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Benjamin F. Cravatt

scripps research

148H-index
866Paper Count
8.1WCitation Count
Published Papers 419
Publication Date
A fatty acid amide activates myeloid cells and improves neurovascular outcomes in retinal degeneration
err2026-06-19
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errGuoqin Wei; Shreyosree Chatterjee; Qinglin Yang; Sanahan Vijayakumar; Daisuke Ogasawara; Sarah Giles; Katie Biscocho; Peter Westenskow; Junhua Wang; Ruhan Fan; Helena Pham; Edith Aguilar; Jacob Robinson; Ayumi Usui-Ouchi; Roberto Bonelli; Kevin Eade; Gary Siuzdak; Benjamin Cravatt; Michael J. Sailor; Dale Boger; Martin Friedlander
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Genetic and pharmacological inactivation of peptidoglycan remodeling increases antibiotic susceptibility of vancomycin-resistant Enterococcus faecium
err2026-06-16
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errOAAI
errKyong T. Fam; Pavan Kumar Chodisetti; Zifei Wang; Joshua A. Homer; Christopher J. Smedley; Seiya Kitamura; Benjamin Silva; Yijun Xiong; Althea Hansel-Harris; Matthew Holcomb; Simeon Babarinde; Adrianna M. Turner; Daria Van Tyne; Ian A. Wilson; Stefano Forli; Benjamin F. Cravatt; Donghyun Park; Dennis W. Wolan; John E. Moses; Howard C. Hang
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A Global Ligandability Map of Tryptoline Butynamide Stereoprobes Identifies Covalent Inhibitors of the Actin Maturation Protease
err2026-05-20
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PREAI
errYijun Xiong; Christopher J. Reinhardt; Tracey Nguyen; Melissa A. Hoffman; Gabriel M. Simon; Bruno Melillo; Benjamin F. Cravatt
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High-throughput ligand diversification to discover chemical inducers of proximity
err2026-02-16
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errJames B. Shaum; Miquel Muñoz i Ordoño; Erica A. Steen; Daniela V. Wenge; Hakyung Cheong; Jordan Janowski; Moritz Hunkeler; Eric M. Bilotta; Zoe J. Rutter; Paige A. Barta; Abby M. Thornhill; Natalia Milosevich; Lauren M. Hargis; Timothy R. Bishop; Trever R. Carter; Bryce da Camara; Matthias Hinterndorfer; Lucas Dada; Wen-Ji He; Fabian Offensperger; Hirotake Furihata; Sydney R. Schweber; Charlie Hatton; Yanhe Wen; Benjamin F. Cravatt; Keary M. Engle; Katherine A. Donovan; Bruno Melillo; Seiya Kitamura; Alessio Ciulli; Scott A. Armstrong; Eric S. Fischer; Georg E. Winter; Michael A. Erb
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Cysteine Reactivity Profiling Identifies Host Regulators of Mycobacterium tuberculosis Replication in Human Macrophages
err2026-01-27
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PREAI
errJohn K. Neff; Kristen E. DeMeester; Paola K. Párraga Solórzano; Radu M. Suciu; Melissa M. Dix; Gabriel Simon; Max A. Gianakopoulos; Bruno Melillo; Benjamin F. Cravatt; Michael U. Shiloh
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Ophiobolin A impacts mitochondrial redox biology in an epithelial-mesenchymal transition (EMT)-specific manner
err2026-01-14
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errHaleigh N. Parker; Yongfeng Tao; Jenna Tobin; Kayla L. Haberman; Samantha Davis; Emily York; Alysia Martinez; Nobuyuki Matsumoto; Jaquelin Aroujo; Jun Hyoung Park; Bernd Zechmann; Benny Abraham Kaipparettu; Angela Boari; Christie M. Sayes; Antonio Evidente; Alexander Kornienko; Benjamin Cravatt; Daniel Romo; Joseph H. Taube
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Structural and mechanistic analysis of covalent ligands targeting the RNA-binding protein NONO
err2026-01-13
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errGarrett L. Lindsey; Thomas K. Hockley; Alejandro Villa Gomez; Andrew C. Marshall; William R. Brothers; Colin T. Finney; Jacob Gross; Archa H. Fox; Gene W. Yeo; Bruno Melillo; Charles S. Bond; Benjamin F. Cravatt
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Complexoform-restricted covalent TRMT112 ligands that allosterically agonize METTL5
err2026-01-08
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errF. Wieland Goetzke; Steffen M. Bernard; Cheng-Wei Ju; Jonathan Pollock; Kristen E. DeMeester; Jacob Gross; Gabriel M. Simon; Chuan He; Bruno Melillo; Benjamin F. Cravatt
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Pharmacological targeting of the JAK–STAT pathway: new concepts and emerging indications
err2026-01-05
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PREAI
errTeemu Haikarainen; Anniina T. Virtanen; Benjamin F. Cravatt; Olli Silvennoinen
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Mitochondrial ABHD11 inhibition drives sterol metabolism to modulate T-cell effector function
err2025-11-03
