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Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors Kuijer, Michael Bram; Fulton, Camryn J.; Albert, Talia L.; Knobloch, Paloma; Wang, Jing; Krumm, Brian E.; Che, Tao; Varga, Balazs R.; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H.; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L. Share Save
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Exceptionally Potent Chiral Anandamide Analogs Georgiadis, Markos-Orestis; Ferreras, Elena; Ji, Lipin; Ferreira, Luana Assis; Hainline, John; Tong, Fei; Dang, Vuong Q.; Faragher, Alexandra; Sadybekov, Anastasiia V.; Bohn, Laura M.; Katritch, Vsevolod; Hohmann, Andrea G.; Makriyannis, Alexandros; Nikas, Spyros P. Share Save
ANGIOTENSIN-(1-5) IS A BIOLOGICALLY ACTIVE HORMONE OF THE RENIN-ANGIOTENSIN SYSTEM AND A POTENT AT2-RECEPTOR AGONIST Souza-Silva, Igor M.; Peluso, A. Augusto; Elsaafien, Khalid; Nazarova, Antonina L.; Assersen, Kasper B.; Rodrigues-Ribeiro, Lucas; Rodrigues, Andre F.; Enggaard, Camilla; Nawrocki, Arkadiusz; Jacobsen, Lene A.; Jensen, Pia; de Kloet, Annette D.; Krause, Eric G.; Bader, Michael; Jensen, Boye L.; Larsen, Martin; Verano-Braga, Thiago; Katritch, Vsevolod; Sumners, Colin; Steckelings, Ulrike Muscha Share Save
Structure-guided design of partial agonists at an opioid receptor Varga, Balazs R.; Bernhard, Sarah M.; El Daibani, Amal; Zaidi, Saheem A.; Lam, Jordy H.; Aguilar, Jhoan; Appourchaux, Kevin; Nazarova, Antonina L.; Kouvelis, Alexa; Shinouchi, Ryosuke; Hammond, Haylee R.; Eans, Shainnel O.; Weinreb, Violetta; Margolis, Elyssa B.; Fay, Jonathan F.; Huang, Xi-Ping; Pradhan, Amynah; Katritch, Vsevolod; Mclaughlin, Jay P.; Majumdar, Susruta; Che, Tao Share Save
Modulation of Kappa Opioid Receptor Functional Selectivity, Efficacy and Subtype Selectivity Ramos-Gonzalez, Nokomis; Varga, Balazs R.; Knoll, Alexis; Appourchaux, Kevin; Rangari, Vipin; Bernhard, Sarah; Nazarova, Antonina; Zaidi, Saheem A.; Katritch, Vsevolod; Che, Tao; Majumdar, Susruta Share Save
Structural insights into the high basal activity and inverse agonism of the orphan receptor GPR6 implicated in Parkinson's disease Barekatain, Mahta; Johansson, Linda C.; Lam, Jordy H.; Chang, Hao; Sadybekov, Anastasiia V.; Han, Gye Won; Russo, Joseph; Bliesath, Joshua; Brice, Nicola L.; Carlton, Mark B. L.; Saikatendu, Kumar S.; Sun, Hukai; Murphy, Sean T.; Monenschein, Holger; Schiffer, Hans H.; Popov, Petr; Lutomski, Corinne A.; Robinson, Carol V.; Liu, Zhi-Jie; Hua, Tian; Katritch, Vsevolod; Cherezov, Vadim Share Save
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Oxa-Iboga alkaloids lack cardiac risk and disrupt opioid use in animal models Havel, Vaclav; Kruegel, Andrew C.; Bechand, Benjamin; Mcintosh, Scot; Stallings, Leia; Hodges, Alana; Wulf, Madalee G.; Nelson, Mel; Hunkele, Amanda; Ansonoff, Michael; Pintar, John E.; Hwu, Christopher; Ople, Rohini S.; Abi-Gerges, Najah; Zaidi, Saheem A.; Katritch, Vsevolod; Yang, Mu; Javitch, Jonathan A.; Majumdar, Susruta; Hemby, Scott E.; Sames, Dalibor Share Save
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Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2 Nikas, Spyros P.; Ji, Lipin; Liu, Yingpeng; Georgiadis, Markos-Orestis; Dopeshwarkar, Amey; Straiker, Alex; Kudalkar, Shalley; Sadybekov, Anastasiia V.; Dvorakova, Michaela; Katritch, Vsevolod; Mackie, Ken; Marnett, Lawrence; Makriyannis, Alexandros Share Save
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Virtual Screening of a Chemically Diverse Superscaffold Library Enables Ligand Discovery for a Key GPCR Target Grotsch, Katharina; Sadybekov, Anastasiia V.; Hiller, Sydney; Zaidi, Saheem; Eremin, Dmitry; Le, Austen; Liu, Yongfeng; Smith, Evan Carlton; Illiopoulis-Tsoutsouvas, Christos; Thomas, Joice; Aggarwal, Shubhangi; Pickett, Julie E.; Reyes, Cesar; Picazo, Elias; Roth, Bryan L.; Makriyannis, Alexandros; Katritch, Vsevolod; Fokin, Valery V. Share Save
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Constitutive activation mechanism of a class C GPCR Shin, Jinwoo; Park, Junhyeon; Jeong, Jieun; Lam, Jordy Homing; Qiu, Xingyu; Wu, Di; Kim, Kuglae; Lee, Joo-Youn; Robinson, Carol V.; Hyun, Jaekyung; Katritch, Vsevolod; Kim, Kwang Pyo; Cho, Yunje Share Save
Pharmacological and Physicochemical Properties Optimization for Dual-Target Dopamine D3 (D3R) and μ-Opioid (MOR) Receptor Ligands as Potentially Safer Analgesics Bonifazi, Alessandro; Saab, Elizabeth; Sanchez, Julie; Nazarova, Antonina L.; Zaidi, Saheem A.; Jahan, Khorshada; Katritch, Vsevolod; Canals, Meritxell; Lane, J. Robert; Newman, Amy Hauck Share Save
Structure, Function, and Pharmacology of Delta Opioid Receptor Bitopics Bernhard, Sarah; Varga, Balazs R.; El Daibani, Amal; Lam, Jordy H.; Zaidi, Saheem; Appourchaux, Kevin; Eans, Shainnel; Katritch, Vsevolod; McLaughlin, Jay; Majumdar, Susruta; Che, Tao Share Save
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