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Imidazole Bioisostere Activators of Endopeptidase Neurolysin with Enhanced Potency and Metabolic Stability Rahman, Md. Shafikur; Esfahani, Shiva Hadi; Zhang, Yong; Queen, Aarfa; Aljarrah, Manar; Kandil, Haya; Baez, Andrew; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C. Share Save
Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals Zhang, Yong; Sharma, Sejal; Jonnalagadda, Shirisha; Kumari, Shikha; Queen, Aarfa; Esfahani, Shiva Hadi; Archie, Sabrina Rahman; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J. Share Save
High brain-blood barrier permeability highlights a new class of neurolysin activators as promising candidates for stroke treatment: a pilot pharmacokinetic study in mice Zhang, Yong; Sharma, Sejal; Esfahani, Shiva H.; Jonnalagadda, Shirisha; Queen, Aarfa; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J. Share Save
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In-Vivo and Ex-Vivo Brain Uptake Studies of Peptidomimetic Neurolysin Activators in Healthy and Stroke Animals Nozohouri, Saeideh; Esfahani, Shiva Hadi; Noorani, Behnam; Patel, Dhaval; Villalba, Heidi; Ghanwatkar, Yashwardhan; Rahman, Md Shafikur; Zhang, Yong; Bickel, Ulrich; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J. Share Save
Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability (vol 64, pg 12705, 2021) Rahman, Md. Shafikur; Kumari, Shikha; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Jayaraman, Srinidhi; Kinarivala, Nihar; Kocot, Joanna; Baez, Andrew; Farris, Delaney; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C. Share Save
Identification and Characterization of Two Structurally Related Dipeptides that Enhance Catalytic Efficiency of Neurolysin Jayaraman, Srinidhi; Kocot, Joanna; Esfahani, Shiva Hadi; Wangler, Naomi J.; Uyar, Arzu; Mechref, Yehia; Trippier, Paul C.; Abbruscato, Thomas J.; Dickson, Alex; Aihara, Hideki; Ostrov, David A.; Karamyan, Vardan T. Share Save
Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability Rahman, Md Shafikur; Kumari, Shikha; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Jayaraman, Srinidhi; Kinarivala, Nihar; Kocot, Joanna; Baez, Andrew; Farris, Delaney; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C. Share Save