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Alexander Dömlingꝉ

Palacky University Olomouc

66H-index
583Paper Count
2.8WCitation Count
Published Papers 180
Publication Date
Ugi-Tetrazole-Derived α-Aminomethyl Scaffolds Reveal Unexpected Binding Modes in SARS-CoV-2 3CLpro
err2026-03-04
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errRobin van der Straat; Rick Oerlemans; Yingying Cong; Jeffrey Boxma; Radu G. Bulai; Clàudia Río-Bergé; Lizbé Koekemoer; Tryfon Zarganes Tzitzikas; Zhirui Guan; Peter George Marples; Fulvio Reggiori; Matthew Groves; Alexander Dömling
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Disruption of NLRP3 inflammasome assembly via ligand-induced remodeling of pyrin domain interfaces
err2026-01-09
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errSara Khosravifard; Saman Hosseinkhani; Nuredin Bakhtiary; Maryam Peyvandi; Alexander S. S. Dömling
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Nanoparticle-Mediated Delivery of Adenosine 5′-Monophosphate Enhances 5-Oxoprolinase Activity to Mitigate Oxidative Stress in Heart Failure
err2026-01-01
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errEsquivel-Gaytan, Antonio; Bomer, Nils; Bartolo, Raquel; Arevalo-Gomez, Karla F.; Deiman, Frederik E.; Bras, Maaike; Honarnejad, Saman; Permentier, Hjalmar; Domling, Alexander; Voors, Adriaan A.; Santos, Helder A.; Sillje, Herman H. W.; Van Der Meer, Peter
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Precipitation-first Synthesis and Deep Profiling of a 1; 200-Member Acrylamide Library for Covalent Drug Discovery
err2025-10-23
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errPravin Patil; Emis Ingenito; Riccardo Fusco; Imma Capriello; Zhirui Guan; Anuja Bhalkikar; John Gibbons; Tomas Korba; Stanislav Bashkyrtsev; Oleh Tkachenko; Alexander Dömling
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Balinatunfib: A Clinical Oral Small Molecule TNFα Inhibitor
err2025-06-19
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errAlexander Dömling; Tad A. Holak
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Expert opinion on therapeutic patents - manuscript ID EOTP-2024-ST-0024 has been submitted online
err2024-11-25
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errFusco, Riccardo; Saedi, Zeinab; Capriello, Imma; Lubskyy, Andriy; Domling, Alexander
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Computer- and NMR-Aided Design of Small-Molecule Inhibitors of the Hub1 Protein (vol 27, 8282, 2022)
err2024-06-20
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errRomero, Atilio Reyes; Kubica, Katarzyna; Kitel, Radoslaw; Rodriguez, Ismael; Magiera-Mularz, Katarzyna; Domling, Alexander; Holak, Tad A.; Surmiak, Ewa
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C2-Symmetrical Terphenyl Derivatives as Small Molecule Inhibitors of Programmed Cell Death 1/Programmed Death Ligand 1 Protein-Protein Interaction
err2024-06-04
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errKlimek, Joanna; Kruc, Oskar; Ceklarz, Joanna; Kaminska, Beata; Musielak, Bogdan; van der Straat, Robin; Domling, Alexander; Holak, Tad A.; Muszak, Damian; Kalinowska-Tluscik, Justyna; Skalniak, Lukasz; Surmiak, Ewa
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Joint Effects of Exercise and Ramadan Fasting on Telomere Length: Implications for Cellular Aging
err2024-05-27
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errAlmuraikhy, Shamma; Sellami, Maha; Naja, Khaled; Al-Amri, Hadaia Saleh; Anwardeen, Najeha; Aden, Amina; Domling, Alexander; Elrayess, Mohamed A.
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Novel FOXM1 inhibitor STL001 sensitizes human cancers to a broad-spectrum of cancer therapies
err2024-05-02
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errRaghuwanshi, Sanjeev; Zhang, Xu; Arbieva, Zarema; Khan, Irum; Mohammed, Hisham; Wang, Z.; Domling, Alexander; Camacho, Carlos Jaime; Gartel, Andrei L.
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Novel SK channel positive modulators prevent ferroptosis and excitotoxicity in neuronal cells
err2024-02-01
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errZhang, Yuequ; Shaabani, Shabnam; Vowinkel, Kirsty; Trombetta-Lima, Marina; Sabogal-Guaqueta, Angelica Maria; Chen, Tingting; Hoekstra, Jan; Lembeck, Jan; Schmidt, Martina; Decher, Niels; Doemling, Alexander; Dolga, Amalia M.
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Exploring Phthalimide as the Acid Component in the Passerini Reaction
err2024-01-16
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errLi, Jingyao; Zheng, Qiang; Domling, Alexander
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Crystal Clear: Decoding Isocyanide Intermolecular Interactions through Crystallography
err2024-01-04
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errChatziorfanou, Eleftheria; Romero, Atilio Reyes; Chouchane, Lotfi; Domling, Alexander
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1,5-Disubstituted tetrazoles as PD-1/PD-L1 antagonists
err2024-01-01
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errvan der Straat, Robin; Draijer, Rosalie; Surmiak, Ewa; Butera, Roberto; Land, Lennart; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Plewka, Jacek; Holak, Tad A.; Domling, Alexander
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Direct-to-biology, automated, nano-scale synthesis, and phenotypic screening-enabled E3 ligase modulator discovery
err2023-12-19
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errWang, Zefeng; Shaabani, Shabnam; Gao, Xiang; Ng, Yuen Lam Dora; Sapozhnikova, Valeriia; Mertins, Philipp; Kroenke, Jan; Doemling, Alexander
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Impact of Moderate Physical Activity on Inflammatory Markers and Telomere Length in Sedentary and Moderately Active Individuals with Varied Insulin Sensitivity
err2023-11-01
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errAlmuraikhy, Shamma; Sellami, Maha; Al-Amri, Hadaia Saleh; Domling, Alexander; Althani, Asmaa A.; Elrayess, Mohamed A.
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The isocyanide SN2 reaction
err2023-09-19
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errPatil, Pravin; Zheng, Qiang; Kurpiewska, Katarzyna; Domling, Alexander
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Antioxidative Stress Metabolic Pathways in Moderately Active Individuals
err2023-08-27
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errAlmuraikhy, Shamma; Anwardeen, Najeha; Doudin, Asmma; Sellami, Maha; Domling, Alexander; Agouni, Abdelali; Althani, Asmaa A.; Elrayess, Mohamed A.
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Favorable outcomes of NPM1mut AML patients are due to transcriptional inactivation of FOXM1, presenting a new target to overcome chemoresistance
err2023-08-22
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errKhan, I.; Kaempf, A.; Raghuwanshi, S.; Chesnokov, M.; Zhang, X.; Wang, Z.; Domling, A.; Tyner, J. W.; Camacho, C.; Gartel, A. L.
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