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SaveAlbumin nanocomplex of BCL-2/xL inhibitor reduced platelet toxicity and improved anticancer efficacy in myeloproliferative neoplasm and lymphoma
Hu, Hongxiang; Li, Chengyi; Song, Yudong; Xie, Jizhao; Li, Qiuxia; Ke, Fang; Wen, Bo; Wang, Shaomeng; Gao, Wei; Sun, Duxin
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SaveDesign of Potent Small-Molecule Stimulator of Interferon Gene Inhibitor and Stimulator of Interferon Gene Mutant-Specific Degrader
Zhao, Hong-Yi; Zhang, Luchen; Liu, Zhongwei; He, Miao; Wang, Meilin; Li, Qiuxia; Sarkari, Farzad; Tao, Jinsong; Wen, Bo; Basrur, Venkatesha; Myatt, Hannah; Nesvizhskii, Alexey; Sun, Duxin
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SaveSARS-CoV-2 B Epitope-Guided Neoantigen NanoVaccines Enhance Tumor-Specific CD4/CD8 T Cell Immunity through B Cell Antigen Presentation
Li, CY; Ke, F; Mao, S; Montemayor, Z; Traore, MDM; Balsa, AD; Djibo, M; Karekar, N; Hu, HX; Wen, HN; Gao, W; Sun, DX
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SaveStructure-Based Development of Novel Spiro-Piperidine ASH1L Inhibitors
Huang, Guang; Stevens, Rhiannon; Hucek, Devon G.; Purohit, Trupta; Li, Shuangjiang; Miao, Hongzhi; Trost, Elise; Hewett, Geoff; Clegg, Bradley; Park, Se Ra; Rajanayake, Krishani; Wen, Bo; Sun, Duxin; Cierpicki, Tomasz; Grembecka, Jolanta
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SaveDiscovery of ERD-12310A as an Exceptionally Potent and Orally Efficacious PROTAC Degrader of Estrogen Receptor α (ERα)
Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Acharyya, Ranjan Kumar; Wu, Dimin; Metwally, Hoda; Mceachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Nishimura, Leticia S.; Gersch, Christina L.; Wang, Meilin; Wen, Bo; Sun, Duxin; Carlson, Kathryn; Katzenellenbogen, John A.; Xu, Guozhang; Zhang, Weihong; Wu, Wenxue; Priestley, E. Scott; Sui, Zhihua; Rae, James M.; Wang, Shaomeng
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SaveDiscovery of SD-436: A Potent, Highly Selective and Efficacious STAT3 PROTAC Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression
Xu, Renqi; Zhou, Haibin; Bai, Longchuan; McEachern, Donna; Wu, Dimin; Acharyya, Ranjan Kumar; Wang, Mi; Tosovic, Jelena; Yang, Chao-Yie; Chinnaswamy, Krishnapriya; Meagher, Jennifer L.; Stuckey, Jeanne A.; Liu, Cai; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng
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SaveDiscovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER plus Human Breast Cancer
Acharyya, Ranjan Kumar; Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Wu, Dimin; Lu, Jianfeng; Metwally, Hoda; Mceachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Tosovic, Jelena; Gersch, Christina L.; Xu, Guozhang; Zhang, Weihong; Wu, Wenxue; Priestley, E. Scott; Sui, Zhihua; Sarkari, Farzad; Wen, Bo; Sun, Duxin; Rae, James M.; Wang, Shaomeng
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