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errBenjamin J. Jenkins; Yasmin R. Jenkins; Fernando M. Ponce-Garcia; Chloe Moscrop; Iain A. Perry; Matthew D. Hitchings; Alejandro H. Uribe; Federico Bernuzzi; Simon Eastham; James G. Cronin; Ardena Berisha; Alexandra Howell; Joanne Davies; Julianna Blagih; Marta Williams; Morgan Marsden; Douglas J. Veale; Luke C. Davies; Micah Niphakis; David K. Finlay; Linda V. Sinclair; Benjamin F. Cravatt; Andrew E. Hogan; James A. Nathan; Ian R. Humphreys; Ursula Fearon; David Sumpton; Johan Vande Voorde; Goncalo Dias do Vale; Jeffrey G. McDonald; Gareth W. Jones; James A. Pearson; Emma E. Vincent; Nicholas Jones
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A chemical-genetic interaction between PAF1 and ENL/AF9 YEATS inhibition
err2025-10-24
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errPaige A. Barta; Leopold Garnar-Wortzel; Timothy R. Bishop; Rachel E. Hayward; Lauren M. Hargis; James B. Shaum; Hui Si Kwok; Brian B. Liau; Benjamin F. Cravatt; Michael A. Erb
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NONO Maintains SREBP-Regulated Cholesterol Biosynthesis via RNA Binding in Neuroblastoma
err2025-09-16
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errSong Zhang; Hayley Ingram; Jack Cooper; Alina Naveed; Stefan G. Kathman; Garrett L. Lindsey; Tao Liu; Charles S. Bond; Jamie I. Fletcher; Benjamin F. Cravatt; Archa H. Fox
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Scalable total synthesis of saxitoxin and related natural products
errNature
IF48.5
err2025-08-26
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PREAI
errYinliang Guo; Yiheng Li; Sihan Chen; Yige Wu; Oscar Poll; Zhouyang Ren; Zhonglin Liu; Roman Vlkolinsky; Michal Bajo; Christopher K. Prier; Kai-Jiong Xiao; Benjamin F. Cravatt; Marisa Roberto; Phil S. Baran
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Cysteine allostery and autoinhibition govern human STING oligomer functionality
err2025-07-03
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errRebecca Chan; Xujun Cao; Sabrina L. Ergun; Evert Njomen; Stephen R. Lynch; Christopher Ritchie; Benjamin Cravatt; Lingyin Li
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Dietary control of peripheral adipose storage capacity through membrane lipid remodelling
err2025-06-27
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PREAI
errMarcus J. Tol; Yuta Shimanaka; Alexander H. Bedard; Jennifer Sapia; Liujuan Cui; Mariana Colaço-Gaspar; Peter Hofer; Alessandra Ferrari; Kevin Qian; John P. Kennelly; Stephen D. Lee; Yajing Gao; Xu Xiao; Jie Gao; Julia J. Mack; Thomas A. Weston; Kevin J. Williams; Baolong Su; Calvin Pan; Aldons J. Lusis; Daniel P. Pike; Alex Reed; Natalia Milosevich; Benjamin F. Cravatt; Makoto Arita; Stephen G. Young; David A. Ford; Rudolf Zechner; Stefano Vanni; Peter Tontonoz
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Development of a novel 18F-labeled reversible-binding radioligand for imaging monoacylglycerol lipase with positron emission tomography
err2025-06-03
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errJian Rong; Chunyu Zhao; Ahmad F. Chaudhary; Tim Ware; Richard S. Van; Yinlong Li; Erick R. Calderon Leon; Vivi Dang; Jiahui Chen; Zhiwei Xiao; Xin Zhou; Wei Zhang; Chunyang Bi; Kuo Zhang; Jimmy S. Patel; Yihan Shao; Chongzhao Ran; Ludovic Collin; Achi Haider; Benjamin F. Cravatt
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Radiosynthesis and evaluation of novel 18F labeled PET ligands for imaging monoacylglycerol lipase
err2025-03-01
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PREAI
errLi, Yinlong; Mori, Wakana; Chaudhary, Ahmad; Zhao, Chunyu; Yamasaki, Tomoteru; Zhang, Zachary; Feng, Siyan; Ware, Tim; Rong, Jian; Fujinaga, Masayuki; Chen, Jiahui; Kumata, Katsushi; Zhang, Yiding; Hu, Kuan; Xie, Lin; Zhou, Xin; Song, Zhendong; Gao, Yabiao; Sun, Zhenkun; Patel, Jimmy S.; Zhai, Chuangyan; Yuan, Katherine Y.; Collier, Thomas L.; Ran, Chongzhao; Collin, Ludovic; Haider, Achi; Grether, Uwe; Wittwer, Matthias B.; Cravatt, Benjamin F.; Zhang, Ming-Rong; Liang, Steven H.
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SF3B1 thermostability as an assay for splicing inhibitor interactions
err2025-02-01
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errAmorello, Angela N.; Reddy, Guddeti Chandrashekar; Melillo, Bruno; Cravatt, Benjamin F.; Ghosh, Arun K.; Jurica, Melissa S.
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Chemical probes for the identification of the molecular targets of honokiol
err2025-02-01
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errVazquez-Villa, Henar; Rueda-Zubiaurre, Ainoa; Fernandez, Daniel; Foronda, Roman; Parker, Christopher G.; Cravatt, Benjamin F.; Martin-Fontecha, Mar; Ortega-Gutierrez, Silvia
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Covalent targeting of splicing in T cells
err2025-01-01
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PREAI
errScott, Kevin A.; Kojima, Hiroyuki; Ropek, Nathalie; Warren, Charles D.; Zhang, Tiffany L.; Hogg, Simon J.; Sanford, Henry; Webster, Caroline; Zhang, Xiaoyu; Rahman, Jahan; Melillo, Bruno; Cravatt, Benjamin F.; Lyu, Jiankun; Abdel-Wahab, Omar; Vinogradova, Ekaterina V.
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