danielle M.; Via, Laura E.; Moosa, Atica; Ioerger, Thomas R.; Graf, Michael; Zinshteyn, Boris; Abdelshahid, Maha; Nguyen, Fabian; Arenz, Stefan; Gille, Franziska; Siebke, Maik; Seedorf, Tim; Plettenburg, Oliver; Green, Rachel; Warnke, Anna-Luisa; Ullrich, Joachim; Warrass, Ralf; Barry, Clifton E., III; Warner, Digby F.; Mizrahi, Valerie; Kirschning, Andreas; Wilson, Daniel N.; Mueller, Rolf Share Save
Structure-based design, synthesis and evaluation of a novel family of PEX5-PEX14 interaction inhibitors against Trypanosoma Napolitano, Valeria; Mroz, Piotr; Marciniak, Monika; Kalel, Vishal C.; Softley, Charlotte A.; Olmos, Julian D. Janna; Tippler, Bettina G.; Schorpp, Kenji; Rioton, Sarah; Froehlich, Tony; Plettenburg, Oliver; Hadian, Kamyar; Erdmann, Ralf; Sattler, Michael; Popowicz, Grzegorz M.; Dawidowski, Maciej; Dubin, Grzegorz Share Save
Vps37a regulates hepatic glucose production by controlling glucagon receptor localization to endosomes(vol 34, pg1 2022) Sekar, Revathi; Motzler, Karsten; Kwon, Yun; Novikoff, Aaron; Juelg, Julia; Najafi, Bahar; Wang, Surui; Warnke, Anna-Luisa; Seitz, Susanne; Hass, Daniela; Gancheva, Sofiya; Kahl, Sabine; Yang, Bin; Finan, Brian; Schwarz, Kathrin; Okun, Juergen G.; Roden, Michael; Blueher, Matthias; Mueller, Timo D.; Krahmer, Natalie; Behrends, Christian; Plettenburg, Oliver; Miaczynska, Marta; Herzig, Stephan; Zeigerer, Anja Share Save
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Acriflavine, a clinically approved drug, inhibits SARS-CoV-2 and other betacoronaviruses Napolitano, Valeria; Dabrowska, Agnieszka; Schorpp, Kenji; Mourao, Andre; Barreto-Duran, Emilia; Benedyk, Malgorzata; Botwina, Pawel; Brandner, Stefanie; Bostock, Mark; Chykunova, Yuliya; Czarna, Anna; Dubin, Grzegorz; Froehlich, Tony; Hoelscher, Michael; Jedrysik, Malwina; Matsuda, Alex; Owczarek, Katarzyna; Pachota, Magdalena; Plettenburg, Oliver; Potempa, Jan; Rothenaigner, Ina; Schlauderer, Florian; Slysz, Klaudia; Szczepanski, Artur; Mohn, Kristin Greve-Isdahl; Blomberg, Bjorn; Sattler, Michael; Hadian, Kamyar; Popowicz, Grzegorz Maria; Pyrc, Krzysztof Share Save
A20 and ABIN-1 cooperate in balancing CBM complex-triggered NF-κB signaling in activated T cells Yin, Hongli; Karayel, Ozge; Chao, Ying-Yin; Seeholzer, Thomas; Hamp, Isabel; Plettenburg, Oliver; Gehring, Torben; Zielinski, Christina; Mann, Matthias; Krappmann, Daniel Share Save
Phenotypic drug screening in a human fibrosis model identified a novel class of antifibrotic therapeutics Gerckens, Michael; Schorpp, Kenji; Pelizza, Francesco; Woegrath, Melanie; Reichau, Kora; Ma, Huilong; Dworsky, Armando-Marco; Sengupta, Arunima; Stoleriu, Mircea Gabriel; Heinzelmann, Katharina; Merl-Pham, Juliane; Irmler, Martin; Alsafadi, Hani N.; Trenkenschuh, Eduard; Sarnova, Lenka; Jirouskova, Marketa; Friess, Wolfgang; Hauck, Stefanie M.; Beckers, Johannes; Kneidinger, Nikolaus; Behr, Juergen; Hilgendorff, Anne; Hadian, Kamyar; Lindner, Michael; Koenigshoff, Melanie; Eickelberg, Oliver; Gregor, Martin; Plettenburg, Oliver; Yildirim, Ali Oender; Burgstaller, Gerald Share Save
TRAF6 prevents fatal inflammation by homeostatic suppression of MALT1 protease O'Neill, Thomas J.; Seeholzer, Thomas; Gewies, Andreas; Gehring, Torben; Giesert, Florian; Hamp, Isabel; Grass, Carina; Schmidt, Henrik; Kriegsmann, Katharina; Tofaute, Marie J.; Demski, Katrin; Poth, Tanja; Rosenbaum, Marc; Schnalzger, Theresa; Ruland, Juergen; Goettlicher, Martin; Kriegsmann, Mark; Naumann, Ronald; Heissmeyer, Vigo; Plettenburg, Oliver; Wurst, Wolfgang; Krappmann, Daniel Share Save
Computer-Aided Design and Synthesis of a New Class of PEX14 Inhibitors: Substituted 2,3,4,5-Tetrahydrobenzo[F][1,4]oxazepines as Potential New Trypanocidal Agents Fino, Roberto; Lenhart, Dominik; Kalel, Vishal C.; Softley, Charlotte A.; Napolitano, Valeria; Byrne, Ryan; Schliebs, Wolfgang; Dawidowski, Maciej; Erdmann, Ralf; Sattler, Michael; Schneider, Gisbert; Plettenburg, Oliver; Popowicz, Grzegorz M. Share Save
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