Not logged in The Distinct Roles of CXCR3 Variants and Their Ligands in the Tumor Microenvironment Reynders, Nathan; Abboud, Dayana; Baragli, Alessandra; Noman, Muhammad Zaeem; Rogister, Bernard; Niclou, Simone P.; Heveker, Nikolaus; Janji, Bassam; Hanson, Julien; Szpakowska, Martyna; Chevigne, Andy Share Save
Biased antagonism of CXCR4 avoids antagonist tolerance Hitchinson, Ben; Eby, Jonathan M.; Gao, Xianlong; Guite-Vinet, Francois; Ziarek, Joshua J.; Abdelkarim, Hazem; Lee, Youngshim; Okamoto, Yukari; Shikano, Sojin; Majetschak, Matthias; Heveker, Nikolaus; Volkman, Brian F.; Tarasova, Nadya I.; Gaponenko, Vadim Share Save
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Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3) Sekiguchi, Haruka; Kuroyanagi, Tomoko; Rhainds, David; Kobayashi, Kazuya; Kobayashi, Yuka; Ohno, Hiroaki; Heveker, Nikolaus; Akaji, Kenichi; Fujii, Nobutaka; Oishi, Shinya Share Save
Different contributions of chemokine N-terminal features attest to a different ligand binding mode and a bias towards activation of ACKR3/CXCR7 compared with CXCR4 and CXCR3 Szpakowska, Martyna; Nevins, Amanda M.; Meyrath, Max; Rhainds, David; D'huys, Thomas; Guite-Vinet, Francois; Dupuis, Nadine; Gauthier, Pierre-Arnaud; Counson, Manuel; Kleist, Andrew; St-Onge, Genevieve; Hanson, Julien; Schols, Dominique; Volkman, Brian F.; Heveker, Nikolaus; Chevigne, Andy Share Save
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Structural basis for chemokine recognition by a G protein-coupled receptor and implications for receptor activation Ziarek, Joshua J.; Kleist, Andrew B.; London, Nir; Raveh, Barak; Montpas, Nicolas; Bonneterre, Julien; St-Onge, Genevieve; DiCosmo-Ponticello, Crystal J.; Koplinski, Chad A.; Roy, Ishan; Stephens, Bryan; Thelen, Sylvia; Veldkamp, Christopher T.; Coffman, Frederick D.; Cohen, Marion C.; Dwinell, Michael B.; Thelen, Marcus; Peterson, Francis C.; Heveker, Nikolaus; Volkman, Brian F. Share Save
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Structure-Activity Relationship and Signaling of New Chimeric CXCR4 Agonists Mona, Christine E.; Besserer-Offroy, Elie; Cabana, Jerome; Lefrancois, Marilou; Boulais, Philip E.; Lefebvre, Marie-Reine; Leduc, Richard; Lavigne, Pierre; Heveker, Nikolaus; Marsault, Eric; Escher, Emanuel Share Save
Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold Oishi, Shinya; Kuroyanagi, Tomoko; Kubo, Tatsuhiko; Montpas, Nicolas; Yoshikawa, Yasushi; Misu, Ryosuke; Kobayashi, Yuka; Ohno, Hiroaki; Heveker, Nikolaus; Furuya, Toshio; Fujii, Nobutaka Share Save
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Positive Regulation of Insulin Signaling by Neuraminidase 1 Dridi, Larbi; Seyrantepe, Volkan; Fougerat, Anne; Pan, Xuefang; Bonneil, Eric; Thibault, Pierre; Moreau, Allain; Mitchell, Grant A.; Heveker, Nikolaus; Cairo, Christopher W.; Issad, Tarik; Hinek, Alexander; Pshezhetsky, Alexey V. Share Save
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Direct assessment of CXCR4 mutant conformations reveals complex link between receptor structure and Gαi activation (vol 282, pg 5111, 2007) Berchiche, Yamina A.; Chow, Ken Y.; Lagane, Bernard; Leduc, Martin; Percherancier, Yann; Fujii, Nobutaka; Tamamura, Hirokazu; Bachelerie, Francoise; Heveker, Nikolaus Share Save
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