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Shiva Hadi Esfahani

Oakland University

6H-index
23Paper Count
77Citation Count
Published Papers 10
Publication Date
Discovery of a pyridine-piperazine-based small molecule that enhances the activity of peptidase neurolysin
err2026-02-03
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PREAI
errHeba ElSayed ElZorkany; Haya Kandil; Srinidhi Jayaraman; Asmaa Aly; Shiva Hadi Esfahani; Dhavalkumar Patel; Dennis Dannecker; Monika Maciag; Alyssa Paul; Kaitlin Lowran; Shikha Kumari; Samik Bose; David A. Ostrov; Colin G. Wu; Alex Dickson; Thomas J. Abbruscato; Paul C. Trippier; Benjamin J. Orlando; Vardan T. Karamyan
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Structural basis of divergent substrate recognition and inhibition of human neurolysin
err2024-08-08
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errOAAI
errShi, Ke; Bagchi, Sounak; Bickel, Jordis; Esfahani, Shiva H.; Yin, Lulu; Cheng, Tiffany; Karamyan, Vardan T.; Aihara, Hideki
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Imidazole Bioisostere Activators of Endopeptidase Neurolysin with Enhanced Potency and Metabolic Stability
err2024-03-29
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PREAI
errRahman, Md. Shafikur; Esfahani, Shiva Hadi; Zhang, Yong; Queen, Aarfa; Aljarrah, Manar; Kandil, Haya; Baez, Andrew; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals
err2023-10-13
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PREAI
errZhang, Yong; Sharma, Sejal; Jonnalagadda, Shirisha; Kumari, Shikha; Queen, Aarfa; Esfahani, Shiva Hadi; Archie, Sabrina Rahman; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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High brain-blood barrier permeability highlights a new class of neurolysin activators as promising candidates for stroke treatment: a pilot pharmacokinetic study in mice
err2023-06-01
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errOAAI
errZhang, Yong; Sharma, Sejal; Esfahani, Shiva H.; Jonnalagadda, Shirisha; Queen, Aarfa; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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In-Vivo and Ex-Vivo Brain Uptake Studies of Peptidomimetic Neurolysin Activators in Healthy and Stroke Animals
err2022-03-03
err9
errOAAI
errNozohouri, Saeideh; Esfahani, Shiva Hadi; Noorani, Behnam; Patel, Dhaval; Villalba, Heidi; Ghanwatkar, Yashwardhan; Rahman, Md Shafikur; Zhang, Yong; Bickel, Ulrich; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability (vol 64, pg 12705, 2021)
err2021-12-22
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errOAAI
errRahman, Md. Shafikur; Kumari, Shikha; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Jayaraman, Srinidhi; Kinarivala, Nihar; Kocot, Joanna; Baez, Andrew; Farris, Delaney; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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Identification and Characterization of Two Structurally Related Dipeptides that Enhance Catalytic Efficiency of Neurolysin
err2021-11-01
err10
errOAAI
errJayaraman, Srinidhi; Kocot, Joanna; Esfahani, Shiva Hadi; Wangler, Naomi J.; Uyar, Arzu; Mechref, Yehia; Trippier, Paul C.; Abbruscato, Thomas J.; Dickson, Alex; Aihara, Hideki; Ostrov, David A.; Karamyan, Vardan T.
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Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability
err2021-08-26
err11
errOAAI
errRahman, Md Shafikur; Kumari, Shikha; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Jayaraman, Srinidhi; Kinarivala, Nihar; Kocot, Joanna; Baez, Andrew; Farris, Delaney; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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