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Oleksandr Grytsai

centre national de la recherche scientifique (cnrs)

7H-index
31Paper Count
270Citation Count
Published Papers 7
Publication Date
Optimised arylbiamidine derivative as potent in vivo antimelanoma agent: Drug-to-target approach reveals nanomolar GSK3β inhibition
err2025-05-01
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errOAAI
errGrytsai, Oleksandr; Hamouda-Tekaya, Nedra; Goncalves, Leticia Christina Pires; Bardovskyi, Rostyslav; Abbe, Patricia; Benhida, Rachid; Rocchi, Stephane; Ronco, Cyril
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Discovery of novel series of PKMYT1 inhibitors forcombination therapy with antibody-drug conjugates
err2024-10-01
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PREAI
errMarais, R.; Grabarek, J.; Ioannou, M.; Leung, L.; Raoof, A.; Brown, M.; Smithen, D.; Fitzpatrick, C.; Chester, C.; Leigh, J.; Aljarah, M.; Lisauskaite, M.; Grytsai, O.; Burgin, R.; Niculescu-Duvaz, D.; Thomson, G.; Springer, C.
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A Potent Solution for Tumor Growth and Angiogenesis Suppression via an ELR+CXCL-CXCR1/2 Pathway Inhibitor
err2024-04-03
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PREAI
errGrytsai, Oleksandr; Dufies, Maeva; Le Du, Julie; Rastoin, Olivia; Goncalves, Leticia Christina Pires; Mateo, Lou; Lacas-Gervais, Sandra; Cao, Yihai; Demange, Luc; Pages, Gilles; Benhida, Rachid; Ronco, Cyril
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Design, Synthesis and Biological Evaluation of Novel Anticancer Amidinourea Analogues via Unexpected 1,3,5-Triazin-2-one Ring Opening
err2024-01-15
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errOAAI
errGrytsai, Oleksandr; Hamouda-Tekaya, Nedra; Botton, Thomas; Rocchi, Stephane; Benhida, Rachid; Ronco, Cyril
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Biguanides drugs: Past success stories and promising future for drug discovery
err2021-11-01
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errOAAI
errGrytsai, Oleksandr; Myrgorodska, Iuliia; Rocchi, Stephane; Ronco, Cyril; Benhida, Rachid
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Discovery of a new molecule inducing melanoma cell death: dual AMPK/MELK targeting for novel melanoma therapies
err2021-01-11
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errOAAI
errJaune, Emilie; Cavazza, Elisa; Ronco, Cyril; Grytsai, Oleksandr; Abbe, Patricia; Tekaya, Nedra; Zerhouni, Marwa; Beranger, Guillaume; Kaminski, Lisa; Bost, Frederic; Gesson, Maeva; Tulic, Meri; Hofman, Paul; Ballotti, Robert; Passeron, Thierry; Botton, Thomas; Benhida, Rachid; Rocchi, Stephane
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New CXCR1/CXCR2 inhibitors represent an effective treatment for kidney or head and neck cancers sensitive or refractory to reference treatments
err2019-01-01
err38
errOAAI
errDufies, Maeva; Grytsai, Oleksandr; Ronco, Cyril; Camara, Oumar; Ambrosetti, Damien; Hagege, Anais; Parola, Julien; Mateo, Lou; Ayrault, Marion; Giuliano, Sandy; Grepin, Renaud; Lagarde, Nathalie; Montes, Matthieu; Auberger, Patrick; Demange, Luc; Benhida, Rachid; Pages, Gilles
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