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Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes Ogasawara, Daisuke; Konrad, David B.; Tan, Zher Yin; Carey, Kimberly L.; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever R.; DeMeester, Kristen E.; Njomen, Evert; Schreiber, Stuart L.; Xavier, Ramnik J.; Melillo, Bruno; Cravatt, Benjamin F. Share Save
Redirecting the pioneering function of FOXA1 with covalent small molecules Won, Sang Joon; Zhang, Yuxiang; Reinhardt, Christopher J.; Hargis, Lauren M.; MacRae, Nicole S.; DeMeester, Kristen E.; Njomen, Evert; Remsberg, Jarrett R.; Melillo, Bruno; Cravatt, Benjamin F.; Erb, Michael A. Share Save
Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders Liu, Zhonglin; Remsberg, Jarrett R.; Li, Haoxin; Njomen, Evert; Demeester, Kristen E.; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E.; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M.; Schreiber, Stuart L.; Melillo, Bruno; Cravatt, Benjamin F. Share Save
Covalent Targeting As a Common Mechanism for Inhibiting NLRP3 Inflammasome Assembly Stanton, Caroline; Sun, Jie; Nutsch, Kayla; Rosarda, Jessica D.; Nguyen, Thu; Li-Ma, Chloris; Njomen, Evert; Melillo, Bruno; Kutseikin, Sergei; Saez, Enrique; Cravatt, Benjamin F.; Teijaro, John R.; Wiseman, R. Luke; Bollong, Michael J. Share Save
Proteomic discovery of chemical probes that perturb protein complexes in human cells Lazear, Michael R.; Remsberg, Jarrett R.; Jaeger, Martin G.; Rothamel, Katherine; Her, Hsuan-lin; DeMeester, Kristen E.; Njomen, Evert; Hogg, Simon J.; Rahman, Jahan; Whitby, Landon R.; Won, Sang Joon; Schafroth, Michael A.; Ogasawara, Daisuke; Yokoyama, Minoru; Lindsey, Garrett L.; Li, Haoxin; Germain, Jason; Barbas, Sabrina; Vaughan, Joan; Hanigan, Thomas W.; Vartabedian, Vincent F.; Reinhardt, Christopher J.; Dix, Melissa M.; Koo, Seong Joo; Heo, Inha; Teijaro, John R.; Simon, Gabriel M.; Ghosh, Brahma; Abdel-Wahab, Omar; Ahn, Kay; Saghatelian, Alan; Melillo, Bruno; Schreiber, Stuart L.; Yeo, Gene W.; Cravatt, Benjamin F. Share Save
Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain Feldman, Hannah C.; Merlini, Elisa; Guijas, Carlos; DeMeester, Kristen E.; Njomen, Evert; Kozina, Ellen M.; Yokoyama, Minoru; Vinogradova, Ekaterina; Reardon, Holly T.; Melillo, Bruno; Schreiber, Stuart L.; Loreto, Andrea; Blankman, Jacqueline L.; Cravatt, Benjamin F. Share Save